DK1125940T3 - Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse - Google Patents

Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse

Info

Publication number
DK1125940T3
DK1125940T3 DK01400407T DK01400407T DK1125940T3 DK 1125940 T3 DK1125940 T3 DK 1125940T3 DK 01400407 T DK01400407 T DK 01400407T DK 01400407 T DK01400407 T DK 01400407T DK 1125940 T3 DK1125940 T3 DK 1125940T3
Authority
DK
Denmark
Prior art keywords
quinolinylphosphonic
heteroaryl
aryl
derivatives
acids
Prior art date
Application number
DK01400407T
Other languages
English (en)
Inventor
Alex Cordi
Patrice Desos
Pierre Lestage
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Application granted granted Critical
Publication of DK1125940T3 publication Critical patent/DK1125940T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/60—Quinoline or hydrogenated quinoline ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
DK01400407T 2000-02-18 2001-02-16 Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse DK1125940T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0002013A FR2805262A1 (fr) 2000-02-18 2000-02-18 Nouveaux derives d'acides aryle ou heteroaryle quinolinyl phosphoniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
DK1125940T3 true DK1125940T3 (da) 2003-05-05

Family

ID=8847124

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01400407T DK1125940T3 (da) 2000-02-18 2001-02-16 Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse

Country Status (23)

Country Link
US (1) US6420386B1 (da)
EP (1) EP1125940B1 (da)
JP (1) JP2001278890A (da)
KR (1) KR20010082704A (da)
CN (1) CN1317489A (da)
AR (1) AR027431A1 (da)
AT (1) ATE231154T1 (da)
AU (1) AU2303901A (da)
BR (1) BR0100600A (da)
CA (1) CA2337301A1 (da)
DE (1) DE60100080T2 (da)
DK (1) DK1125940T3 (da)
EA (1) EA200100157A3 (da)
ES (1) ES2190426T3 (da)
FR (1) FR2805262A1 (da)
HK (1) HK1039943A1 (da)
HU (1) HUP0100751A3 (da)
MX (1) MXPA01001559A (da)
NO (1) NO20010802L (da)
NZ (1) NZ510003A (da)
PL (1) PL345917A1 (da)
SI (1) SI1125940T1 (da)
ZA (1) ZA200101337B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2805260A1 (fr) * 2000-02-18 2001-08-24 Adir Nouveaux derives d'acides 6-sulfamoyl-3-quinolinyl phosphoniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP2348018A4 (en) 2008-09-25 2012-04-25 Kyorin Seiyaku Kk HETEROCYCLIC BIARYLIC DERIVATIVE AND PDE INHIBITOR COMPRISING THE SAME AS ACTIVE INGREDIENT
WO2010041711A1 (ja) 2008-10-09 2010-04-15 杏林製薬株式会社 イソキノリン誘導体及びそれらを有効成分とするｐｄｅ阻害剤

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2683818B1 (fr) * 1991-11-14 1993-12-31 Adir Cie Nouveaux derives de 3-sulfonylamino-2-(1h)-quinoleinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5342946A (en) * 1992-12-02 1994-08-30 Guilford Pharmaceuticals Inc. Phosphonoalkylquinolin-2-ones as novel antagonists of non-NMDA ionotropic excitatory amino acid receptors
FR2709489B1 (fr) * 1993-08-31 1995-10-20 Adir Nouveaux dérivés de 2-(1H)-quinoléinone, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
FR2750988B1 (fr) * 1996-07-11 1998-09-18 Adir Nouveaux derives de 2-(1h)-quinoleinone, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
HUP0100751A3 (en) 2002-09-30
HUP0100751A2 (hu) 2002-01-28
PL345917A1 (en) 2001-08-27
EP1125940B1 (fr) 2003-01-15
HU0100751D0 (en) 2001-04-28
BR0100600A (pt) 2001-09-18
EA200100157A2 (ru) 2001-08-27
NZ510003A (en) 2001-09-28
AR027431A1 (es) 2003-03-26
SI1125940T1 (en) 2003-04-30
CN1317489A (zh) 2001-10-17
ATE231154T1 (de) 2003-02-15
AU2303901A (en) 2001-08-23
CA2337301A1 (fr) 2001-08-18
NO20010802L (no) 2001-08-20
ZA200101337B (en) 2001-08-21
KR20010082704A (ko) 2001-08-30
DE60100080D1 (de) 2003-02-20
NO20010802D0 (no) 2001-02-16
ES2190426T3 (es) 2003-08-01
EA200100157A3 (ru) 2001-10-22
MXPA01001559A (es) 2002-08-06
EP1125940A1 (fr) 2001-08-22
FR2805262A1 (fr) 2001-08-24
HK1039943A1 (zh) 2002-05-17
JP2001278890A (ja) 2001-10-10
US6420386B1 (en) 2002-07-16
DE60100080T2 (de) 2003-11-20

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DK1125940T3 (da) Derivater af aryl- eller heteroaryl-quinolinylphosphonsyrer, fremgangsmåde til fremstilling heraf og farmaceutiske lægemidler som indeholder disse