DK0937100T3 - En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf - Google Patents

En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf

Info

Publication number
DK0937100T3
DK0937100T3 DK97909496T DK97909496T DK0937100T3 DK 0937100 T3 DK0937100 T3 DK 0937100T3 DK 97909496 T DK97909496 T DK 97909496T DK 97909496 T DK97909496 T DK 97909496T DK 0937100 T3 DK0937100 T3 DK 0937100T3
Authority
DK
Denmark
Prior art keywords
crystalline form
polymorphic crystalline
fluticasone propionate
new polymorphic
preparation
Prior art date
Application number
DK97909496T
Other languages
Danish (da)
English (en)
Inventor
Simon Murray Cooper
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DK0937100T3 publication Critical patent/DK0937100T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Disintegrating Or Milling (AREA)
  • Formation And Processing Of Food Products (AREA)
DK97909496T 1996-10-24 1997-10-23 En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf DK0937100T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9622173.4A GB9622173D0 (en) 1996-10-24 1996-10-24 Particulate Products
PCT/GB1997/002929 WO1998017676A1 (en) 1996-10-24 1997-10-23 A novel polymorphic crystalline form of fluticasone propionate, a method for its production and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
DK0937100T3 true DK0937100T3 (da) 2003-09-01

Family

ID=10801903

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97909496T DK0937100T3 (da) 1996-10-24 1997-10-23 En ny polymorfisk krystallinsk form af fluticasonpropionat, fremgangsmåder til fremstilling deraf og farmaceutiske præparater deraf

Country Status (13)

Country Link
US (1) US6406718B1 (ja)
EP (1) EP0937100B1 (ja)
JP (1) JP2001502350A (ja)
AT (1) ATE240345T1 (ja)
AU (1) AU4717197A (ja)
CA (1) CA2269134C (ja)
DE (1) DE69722023T2 (ja)
DK (1) DK0937100T3 (ja)
ES (1) ES2198555T3 (ja)
GB (1) GB9622173D0 (ja)
PE (1) PE68099A1 (ja)
PT (1) PT937100E (ja)
WO (1) WO1998017676A1 (ja)

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US9815865B2 (en) 2013-01-07 2017-11-14 Nicox Ophthalmics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof
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US8778365B1 (en) 2013-01-31 2014-07-15 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9452173B2 (en) 2013-01-31 2016-09-27 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9446131B2 (en) 2013-01-31 2016-09-20 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
CN104004044A (zh) * 2013-02-25 2014-08-27 武汉诺安药业有限公司 高纯度丙酸氟替卡松制备方法
EP3508196B1 (en) 2014-08-18 2021-07-14 Alkermes Pharma Ireland Limited Aripiprazole prodrug compositions
US10016415B2 (en) 2014-08-18 2018-07-10 Alkermes Pharma Ireland Limited Aripiprazole prodrug compositions
CN108066329B (zh) * 2016-11-11 2021-11-16 江苏恒瑞医药股份有限公司 一种吸入用氟替卡松或其衍生物的微粒的制备方法
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US5658549A (en) 1991-12-12 1997-08-19 Glaxo Group Limited Aerosol formulations containing propellant 134a and fluticasone propionate
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GB9313650D0 (en) 1993-07-01 1993-08-18 Glaxo Group Ltd Method and apparatus for the formation of particles

Also Published As

Publication number Publication date
GB9622173D0 (en) 1996-12-18
ES2198555T3 (es) 2004-02-01
CA2269134C (en) 2007-01-09
WO1998017676A1 (en) 1998-04-30
PT937100E (pt) 2003-09-30
CA2269134A1 (en) 1998-04-30
JP2001502350A (ja) 2001-02-20
DE69722023D1 (de) 2003-06-18
ATE240345T1 (de) 2003-05-15
PE68099A1 (es) 1999-07-19
EP0937100A1 (en) 1999-08-25
US6406718B1 (en) 2002-06-18
AU4717197A (en) 1998-05-15
DE69722023T2 (de) 2004-04-08
EP0937100B1 (en) 2003-05-14

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