DK0952157T3 - 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin - Google Patents

9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin

Info

Publication number
DK0952157T3
DK0952157T3 DK99302289T DK99302289T DK0952157T3 DK 0952157 T3 DK0952157 T3 DK 0952157T3 DK 99302289 T DK99302289 T DK 99302289T DK 99302289 T DK99302289 T DK 99302289T DK 0952157 T3 DK0952157 T3 DK 0952157T3
Authority
DK
Denmark
Prior art keywords
methylerythromycin
keto
oxime
compounds
formula
Prior art date
Application number
DK99302289T
Other languages
English (en)
Inventor
Yong-Jin Wu
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK0952157T3 publication Critical patent/DK0952157T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Cephalosporin Compounds (AREA)
DK99302289T 1998-04-24 1999-03-25 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin DK0952157T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8292298P 1998-04-24 1998-04-24

Publications (1)

Publication Number Publication Date
DK0952157T3 true DK0952157T3 (da) 2003-10-13

Family

ID=22174315

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99302289T DK0952157T3 (da) 1998-04-24 1999-03-25 9a, 11b-dehydroderivater af 9-oxim-3-keto-6-0-methylerythromycin

Country Status (11)

Country Link
US (1) US6482801B2 (da)
EP (1) EP0952157B1 (da)
JP (1) JP3432448B2 (da)
AT (1) ATE243219T1 (da)
BR (1) BR9902049A (da)
CA (1) CA2270124C (da)
DE (1) DE69908855T2 (da)
DK (1) DK0952157T3 (da)
ES (1) ES2199524T3 (da)
MX (1) MXPA99003849A (da)
PT (1) PT952157E (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100710605B1 (ko) * 1999-04-16 2007-04-24 코산 바이오사이언시즈, 인코포레이티드 매크롤라이드 항감염제
CN102459296B (zh) * 2009-05-27 2014-10-29 沃克哈特研究中心 具有抗微生物活性的酮内酯类化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69127457T2 (de) 1990-11-28 1998-01-22 Taisho Pharmaceutical Co., Ltd., Tokio/Tokyo 6-0-methylerythromycin a-derivat
US5591837A (en) * 1992-04-22 1997-01-07 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide a derivative
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
DE69631609T2 (de) * 1995-11-08 2005-01-05 Abbott Laboratories, Abbott Park Tricyclische erythromycinderivate
WO1998009978A1 (en) 1996-09-04 1998-03-12 Abbott Laboratories 6-o-substituted ketolides having antibacterial activity
PA8461401A1 (es) * 1997-10-29 2000-05-24 Pfizer Prod Inc Derivados de eritromicina triciclicos
WO1999062920A1 (en) * 1998-06-03 1999-12-09 Pfizer Products Inc. Tricyclic 3-keto derivatives of 6-o-methylerythromycin

Also Published As

Publication number Publication date
US6482801B2 (en) 2002-11-19
MXPA99003849A (es) 2003-09-23
ES2199524T3 (es) 2004-02-16
ATE243219T1 (de) 2003-07-15
PT952157E (pt) 2003-11-28
JPH11322777A (ja) 1999-11-24
EP0952157A1 (en) 1999-10-27
CA2270124A1 (en) 1999-10-24
BR9902049A (pt) 2000-05-02
EP0952157B1 (en) 2003-06-18
CA2270124C (en) 2002-07-09
JP3432448B2 (ja) 2003-08-04
DE69908855T2 (de) 2004-05-19
US20010016574A1 (en) 2001-08-23
DE69908855D1 (de) 2003-07-24

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