DK115474B - Analogifremgangsmåde til fremstilling af N-p-chlorbenzoyl-5-fluorcytosin. - Google Patents
Analogifremgangsmåde til fremstilling af N-p-chlorbenzoyl-5-fluorcytosin.Info
- Publication number
- DK115474B DK115474B DK547566AA DK547566A DK115474B DK 115474 B DK115474 B DK 115474B DK 547566A A DK547566A A DK 547566AA DK 547566 A DK547566 A DK 547566A DK 115474 B DK115474 B DK 115474B
- Authority
- DK
- Denmark
- Prior art keywords
- fluorocytosine
- chlorobenzoyl
- preparation
- analogous process
- analogous
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US502586A US3309359A (en) | 1965-10-22 | 1965-10-22 | N-mono-acyl-5-fluorocytosine derivatives and process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK115474B true DK115474B (da) | 1969-10-13 |
Family
ID=23998481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK547566AA DK115474B (da) | 1965-10-22 | 1966-10-21 | Analogifremgangsmåde til fremstilling af N-p-chlorbenzoyl-5-fluorcytosin. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US3309359A (da) |
| BE (1) | BE688539A (da) |
| BR (1) | BR6683864D0 (da) |
| CH (1) | CH475258A (da) |
| DE (1) | DE1695160A1 (da) |
| DK (1) | DK115474B (da) |
| FR (1) | FR5908M (da) |
| GB (1) | GB1110357A (da) |
| IL (1) | IL26726A (da) |
| NL (1) | NL6614240A (da) |
| SE (1) | SE330176B (da) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3894000A (en) * | 1971-01-27 | 1975-07-08 | Upjohn Co | Ara-cytidine derivatives and process of preparation |
| US3975367A (en) * | 1971-06-08 | 1976-08-17 | The Upjohn Company | Arabinofuranosyl N4 -aminoacyl cytosine containing compounds |
| US4022963A (en) * | 1972-06-08 | 1977-05-10 | Deutsch Daniel Harold | Acetylation process for nucleoside compounds |
| US3991045A (en) * | 1973-05-30 | 1976-11-09 | Asahi Kasei Kogyo Kabushiki Kaisha | N4 -acylarabinonucleosides |
| JPS5159880A (en) * | 1974-11-22 | 1976-05-25 | Asahi Chemical Ind | N44 ashirunukureoshidojikarubonsanesuteruno seiho |
| JPS5924999B2 (ja) * | 1978-06-10 | 1984-06-13 | 富山化学工業株式会社 | 新規な５−フルオロ−２′−デオキシ−β−ウリジン誘導体の製造法 |
| JPS5535057A (en) * | 1978-09-05 | 1980-03-11 | Funai Corp | 2'-deoxy-5-fluorouridine derivative, its preparation, and antitumor agent comprising it |
| JPS59167600A (ja) * | 1983-03-14 | 1984-09-21 | Microbial Chem Res Found | ２′−デオキシオキザノシンおよびその製造法 |
| CN100560073C (zh) | 2001-12-14 | 2009-11-18 | 法玛塞特公司 | 用于治疗病毒感染的n4-酰基胞嘧啶核苷 |
| DK2562162T3 (da) | 2008-01-22 | 2015-11-23 | Dow Agrosciences Llc | N-cyano-4-amino-5-fluor-pyrimidinderivater som fungicider |
| PL2317851T3 (pl) | 2008-08-01 | 2014-06-30 | Dow Agrosciences Llc | Zastosowanie 5-fluorocytozyny jako fungicydu |
| DK2462134T3 (da) | 2009-08-07 | 2014-08-11 | Dow Agrosciences Llc | N1-sulfonyl-5-fluorpyrimidinonderivater |
| UA112284C2 (uk) * | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| UA109780C2 (uk) * | 2010-01-07 | 2015-10-12 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | ТІАЗОЛО[5,4-d]ПІРИМІДИНИ І ЇХ ЗАСТОСУВАННЯ ЯК АГРОХІМІЧНИХ ЗАСОБІВ |
| LT2775842T (lt) | 2011-08-17 | 2017-12-11 | Adama Makhteshim Ltd. | 1-pakeisti-5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinono dariniai, kaip fungicidiniai agentai, skirti panaudoti augalų apsaugai |
| UA117743C2 (uk) | 2012-12-28 | 2018-09-25 | Адама Махтешім Лтд. | N-(заміщені)-5-фтор-4-іміно-3-метил-2-оксо-3,4-дигідропіримідин-1(2h)-карбоксамідні похідні |
| RU2656101C2 (ru) | 2012-12-28 | 2018-05-31 | Адама Мактешим Лтд. | Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она |
| RU2638556C2 (ru) | 2012-12-28 | 2017-12-14 | Адама Мактешим Лтд. | Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата |
| RU2644014C2 (ru) | 2012-12-31 | 2018-02-07 | Адама Мактешим Лтд. | Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов |
| BR112016015155A2 (pt) | 2013-12-31 | 2017-08-08 | Adama Makhteshim Ltd | Misturas fungicidas sinergísticas para controle fúngico em cereais |
| CR20210172A (es) | 2013-12-31 | 2021-05-11 | Adama Makhteshim Ltd | 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2 (1h)-ona y los procesos para su preparación |
