DK1173176T3 - Anvendelse af polycycliske 2-aminothiazolsystemer til fremstilling af medikamenter til forebyggelse eller behandling af obesitas - Google Patents
Anvendelse af polycycliske 2-aminothiazolsystemer til fremstilling af medikamenter til forebyggelse eller behandling af obesitasInfo
- Publication number
- DK1173176T3 DK1173176T3 DK00905028T DK00905028T DK1173176T3 DK 1173176 T3 DK1173176 T3 DK 1173176T3 DK 00905028 T DK00905028 T DK 00905028T DK 00905028 T DK00905028 T DK 00905028T DK 1173176 T3 DK1173176 T3 DK 1173176T3
- Authority
- DK
- Denmark
- Prior art keywords
- treatment
- aminothiazole
- obesity
- polycyclic
- systems
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Child & Adolescent Psychology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19908537A DE19908537A1 (de) | 1999-02-26 | 1999-02-26 | Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1173176T3 true DK1173176T3 (da) | 2004-09-27 |
Family
ID=7899081
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00905028T DK1173176T3 (da) | 1999-02-26 | 2000-02-05 | Anvendelse af polycycliske 2-aminothiazolsystemer til fremstilling af medikamenter til forebyggelse eller behandling af obesitas |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6476059B1 (ja) |
| EP (1) | EP1173176B1 (ja) |
| JP (1) | JP4728483B2 (ja) |
| KR (1) | KR20020002394A (ja) |
| CN (1) | CN1161120C (ja) |
| AT (1) | ATE267597T1 (ja) |
| AU (1) | AU766295B2 (ja) |
| BR (1) | BR0008557A (ja) |
| CA (1) | CA2362554A1 (ja) |
| DE (2) | DE19908537A1 (ja) |
| DK (1) | DK1173176T3 (ja) |
| ES (1) | ES2218122T3 (ja) |
| HK (1) | HK1045809B (ja) |
| PT (1) | PT1173176E (ja) |
| WO (1) | WO2000051602A1 (ja) |
| ZA (1) | ZA200106199B (ja) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19908538A1 (de) * | 1999-02-26 | 2000-08-31 | Aventis Pharma Gmbh | Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen |
| JP2002543067A (ja) * | 1999-04-22 | 2002-12-17 | シナプティック・ファーマスーティカル・コーポレーション | 選択的なｎｐｙ（ｙ５）のアンタゴニスト |
| AU2001246494A1 (en) * | 2000-03-03 | 2001-09-12 | Novartis Ag | Condensed thiazolamines and their use as neuropeptide y5 antagonists |
| EP1305023A4 (en) * | 2000-08-01 | 2005-02-23 | Univ Virginia | USE OF SELECTIVE AGONISTS, ANTAGONISTS AND ALLOSTERIC AMPLIFIERS OF THE ADENOSINE A1 RECEPTOR TO INFLUENCE THE ANGIOGENESIS |
| WO2003061655A1 (en) * | 2002-01-16 | 2003-07-31 | University Of Virginia Patent Foundation | 2-aminothiazole allosteric enhancers of a1 adenosine receptors |
| WO2004110338A2 (en) * | 2003-06-12 | 2004-12-23 | Biomas Ltd. | Methods of treating obesity and related disorders using tellurium and selenium compounds |
| JP2008508336A (ja) | 2004-08-05 | 2008-03-21 | エフ．ホフマン−ラ ロシュ アーゲー | 置換されたｎ−アシル−２−アミノチアゾール |
| WO2006080406A1 (ja) * | 2005-01-28 | 2006-08-03 | Taisho Pharmaceutical Co., Ltd. | 三環性化合物 |
| PL2276767T3 (pl) | 2008-03-31 | 2014-09-30 | Genentech Inc | Związki benzopiranowe i benzoksepinowe będące inhibitorami pi3k oraz metody ich stosowania |
| SG10201407781SA (en) | 2009-09-28 | 2015-01-29 | Hoffmann La Roche | Benzoxepin PI3K Inhibitor Compounds And Methods Of Use |
| RS53164B (en) | 2009-09-28 | 2014-06-30 | F. Hoffmann-La Roche Ag | BENZOXAZEPINE PI3K INHIBITOR COMPOUNDS AND THEIR USE IN CANCER TREATMENT |
