DK0700390T3 - Mellemprodukter og fremgangsmåder til syntese af anthrapyrazolonmidler mod cancer - Google Patents

Mellemprodukter og fremgangsmåder til syntese af anthrapyrazolonmidler mod cancer

Info

Publication number
DK0700390T3
DK0700390T3 DK94915874T DK94915874T DK0700390T3 DK 0700390 T3 DK0700390 T3 DK 0700390T3 DK 94915874 T DK94915874 T DK 94915874T DK 94915874 T DK94915874 T DK 94915874T DK 0700390 T3 DK0700390 T3 DK 0700390T3
Authority
DK
Denmark
Prior art keywords
synthesis
intermediates
methods
anticancer drugs
anthrapyrazolone
Prior art date
Application number
DK94915874T
Other languages
Danish (da)
English (en)
Inventor
Joseph Auerbach
Lin-Hua Zhang
Original Assignee
Du Pont Merck Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont Merck Pharma filed Critical Du Pont Merck Pharma
Application granted granted Critical
Publication of DK0700390T3 publication Critical patent/DK0700390T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK94915874T 1993-05-05 1994-04-29 Mellemprodukter og fremgangsmåder til syntese af anthrapyrazolonmidler mod cancer DK0700390T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5703593A 1993-05-05 1993-05-05
US08/142,635 US5393886A (en) 1993-05-05 1993-10-25 Intermediates for the synthesis of anthrapyrazolone anticancer agents
PCT/US1994/004506 WO1994025441A1 (en) 1993-05-05 1994-04-29 Intermediates and methods for the synthesis of anthrapyrazolone anticancer agents

Publications (1)

Publication Number Publication Date
DK0700390T3 true DK0700390T3 (da) 1999-08-02

Family

ID=26735975

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94915874T DK0700390T3 (da) 1993-05-05 1994-04-29 Mellemprodukter og fremgangsmåder til syntese af anthrapyrazolonmidler mod cancer

Country Status (26)

Country Link
US (2) US5393886A (de)
EP (1) EP0700390B1 (de)
JP (1) JPH08509732A (de)
KR (1) KR960701846A (de)
CN (1) CN1122597A (de)
AT (1) ATE173469T1 (de)
AU (1) AU695772B2 (de)
BR (1) BR9406674A (de)
CA (1) CA2162018A1 (de)
CZ (1) CZ281995A3 (de)
DE (1) DE69414706T2 (de)
DK (1) DK0700390T3 (de)
ES (1) ES2128561T3 (de)
FI (1) FI955225A0 (de)
HR (1) HRP940284A2 (de)
HU (1) HUT74737A (de)
IL (1) IL109533A0 (de)
MX (1) MX9403285A (de)
NO (2) NO954405L (de)
NZ (1) NZ266301A (de)
PL (1) PL311634A1 (de)
RU (1) RU2142456C1 (de)
SG (1) SG50510A1 (de)
SK (1) SK137595A3 (de)
TW (1) TW274082B (de)
WO (1) WO1994025441A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1283633B1 (it) * 1996-05-10 1998-04-23 Indena Spa Derivati tassanici loro sintesi e formulazioni che li contengono
WO2008116161A2 (en) 2007-03-22 2008-09-25 The General Hospital Corporation Pyrazoloanthrone and derivatives thereof for the treatment of cancer expressing 'mullerian inhibiting substance' type ii receptor (misrii) and of excess androgen states
US9376406B2 (en) 2011-03-03 2016-06-28 Indiana University Research And Technology Corporation uPAR-uPA interaction inhibitors and methods for treating cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4556654A (en) * 1983-06-28 1985-12-03 Warner-Lambert Company Antimicrobial substituted anthra[1,9-cd]pyrazol-6(2H)-ones
IL69211A (en) * 1982-07-23 1987-01-30 Warner Lambert Co Substituted anthra(1,9-cd)pyrazol-6(2h)-ones,their preparation and pharmaceutical compositions containing them
US4608439A (en) * 1985-04-26 1986-08-26 Warner-Lambert Company Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones
US4672129A (en) * 1986-05-05 1987-06-09 Warner-Lambert Company Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones

Also Published As

Publication number Publication date
HU9503145D0 (en) 1996-01-29
TW274082B (de) 1996-04-11
NO954405D0 (no) 1995-11-03
CA2162018A1 (en) 1994-11-10
NO991975L (no) 1996-01-05
SG50510A1 (en) 1998-07-20
NO954405L (no) 1996-01-05
FI955225A (fi) 1995-11-01
HRP940284A2 (en) 1997-04-30
FI955225A0 (fi) 1995-11-01
ATE173469T1 (de) 1998-12-15
SK137595A3 (en) 1998-12-02
JPH08509732A (ja) 1996-10-15
US5393886A (en) 1995-02-28
MX9403285A (es) 1995-01-31
DE69414706T2 (de) 1999-04-08
RU2142456C1 (ru) 1999-12-10
CN1122597A (zh) 1996-05-15
EP0700390A1 (de) 1996-03-13
NO991975D0 (no) 1999-04-26
AU6773194A (en) 1994-11-21
NZ266301A (en) 1997-05-26
ES2128561T3 (es) 1999-05-16
US5618944A (en) 1997-04-08
AU695772B2 (en) 1998-08-20
CZ281995A3 (en) 1996-03-13
WO1994025441A1 (en) 1994-11-10
HUT74737A (en) 1997-02-28
DE69414706D1 (de) 1998-12-24
PL311634A1 (en) 1996-03-04
KR960701846A (ko) 1996-03-28
IL109533A0 (en) 1994-08-26
BR9406674A (pt) 1996-03-19
EP0700390B1 (de) 1998-11-18

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