DK129844B - Analogifremgangsmåde til fremstilling af thieno[3,2-d]pyrimidiner. - Google Patents

Analogifremgangsmåde til fremstilling af thieno[3,2-d]pyrimidiner.

Info

Publication number
DK129844B
DK129844B DK219672AA DK219672A DK129844B DK 129844 B DK129844 B DK 129844B DK 219672A A DK219672A A DK 219672AA DK 219672 A DK219672 A DK 219672A DK 129844 B DK129844 B DK 129844B
Authority
DK
Denmark
Prior art keywords
thieno
pyrimidines
preparation
analogous process
analogous
Prior art date
Application number
DK219672AA
Other languages
Danish (da)
English (en)
Other versions
DK129844C (cg-RX-API-DMAC7.html
Inventor
B Narr
J Roch
E Mueller
J Nickl
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19712121950 external-priority patent/DE2121950A1/de
Priority claimed from DE19712137341 external-priority patent/DE2137341A1/de
Priority claimed from DE19722215299 external-priority patent/DE2215299A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DK129844B publication Critical patent/DK129844B/da
Application granted granted Critical
Publication of DK129844C publication Critical patent/DK129844C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DK219672AA 1971-05-04 1972-05-03 Analogifremgangsmåde til fremstilling af thieno[3,2-d]pyrimidiner. DK129844B (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19712121950 DE2121950A1 (en) 1971-05-04 1971-05-04 Thieno(3,2-d)pyrimidine derivs - with thrombocyte aggregation inhibiting activity
DE19712137341 DE2137341A1 (de) 1971-07-26 1971-07-26 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine
DE19722215299 DE2215299A1 (de) 1972-03-29 1972-03-29 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine

Publications (2)

Publication Number Publication Date
DK129844B true DK129844B (da) 1974-11-25
DK129844C DK129844C (cg-RX-API-DMAC7.html) 1975-05-12

Family

ID=27183398

Family Applications (1)

Application Number Title Priority Date Filing Date
DK219672AA DK129844B (da) 1971-05-04 1972-05-03 Analogifremgangsmåde til fremstilling af thieno[3,2-d]pyrimidiner.

Country Status (15)