| CA2825966A1 (en) | 2011-03-21 | 2012-09-27 | F. Hoffmann-La Roche Ag | Benzoxazepin compounds selective for pi3k p110 delta and methods of use |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3507868A (en) * | 1968-10-21 | 1970-04-21 | Sandoz Ag | Imidazo(2,1-b)thiazoles and thiazolo(3,2-a)pyrimidines |
| DE2640358A1 (de) * | 1976-09-08 | 1978-03-16 | Hoechst Ag | Thiazolidinderivate und verfahren zu ihrer herstellung |
| JPS5334471A (en) * | 1976-09-10 | 1978-03-31 | Toshiba Corp | Manufacture for semiconductor device |
| CA1292226C (en) * | 1986-01-16 | 1991-11-19 | Terumi Hachiya | Indenothiazole derivative and process for preparing the same |
| IE68593B1 (en) * | 1989-12-06 | 1996-06-26 | Sanofi Sa | Heterocyclic substituted acylaminothiazoles their preparation and pharmaceutical compositions containing them |
| DE19831878C2 (de) * | 1998-07-17 | 2001-05-17 | Aventis Pharma Gmbh | Polycyclische Thiazolidin-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| DE19908538A1 (de) * | 1999-02-26 | 2000-08-31 | Aventis Pharma Gmbh | Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen |
-
1999
- 1999-02-26 DE DE19908537A patent/DE19908537A1/de not_active Withdrawn
-
2000
- 2000-02-05 WO PCT/EP2000/000925 patent/WO2000051602A1/de not_active Application Discontinuation
- 2000-02-05 KR KR1020017010840A patent/KR20020002394A/ko not_active Application Discontinuation
- 2000-02-05 ES ES00905028T patent/ES2218122T3/es not_active Expired - Lifetime
- 2000-02-05 CN CNB008042209A patent/CN1161120C/zh not_active Expired - Fee Related
- 2000-02-05 AT AT00905028T patent/ATE267597T1/de not_active IP Right Cessation
- 2000-02-05 CA CA002362554A patent/CA2362554A1/en not_active Abandoned
- 2000-02-05 DE DE50006603T patent/DE50006603D1/de not_active Expired - Lifetime
- 2000-02-05 EP EP00905028A patent/EP1173176B1/de not_active Expired - Lifetime
- 2000-02-05 BR BR0008557-0A patent/BR0008557A/pt not_active IP Right Cessation
- 2000-02-05 JP JP2000602070A patent/JP4728483B2/ja not_active Expired - Fee Related
- 2000-02-05 PT PT00905028T patent/PT1173176E/pt unknown
- 2000-02-05 DK DK00905028T patent/DK1173176T3/da active
- 2000-02-05 AU AU26703/00A patent/AU766295B2/en not_active Ceased
- 2000-02-10 US US09/501,209 patent/US6476059B1/en not_active Expired - Lifetime
-
2001
- 2001-07-27 ZA ZA200106199A patent/ZA200106199B/en unknown
-
2002
- 2002-09-26 HK HK02107056.4A patent/HK1045809B/zh not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20020002394A (ko) | 2002-01-09 |
| DE50006603D1 (de) | 2004-07-01 |
| ATE267597T1 (de) | 2004-06-15 |
| WO2000051602A1 (de) | 2000-09-08 |
| BR0008557A (pt) | 2001-12-18 |
| CN1161120C (zh) | 2004-08-11 |
| HK1045809A1 (en) | 2002-12-13 |
| JP2002538117A (ja) | 2002-11-12 |
| CN1349404A (zh) | 2002-05-15 |
| JP4728483B2 (ja) | 2011-07-20 |
| PT1173176E (pt) | 2004-09-30 |
| AU766295B2 (en) | 2003-10-16 |
| EP1173176A1 (de) | 2002-01-23 |
| EP1173176B1 (de) | 2004-05-26 |
| ES2218122T3 (es) | 2004-11-16 |
| ZA200106199B (en) | 2002-03-06 |
| AU2670300A (en) | 2000-09-21 |
| CA2362554A1 (en) | 2000-09-08 |
| US6476059B1 (en) | 2002-11-05 |
| DE19908537A1 (de) | 2000-08-31 |
| HK1045809B (zh) | 2005-04-22 |
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