DE69918050D1 - Verfahren zur herstellung von (2r, 3s)-amino-1,2-oxiran - Google Patents
Verfahren zur herstellung von (2r, 3s)-amino-1,2-oxiranInfo
- Publication number
- DE69918050D1 DE69918050D1 DE69918050T DE69918050T DE69918050D1 DE 69918050 D1 DE69918050 D1 DE 69918050D1 DE 69918050 T DE69918050 T DE 69918050T DE 69918050 T DE69918050 T DE 69918050T DE 69918050 D1 DE69918050 D1 DE 69918050D1
- Authority
- DE
- Germany
- Prior art keywords
- amino
- phenylbutane
- compound
- quaternary ammonium
- ammonium salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/36—Compounds containing oxirane rings with hydrocarbon radicals, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
- C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
- C07C211/27—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring having amino groups linked to the six-membered aromatic ring by saturated carbon chains
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
- C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
- C07C211/29—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Epoxy Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP23854198 | 1998-08-25 | ||
| JP23854198 | 1998-08-25 | ||
| PCT/JP1999/004579 WO2000010986A1 (fr) | 1998-08-25 | 1999-08-25 | Procede de preparation de (2r, 3s)-3-amino-1,2-oxirane |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69918050D1 true DE69918050D1 (de) | 2004-07-22 |
| DE69918050T2 DE69918050T2 (de) | 2005-06-30 |
Family
ID=17031796
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69918050T Expired - Fee Related DE69918050T2 (de) | 1998-08-25 | 1999-08-25 | Verfahren zur herstellung von (2r,3s)-3-amino-1,2-oxiran |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US6278002B1 (de) |
| EP (1) | EP1029856B1 (de) |
| KR (1) | KR20010031394A (de) |
| AT (1) | ATE269314T1 (de) |
| CA (1) | CA2306741A1 (de) |
| DE (1) | DE69918050T2 (de) |
| WO (1) | WO2000010986A1 (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2369356B (en) * | 2000-09-18 | 2004-02-04 | Phoenix Chemicals Ltd | Process |
| KR20030089948A (ko) * | 2002-05-20 | 2003-11-28 | 삼성정밀화학 주식회사 | (ｒ)-3,4-에폭시-1-부탄올의 제조방법 |
| DK2089371T3 (da) | 2006-11-09 | 2011-05-16 | Tibotec Pharm Ltd | Fremstillingsmåde til fremstilling af hexahydrofuro[2,3-b]furan-3-OL |
| MX2009011574A (es) | 2007-04-27 | 2009-11-09 | Tibotec Pharm Ltd | Metodos para la preparacion de derivados de n-isobutil-n-(2-hidrox i-3-amino-4-fenilbutil)-p-nitrobencensulfonilamida. |
| ES2310143B1 (es) * | 2007-06-15 | 2010-02-08 | Universitat Jaume I | Inhibidores de cisteina proteasas. |
| EP2288593A1 (de) * | 2008-05-08 | 2011-03-02 | Ranbaxy Laboratories Limited | Verfahren zur herstellung von 3,4-epoxy-2-amino-1-substituierten butanderivaten und zwischenprodukte dafür |
| TWI482775B (zh) | 2008-09-01 | 2015-05-01 | Tibotec Pharm Ltd | 用於製備（３ｒ，３ａｓ，６ａｒ）－六氫呋喃并〔２，３－ｂ〕呋喃－３－基（１ｓ，２ｒ）－３－〔〔（４－胺基苯基）磺醯基〕（異丁基）胺基〕－１－苯甲基－２－羥基丙基胺基甲酸酯之方法 |
| US8921415B2 (en) | 2009-01-29 | 2014-12-30 | Mapi Pharma Ltd. | Polymorphs of darunavir |
| PL2528923T3 (pl) | 2010-01-28 | 2015-01-30 | Mapi Pharma Ltd | Sposób wytwarzania darunawiru i pochodnych darunawiru |
| TWI429620B (zh) * | 2011-02-28 | 2014-03-11 | Scinopharm Taiwan Ltd | 還原α－醯氧基硫化物衍生物之方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5475013A (en) * | 1990-11-19 | 1995-12-12 | Monsanto Company | Retroviral protease inhibitors |
| US5559256A (en) * | 1992-07-20 | 1996-09-24 | E. R. Squibb & Sons, Inc. | Aminediol protease inhibitors |
| JPH06260857A (ja) | 1993-03-04 | 1994-09-16 | Mitsubishi Electric Corp | 半導体装置 |
| ES2116513T3 (es) * | 1993-12-06 | 1998-07-16 | Nippon Kayaku Kk | Procedimiento para la preparacion de derivados de eritro-3-amino-1,2-epoxidos opticamente activos. |
| CA2319088A1 (en) | 1998-01-28 | 1999-08-05 | Nippon Kayaku Kabushiki Kaisha | Process for producing optically active threo-3-amino-1,2-epoxy compounds |
-
1999
- 1999-08-25 US US09/530,106 patent/US6278002B1/en not_active Expired - Fee Related
- 1999-08-25 EP EP99940471A patent/EP1029856B1/de not_active Expired - Lifetime
- 1999-08-25 KR KR1020007004411A patent/KR20010031394A/ko not_active Application Discontinuation
- 1999-08-25 CA CA002306741A patent/CA2306741A1/en not_active Abandoned
- 1999-08-25 AT AT99940471T patent/ATE269314T1/de not_active IP Right Cessation
- 1999-08-25 DE DE69918050T patent/DE69918050T2/de not_active Expired - Fee Related
- 1999-08-25 WO PCT/JP1999/004579 patent/WO2000010986A1/ja not_active Application Discontinuation
-
2001
- 2001-05-11 US US09/852,652 patent/US6348615B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP1029856A1 (de) | 2000-08-23 |
| KR20010031394A (ko) | 2001-04-16 |
| EP1029856A4 (de) | 2003-01-22 |
| CA2306741A1 (en) | 2000-03-02 |
| DE69918050T2 (de) | 2005-06-30 |
| ATE269314T1 (de) | 2004-07-15 |
| US6278002B1 (en) | 2001-08-21 |
| WO2000010986A1 (fr) | 2000-03-02 |
| EP1029856B1 (de) | 2004-06-16 |
| US6348615B2 (en) | 2002-02-19 |
| US20010018532A1 (en) | 2001-08-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8339 | Ceased/non-payment of the annual fee |