DK121125B - Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller syreadditionssalte deraf. - Google Patents

Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller syreadditionssalte deraf.

Info

Publication number
DK121125B
DK121125B DK113168AA DK113168A DK121125B DK 121125 B DK121125 B DK 121125B DK 113168A A DK113168A A DK 113168AA DK 113168 A DK113168 A DK 113168A DK 121125 B DK121125 B DK 121125B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
benzodiazepine derivatives
benzodiazepine
Prior art date
Application number
DK113168AA
Other languages
Danish (da)
English (en)
Inventor
G Archer
L Sternbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK121125B publication Critical patent/DK121125B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK113168AA 1967-03-17 1968-03-15 Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller syreadditionssalte deraf. DK121125B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62383467A 1967-03-17 1967-03-17

Publications (1)

Publication Number Publication Date
DK121125B true DK121125B (da) 1971-09-13

Family

ID=24499574

Family Applications (1)

Application Number Title Priority Date Filing Date
DK113168AA DK121125B (da) 1967-03-17 1968-03-15 Fremgangsmåde til fremstilling af 1,4-benzodiazepinderivater eller syreadditionssalte deraf.

Country Status (16)

Country Link
US (1) US3553199A (fi)
AT (1) AT278820B (fi)
BE (1) BE712207A (fi)
CH (1) CH493539A (fi)
DE (1) DE1695226A1 (fi)
DK (1) DK121125B (fi)
ES (1) ES351720A1 (fi)
FI (1) FI48088C (fi)
FR (1) FR1556196A (fi)
GB (1) GB1148288A (fi)
IL (1) IL29640A (fi)
MY (1) MY6900399A (fi)
NL (1) NL6803724A (fi)
NO (1) NO123037B (fi)
SE (1) SE335736B (fi)
YU (1) YU34201B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3817984A (en) * 1969-07-08 1974-06-18 Sumitomo Chemical Co Process for producing benzodiazepine derivatives
FR2054476A1 (en) * 1969-07-09 1971-04-23 Sumitomo Chemical Co Dihydro benzodiazpine derivs with tranqui- - lising, muscle-relaxant, antispasmodic and
BE785937A (fr) * 1971-07-08 1973-01-08 Sandoz Sa Nouveaux derives de la quinazoline, leur preparation et leur application comme medicaments
JPS6019753A (ja) * 1983-07-13 1985-01-31 Shionogi & Co Ltd オルト−(モノ置換アミノ)フエニルイミン類およびその製造法

Also Published As

Publication number Publication date
NL6803724A (fi) 1968-09-18
NO123037B (fi) 1971-09-20
FI48088B (fi) 1974-02-28
DE1695226A1 (de) 1971-03-18
SE335736B (fi) 1971-06-07
GB1148288A (en) 1969-04-10
AT278820B (de) 1970-02-10
ES351720A1 (es) 1969-06-16
YU34201B (en) 1979-02-28
CH493539A (de) 1970-07-15
MY6900399A (en) 1969-12-31
YU58368A (en) 1978-06-30
BE712207A (fi) 1968-09-16
FI48088C (fi) 1974-06-10
IL29640A (en) 1972-06-28
US3553199A (en) 1971-01-05
FR1556196A (fi) 1969-01-31

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