DK1125940T3 - Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse - Google Patents

Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse

Info

Publication number
DK1125940T3
DK1125940T3 DK01400407T DK01400407T DK1125940T3 DK 1125940 T3 DK1125940 T3 DK 1125940T3 DK 01400407 T DK01400407 T DK 01400407T DK 01400407 T DK01400407 T DK 01400407T DK 1125940 T3 DK1125940 T3 DK 1125940T3
Authority
DK
Denmark
Prior art keywords
quinolinylphosphonic
heteroaryl
aryl
derivatives
acids
Prior art date
Application number
DK01400407T
Other languages
Danish (da)
English (en)
Inventor
Alex Cordi
Patrice Desos
Pierre Lestage
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Application granted granted Critical
Publication of DK1125940T3 publication Critical patent/DK1125940T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/60Quinoline or hydrogenated quinoline ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK01400407T 2000-02-18 2001-02-16 Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse DK1125940T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0002013A FR2805262A1 (fr) 2000-02-18 2000-02-18 Nouveaux derives d'acides aryle ou heteroaryle quinolinyl phosphoniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
DK1125940T3 true DK1125940T3 (da) 2003-05-05

Family

ID=8847124

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01400407T DK1125940T3 (da) 2000-02-18 2001-02-16 Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse

Country Status (23)

Country Link
US (1) US6420386B1 (hu)
EP (1) EP1125940B1 (hu)
JP (1) JP2001278890A (hu)
KR (1) KR20010082704A (hu)
CN (1) CN1317489A (hu)
AR (1) AR027431A1 (hu)
AT (1) ATE231154T1 (hu)
AU (1) AU2303901A (hu)
BR (1) BR0100600A (hu)
CA (1) CA2337301A1 (hu)
DE (1) DE60100080T2 (hu)
DK (1) DK1125940T3 (hu)
EA (1) EA200100157A3 (hu)
ES (1) ES2190426T3 (hu)
FR (1) FR2805262A1 (hu)
HK (1) HK1039943A1 (hu)
HU (1) HUP0100751A3 (hu)
MX (1) MXPA01001559A (hu)
NO (1) NO20010802L (hu)
NZ (1) NZ510003A (hu)
PL (1) PL345917A1 (hu)
SI (1) SI1125940T1 (hu)
ZA (1) ZA200101337B (hu)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2805260A1 (fr) * 2000-02-18 2001-08-24 Adir Nouveaux derives d'acides 6-sulfamoyl-3-quinolinyl phosphoniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US20110178041A1 (en) 2008-09-25 2011-07-21 Yasushi Kohno Heterocyclic biaryl derivative and pde inhibitor comprising same as active ingredient
US20110224250A1 (en) * 2008-10-09 2011-09-15 Yasushi Kohno Isoquinoline derivative, and pde inhibitor comprising same as active ingredient

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2683818B1 (fr) * 1991-11-14 1993-12-31 Adir Cie Nouveaux derives de 3-sulfonylamino-2-(1h)-quinoleinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5342946A (en) * 1992-12-02 1994-08-30 Guilford Pharmaceuticals Inc. Phosphonoalkylquinolin-2-ones as novel antagonists of non-NMDA ionotropic excitatory amino acid receptors
FR2709489B1 (fr) * 1993-08-31 1995-10-20 Adir Nouveaux dérivés de 2-(1H)-quinoléinone, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
FR2750988B1 (fr) * 1996-07-11 1998-09-18 Adir Nouveaux derives de 2-(1h)-quinoleinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
ATE231154T1 (de) 2003-02-15
AU2303901A (en) 2001-08-23
DE60100080D1 (de) 2003-02-20
EA200100157A3 (ru) 2001-10-22
ZA200101337B (en) 2001-08-21
FR2805262A1 (fr) 2001-08-24
JP2001278890A (ja) 2001-10-10
MXPA01001559A (es) 2002-08-06
SI1125940T1 (en) 2003-04-30
CN1317489A (zh) 2001-10-17
BR0100600A (pt) 2001-09-18
HK1039943A1 (zh) 2002-05-17
ES2190426T3 (es) 2003-08-01
HUP0100751A2 (hu) 2002-01-28
CA2337301A1 (fr) 2001-08-18
EP1125940B1 (fr) 2003-01-15
EP1125940A1 (fr) 2001-08-22
PL345917A1 (en) 2001-08-27
EA200100157A2 (ru) 2001-08-27
KR20010082704A (ko) 2001-08-30
NO20010802D0 (no) 2001-02-16
NZ510003A (en) 2001-09-28
HU0100751D0 (en) 2001-04-28
NO20010802L (no) 2001-08-20
AR027431A1 (es) 2003-03-26
HUP0100751A3 (en) 2002-09-30
DE60100080T2 (de) 2003-11-20
US6420386B1 (en) 2002-07-16

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