Country Link
US (1) US3888851A (cg-RX-API-DMAC7.html)
AT (1) AT318619B (cg-RX-API-DMAC7.html)
AU (1) AU4181572A (cg-RX-API-DMAC7.html)
BE (1) BE783044A (cg-RX-API-DMAC7.html)
BG (1) BG20593A3 (cg-RX-API-DMAC7.html)
DD (1) DD97656A5 (cg-RX-API-DMAC7.html)
DK (1) DK129844B (cg-RX-API-DMAC7.html)
ES (1) ES402302A1 (cg-RX-API-DMAC7.html)
FR (1) FR2135294B1 (cg-RX-API-DMAC7.html)
GB (1) GB1393161A (cg-RX-API-DMAC7.html)
HU (1) HU163960B (cg-RX-API-DMAC7.html)
IL (1) IL39341A (cg-RX-API-DMAC7.html)
NL (1) NL7206041A (cg-RX-API-DMAC7.html)
PL (1) PL82381B1 (cg-RX-API-DMAC7.html)
RO (1) RO62428A (cg-RX-API-DMAC7.html)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
US5098902A (en) * 1991-03-18 1992-03-24 Warner-Lambert Company Method of treating neurodegenerative diseases
FI943798A7 (fi) * 1992-02-19 1994-08-18 Pfizer Kasvaimenvastaisen vaikutuksen lisäämiseen tarkoitettuja heterosyklisi ä yhdisteitä
HRP20000209A2 (en) 1997-10-20 2001-04-30 Hoffmann La Roche Bicyclic kinase inhibitors
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
HRP20090395T1 (hr) * 2006-04-19 2009-08-31 Boehringer Ingelheim International Gmbh Dihidrotienpirimidini za liječenje upalnih bolesti
KR101533461B1 (ko) 2006-04-26 2015-07-02 에프. 호프만-라 로슈 아게 Ｐｉ３ｋ저해제로 유용한 티에노［3,2-ｄ］피리미딘 유도체
PL2041139T3 (pl) 2006-04-26 2012-05-31 Hoffmann La Roche Związki farmaceutyczne
AU2007243466B2 (en) 2006-04-26 2012-01-19 F. Hoffmann-La Roche Ag Phosphoinositide 3-kinase inhibitor compounds and pharmaceutical compositions containing them
CA2671845C (en) * 2006-12-07 2015-03-24 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and methods of use
PE20081679A1 (es) * 2006-12-07 2008-12-18 Hoffmann La Roche Compuestos del inhibidor de fosfoinositida 3-cinasa y metodos de uso
CN101932587A (zh) 2007-09-24 2010-12-29 吉宁特有限公司 噻唑并嘧啶pi3k抑制剂化合物及使用方法
RU2500681C2 (ru) * 2007-10-19 2013-12-10 Берингер Ингельхайм Интернациональ Гмбх Замещенные гетероциклом пиперазинодигидротиенопиримидины
WO2009055730A1 (en) 2007-10-25 2009-04-30 Genentech, Inc. Process for making thienopyrimidine compounds
GB0721095D0 (en) 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
JP5709766B2 (ja) 2009-03-12 2015-04-30 ジェネンテック， インコーポレイテッド 造血器腫瘍の治療のためのホスホイノシチド３キナーゼ阻害剤化合物と化学療法剤の併用
MX2011012520A (es) 2009-05-27 2011-12-12 Hoffmann La Roche Compuestos inhibidores de pi3k de pirimidina biciclicos selectivos para p110 delta y metodos de uso de los mismos.
SG182247A1 (en) * 2009-05-27 2012-08-30 Hoffmann La Roche Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
KR20130058672A (ko) 2010-04-16 2013-06-04 제넨테크, 인크. ＰＩ3Ｋ/ＡＫＴ 키나제 경로 억제제 효능에 대한 예측 바이오마커로서의 ＦＯＸＯ３ａ
US20140004209A1 (en) 2010-12-22 2014-01-02 Genentech, Inc. Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms
RU2015140573A (ru) 2013-02-25 2017-03-30 Дженентек, Инк. Способы и композиции для обнаружения и лечения устойчивого к лекарственным средствам мутанта акт
GB201410816D0 (en) * 2014-06-17 2014-07-30 Ucb Biopharma Sprl And Katholieke Universiteit Leuven Therapeutic agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3259623A (en) * 1963-06-14 1966-07-05 Olin Mathieson Process for preparing 2-(secondary amino)-halogenopyrimidines
DE1470356A1 (de) * 1964-01-15 1970-04-30 Thomae Gmbh Dr K Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
US3210368A (en) * 1964-09-29 1965-10-05 Ciba Geigy Corp Certain 2-amino-4-aryl-5-n, n-disubstituted amino-lower alkyl-thiazole compounds

Also Published As

Publication number Publication date
DK129844C (cg-RX-API-DMAC7.html) 1975-05-12
DD97656A5 (cg-RX-API-DMAC7.html) 1973-05-12
HU163960B (cg-RX-API-DMAC7.html) 1973-11-28
GB1393161A (en) 1975-05-07
ES402302A1 (es) 1975-04-01
IL39341A0 (en) 1972-07-26
IL39341A (en) 1975-08-31
NL7206041A (cg-RX-API-DMAC7.html) 1972-11-07
BG20593A3 (bg) 1975-12-05
US3888851A (en) 1975-06-10
PL82381B1 (cg-RX-API-DMAC7.html) 1975-10-31
FR2135294A1 (cg-RX-API-DMAC7.html) 1972-12-15
BE783044A (fr) 1972-11-06
AT318619B (de) 1974-11-11
RO62428A (fr) 1978-01-15
FR2135294B1 (cg-RX-API-DMAC7.html) 1975-10-17
AU4181572A (en) 1973-11-08

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