DK124680B - Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken. - Google Patents

Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken.

Info

Publication number
DK124680B
DK124680B DK224769AA DK224769A DK124680B DK 124680 B DK124680 B DK 124680B DK 224769A A DK224769A A DK 224769AA DK 224769 A DK224769 A DK 224769A DK 124680 B DK124680 B DK 124680B
Authority
DK
Denmark
Prior art keywords
oxazolines
preparation
substituted steroid
pregnane series
pregnane
Prior art date
Application number
DK224769AA
Other languages
Danish (da)
English (en)
Inventor
G Winters
G Nathansohn
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Priority to DK569670A priority Critical patent/DK129452B/da
Publication of DK124680B publication Critical patent/DK124680B/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0057—Nitrogen and oxygen
    • C07J71/0068—Nitrogen and oxygen at position 16(17)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011—Unsubstituted amino radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK224769AA 1968-05-03 1969-04-24 Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken. DK124680B (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK569670A DK129452B (da) 1968-05-03 1970-11-10 Analogifremgangsmåde til fremstilling af 9α-fluor-11β,21-dihydroxy-pregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidiner eller oxazolidinooxaziner.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1602968 1968-05-03

Publications (1)

Publication Number Publication Date
DK124680B true DK124680B (da) 1972-11-13

Family

ID=11148457

Family Applications (2)

Application Number Title Priority Date Filing Date
DK224769AA DK124680B (da) 1968-05-03 1969-04-24 Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken.
DK569770AA DK128352B (da) 1968-05-03 1970-11-10 Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK569770AA DK128352B (da) 1968-05-03 1970-11-10 Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner.

Country Status (16)

Country Link
US (1) US3631033A (de)
AT (2) AT300218B (de)
BE (1) BE731718A (de)
BR (1) BR6908511D0 (de)
CH (1) CH511823A (de)
DE (1) DE1921778A1 (de)
DK (2) DK124680B (de)
ES (2) ES366738A1 (de)
FI (3) FI46374C (de)
FR (1) FR2007756B1 (de)
GB (1) GB1254487A (de)
IL (1) IL31997A (de)
LU (1) LU58451A1 (de)
NL (2) NL6906149A (de)
NO (1) NO128608B (de)
SE (4) SE363098B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7107998A (de) * 1970-07-09 1972-01-11
IT1134455B (it) * 1980-11-26 1986-08-13 Lepetit Spa Procedimento per la preparazione di derivati 16alfa-idrossi-17alfa-aminopregnanici
US20030083231A1 (en) * 1998-11-24 2003-05-01 Ahlem Clarence N. Blood cell deficiency treatment method
CA2496867A1 (en) * 2002-08-28 2004-03-11 Hollis-Eden Pharmaceuticals, Inc. Therapeutic treatment methods
US20050101581A1 (en) * 2002-08-28 2005-05-12 Reading Christopher L. Therapeutic treatment methods 2
CN102482318B (zh) * 2009-09-11 2015-11-25 奇斯药制品公司 异噁唑烷衍生物
EP2716648B1 (de) * 2011-03-15 2017-06-14 CHIESI FARMACEUTICI S.p.A. Isoxazolidin-derivate
KR20140039161A (ko) 2011-03-15 2014-04-01 키에시 파르마슈티시 엣스. 피. 에이. 이소옥사졸리딘 유도체
US9155747B2 (en) * 2012-09-13 2015-10-13 Chiesi Farmaceutici S.P.A. Isoxazolidine derivatives

Also Published As

Publication number Publication date
FR2007756A1 (de) 1970-01-09
NL7709675A (nl) 1977-12-30
FI46374C (fi) 1973-03-12
BE731718A (de) 1969-10-01
DK128352B (da) 1974-04-16
FI46376B (de) 1972-11-30
GB1254487A (en) 1971-11-24
BR6908511D0 (pt) 1973-02-08
SE373578B (sv) 1975-02-10
US3631033A (en) 1971-12-28
DE1965963A1 (de) 1970-12-23
NL6906149A (de) 1969-11-05
AT291450B (de) 1971-07-12
IL31997A (en) 1974-03-14
SE373131B (de) 1975-01-27
FR2007756B1 (de) 1975-10-10
ES371991A1 (es) 1971-12-01
DE1965963B2 (de) 1973-02-08
FI46374B (de) 1972-11-30
ES366738A1 (es) 1971-03-16
FI46377B (de) 1972-11-30
CH511823A (fr) 1971-08-31
NO128608B (de) 1973-12-17
FI46377C (fi) 1973-03-12
FI46376C (fi) 1973-03-12
LU58451A1 (de) 1969-07-21
SE363098B (de) 1974-01-07
IL31997A0 (en) 1969-06-25
DE1921778A1 (de) 1969-11-20
SE378250B (de) 1975-08-25
AT300218B (de) 1972-07-25

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