| EP3655396A1 (en) | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| CN109651467A (zh) * | 2019-01-15 | 2019-04-19 | 齐鲁天和惠世制药有限公司 | 一种卡培他滨杂质及其制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2949451A (en) * | 1959-04-21 | 1960-08-16 | Hoffmann La Roche | Preparation of thymidine and deoxyfluorouridine, and intermediates therefor |
| NL299755A (da) * | 1959-06-03 | |||
| GB1070413A (en) * | 1962-11-15 | 1967-06-01 | Sankyo Co | A process for preparing purine and pyrimidine nucleosides |
-
1965
- 1965-10-22 US US502586A patent/US3309359A/en not_active Expired - Lifetime
-
1966
- 1966-09-23 CH CH1376966A patent/CH475258A/de not_active IP Right Cessation
- 1966-09-26 DE DE19661695160 patent/DE1695160A1/de active Pending
- 1966-10-10 NL NL6614240A patent/NL6614240A/xx unknown
- 1966-10-20 SE SE14339/66A patent/SE330176B/xx unknown
- 1966-10-20 IL IL26726A patent/IL26726A/xx unknown
- 1966-10-20 BE BE688539D patent/BE688539A/xx unknown
- 1966-10-20 FR FR80695A patent/FR5908M/fr not_active Expired
- 1966-10-21 BR BR183864/66A patent/BR6683864D0/pt unknown
- 1966-10-21 DK DK547566AA patent/DK115474B/da unknown
- 1966-10-21 GB GB47304/66A patent/GB1110357A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FR5908M (da) | 1968-03-25 |
| CH475258A (de) | 1969-07-15 |
| DE1695160A1 (de) | 1970-12-17 |
| US3309359A (en) | 1967-03-14 |
| GB1110357A (en) | 1968-04-18 |
| SE330176B (da) | 1970-11-09 |
| NL6614240A (da) | 1967-04-24 |
| BE688539A (da) | 1967-04-20 |
| BR6683864D0 (pt) | 1973-12-26 |
| IL26726A (en) | 1970-06-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK133618B (da) | Analogifremgangsmåde til fremstilling af 1-hydroxyaryl-2-aminoalkanoler. | |
| DK118769B (da) | Fremgangsmåde til fremstilling af O-methyl-S-methyl-phosphoroamidothioat. | |
| DK115474B (da) | Analogifremgangsmåde til fremstilling af N-p-chlorbenzoyl-5-fluorcytosin. | |
| DK111892B (da) | Fremgangsmåde til fremstilling af pyrazinimidoyl-guanidinforbindelser. | |
| DK127415B (da) | Fremgangsmåde til fremstilling af α-benzyl-β,β-dialkoxypropionitriler. | |
| DK118505B (da) | Fremgangsmåde til fremstilling af isoindolin-2-sulfonylurinstoffer. | |
| DK118239B (da) | Fremgangsmåde til fremstilling af substituerede 4-hydroxykinoliner. | |
| DK135234B (da) | Analogifremgangsmåde til fremstilling af piperazin-phenylethanolforbindelser. | |
| DK120193B (da) | Fremgangsmåde til fremstilling af 3-amino-isoxazolderivater. | |
| DK117954B (da) | Fremgangsmåde til fremstilling af 3-amino-2-cyanoacrylamid. | |
| DK124886B (da) | Fremgangsnmåde til fremstilling af 1-hydroxy-benzimidazol-N-oxider. | |
| DK121759B (da) | Analogifremgangsmåde til fremstilling af 3-oxo-7α-methylgona-4,9-diener. | |
| DK115551B (da) | Fremgangsmåde til fremstilling af 6-aminouracil-5-carbonamid-N-sulfonamider. | |
| DK118670B (da) | Fremgangsmåde til fremstilling af cyanphenoler. | |
| DK118458B (da) | Fremgangsmåde til fremstilling af 5-halogen-2-amino-benzophenoniminer. | |
| DK118132B (da) | Fremgangsmåde til fremstilling af derivater af 5-nitro-2-furyl-isoxazoler. | |
| DK114063B (da) | Fremgangsmåde til fremstilling af 1-methyl-2-isopropyl-5-nitro-imidazol. | |
| DK120344B (da) | Fremgangsmåde til fremstilling af 5-benzyl-pyrimidiner. | |
| DK122527B (da) | Fremgangsmåde til fremstilling af 3-nitro-2-oxo-tetrahydro-imidazoler. | |
| DK119980B (da) | Fremgangsmåde til fremstilling af 2-alkoxy-4-sulfanilamido-quinazolinderivater. | |
| DK117956B (da) | Fremgangsmåde til fremstilling af 3-oxogona-4,9-diener. | |
| DK114204B (da) | Fremgangsmåde til fremstilling af carboxamidoalkyl-1,3-benzoxaziner. | |
| DK114626B (da) | Fremgangsmåde til fremstilling af 2-substitueret-4-amino-5-acylamidometylpyrimidin. | |
| DK119830B (da) | Analogifremgangsmåde til fremstilling af arylsulfonylsemicarbazider. | |
| DK126378B (da) | Analogifremgangsmåde til fremstilling af 17α-acyloxy-9α-chlor-11β-hydroxy-progesteroner. |