NO991975L - Mellomprodukter og metoder for syntese av anthrapyrazolonanticancermidler - Google Patents

Mellomprodukter og metoder for syntese av anthrapyrazolonanticancermidler

Info

Publication number
NO991975L
NO991975L NO991975A NO991975A NO991975L NO 991975 L NO991975 L NO 991975L NO 991975 A NO991975 A NO 991975A NO 991975 A NO991975 A NO 991975A NO 991975 L NO991975 L NO 991975L
Authority
NO
Norway
Prior art keywords
synthesis
anticancer agents
intermediates
methods
anthrapyrazolone
Prior art date
Application number
NO991975A
Other languages
English (en)
Other versions
NO991975D0 (no
Inventor
Lin-Hua Zhang
Joseph Auerbach
Original Assignee
Du Pont Merck Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Publication of NO991975L publication Critical patent/NO991975L/no
Application filed by Du Pont Merck Pharma filed Critical Du Pont Merck Pharma
Publication of NO991975D0 publication Critical patent/NO991975D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Fremgangsmåte for fremstilling av forbindelser, innbefattende 5-klor-2-[2-[[(4- metylfenyl)sulfonyl]oksy]etyl]-7-[2,4,6-trimetylfenyl)metoksy]anthra[l,9-cd]pyrazol- 6(2H)-on og analoger derav som er anvendbare som mellomprodukter for syntesen av anthrapyrazolon-anticancermidler, innbefattende losoxantron.
NO991975A 1993-05-05 1999-04-26 Mellomprodukter og metoder for syntese av anthrapyrazolonanticancermidler NO991975D0 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5703593A 1993-05-05 1993-05-05
US08/142,635 US5393886A (en) 1993-05-05 1993-10-25 Intermediates for the synthesis of anthrapyrazolone anticancer agents
PCT/US1994/004506 WO1994025441A1 (en) 1993-05-05 1994-04-29 Intermediates and methods for the synthesis of anthrapyrazolone anticancer agents

Publications (2)

Publication Number Publication Date
NO991975L true NO991975L (no) 1996-01-05
NO991975D0 NO991975D0 (no) 1999-04-26

Family

ID=26735975

Family Applications (2)

Application Number Title Priority Date Filing Date
NO954405A NO954405L (no) 1993-05-05 1995-11-03 Mellomprodukter og metoder for syntese av anthrapyrazolon-anticancermidler
NO991975A NO991975D0 (no) 1993-05-05 1999-04-26 Mellomprodukter og metoder for syntese av anthrapyrazolonanticancermidler

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO954405A NO954405L (no) 1993-05-05 1995-11-03 Mellomprodukter og metoder for syntese av anthrapyrazolon-anticancermidler

Country Status (26)

Country Link
US (2) US5393886A (no)
EP (1) EP0700390B1 (no)
JP (1) JPH08509732A (no)
KR (1) KR960701846A (no)
CN (1) CN1122597A (no)
AT (1) ATE173469T1 (no)
AU (1) AU695772B2 (no)
BR (1) BR9406674A (no)
CA (1) CA2162018A1 (no)
CZ (1) CZ281995A3 (no)
DE (1) DE69414706T2 (no)
DK (1) DK0700390T3 (no)
ES (1) ES2128561T3 (no)
FI (1) FI955225A0 (no)
HR (1) HRP940284A2 (no)
HU (1) HUT74737A (no)
IL (1) IL109533A0 (no)
MX (1) MX9403285A (no)
NO (2) NO954405L (no)
NZ (1) NZ266301A (no)
PL (1) PL311634A1 (no)
RU (1) RU2142456C1 (no)
SG (1) SG50510A1 (no)
SK (1) SK137595A3 (no)
TW (1) TW274082B (no)
WO (1) WO1994025441A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1283633B1 (it) * 1996-05-10 1998-04-23 Indena Spa Derivati tassanici loro sintesi e formulazioni che li contengono
WO2008116161A2 (en) 2007-03-22 2008-09-25 The General Hospital Corporation Pyrazoloanthrone and derivatives thereof for the treatment of cancer expressing 'mullerian inhibiting substance' type ii receptor (misrii) and of excess androgen states
US9376406B2 (en) 2011-03-03 2016-06-28 Indiana University Research And Technology Corporation uPAR-uPA interaction inhibitors and methods for treating cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL69211A (en) * 1982-07-23 1987-01-30 Warner Lambert Co Substituted anthra(1,9-cd)pyrazol-6(2h)-ones,their preparation and pharmaceutical compositions containing them
US4556654A (en) * 1983-06-28 1985-12-03 Warner-Lambert Company Antimicrobial substituted anthra[1,9-cd]pyrazol-6(2H)-ones
US4608439A (en) * 1985-04-26 1986-08-26 Warner-Lambert Company Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones
US4672129A (en) * 1986-05-05 1987-06-09 Warner-Lambert Company Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones

Also Published As

Publication number Publication date
HRP940284A2 (en) 1997-04-30
NO954405D0 (no) 1995-11-03
PL311634A1 (en) 1996-03-04
HU9503145D0 (en) 1996-01-29
DK0700390T3 (da) 1999-08-02
NO954405L (no) 1996-01-05
SK137595A3 (en) 1998-12-02
JPH08509732A (ja) 1996-10-15
EP0700390B1 (en) 1998-11-18
CN1122597A (zh) 1996-05-15
FI955225A (fi) 1995-11-01
ES2128561T3 (es) 1999-05-16
KR960701846A (ko) 1996-03-28
NZ266301A (en) 1997-05-26
IL109533A0 (en) 1994-08-26
MX9403285A (es) 1995-01-31
RU2142456C1 (ru) 1999-12-10
US5618944A (en) 1997-04-08
ATE173469T1 (de) 1998-12-15
WO1994025441A1 (en) 1994-11-10
HUT74737A (en) 1997-02-28
CA2162018A1 (en) 1994-11-10
DE69414706D1 (de) 1998-12-24
BR9406674A (pt) 1996-03-19
AU695772B2 (en) 1998-08-20
DE69414706T2 (de) 1999-04-08
EP0700390A1 (en) 1996-03-13
US5393886A (en) 1995-02-28
FI955225A0 (fi) 1995-11-01
SG50510A1 (en) 1998-07-20
TW274082B (no) 1996-04-11
NO991975D0 (no) 1999-04-26
CZ281995A3 (en) 1996-03-13
AU6773194A (en) 1994-11-21

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