DK115771B - Fremgangsmåde til fremstilling af (3,5-diamino-6-halogenpyrazinoyl) guanidin- eller (3,5-diamino-6-halogenpyrazinamido) guanidin-forbindelser eller syreadditionssalte deraf. - Google Patents

Fremgangsmåde til fremstilling af (3,5-diamino-6-halogenpyrazinoyl) guanidin- eller (3,5-diamino-6-halogenpyrazinamido) guanidin-forbindelser eller syreadditionssalte deraf.

Info

Publication number
DK115771B
DK115771B DK286467AA DK286467A DK115771B DK 115771 B DK115771 B DK 115771B DK 286467A A DK286467A A DK 286467AA DK 286467 A DK286467 A DK 286467A DK 115771 B DK115771 B DK 115771B
Authority
DK
Denmark
Prior art keywords
diamino
guanidine
halopyrazinoyl
halopyrazinamido
preparation
Prior art date
Application number
DK286467AA
Other languages
English (en)
Inventor
P Pollak
R Tull
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK115771B publication Critical patent/DK115771B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK286467AA 1966-08-25 1967-06-01 Fremgangsmåde til fremstilling af (3,5-diamino-6-halogenpyrazinoyl) guanidin- eller (3,5-diamino-6-halogenpyrazinamido) guanidin-forbindelser eller syreadditionssalte deraf. DK115771B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57490966A 1966-08-25 1966-08-25

Publications (1)

Publication Number Publication Date
DK115771B true DK115771B (da) 1969-11-10

Family

ID=24298146

Family Applications (1)

Application Number Title Priority Date Filing Date
DK286467AA DK115771B (da) 1966-08-25 1967-06-01 Fremgangsmåde til fremstilling af (3,5-diamino-6-halogenpyrazinoyl) guanidin- eller (3,5-diamino-6-halogenpyrazinamido) guanidin-forbindelser eller syreadditionssalte deraf.

Country Status (7)

Country Link
US (1) US3432502A (da)
BE (1) BE699435A (da)
CH (1) CH484161A (da)
DK (1) DK115771B (da)
ES (1) ES341321A1 (da)
GB (1) GB1184709A (da)
NL (1) NL6707563A (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3506662A (en) * 1968-04-30 1970-04-14 Merck & Co Inc Process for preparation of pyrazinoyland pyrazinamidoguanidines
US4246406A (en) * 1979-03-27 1981-01-20 Merck & Co., Inc. Heterocyclic substituted pyrazinoylguanidines
US4224447A (en) * 1979-03-27 1980-09-23 Merck & Co., Inc. Novel pyrazinecarboxamides and processes for preparing same
EA017919B1 (ru) 2007-12-10 2013-04-30 Новартис Аг Производные пиразин-2-карбоксамида для лечения заболеваний, которые поддаются лечению путем блокирования эпителиальных натриевых каналов

Also Published As

Publication number Publication date
NL6707563A (da) 1968-02-26
CH484161A (de) 1970-01-15
GB1184709A (en) 1970-03-18
BE699435A (da) 1967-12-04
US3432502A (en) 1969-03-11
ES341321A1 (es) 1968-10-16

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