DE69911203D1 - 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidin-monomethanesulfonat - Google Patents
3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidin-monomethanesulfonatInfo
- Publication number
- DE69911203D1 DE69911203D1 DE69911203T DE69911203T DE69911203D1 DE 69911203 D1 DE69911203 D1 DE 69911203D1 DE 69911203 T DE69911203 T DE 69911203T DE 69911203 T DE69911203 T DE 69911203T DE 69911203 D1 DE69911203 D1 DE 69911203D1
- Authority
- DE
- Germany
- Prior art keywords
- pyrrolidine
- monomethanesulfonat
- methylamino
- benzyl
- ethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- WEWYBOJOBPEIAK-UHFFFAOYSA-N pyrrolidin-1-ylmethanesulfonic acid Chemical compound OS(=O)(=O)CN1CCCC1 WEWYBOJOBPEIAK-UHFFFAOYSA-N 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- KYGZCKSPAKDVKC-UHFFFAOYSA-N Oxolinic acid Chemical compound C1=C2N(CC)C=C(C(O)=O)C(=O)C2=CC2=C1OCO2 KYGZCKSPAKDVKC-UHFFFAOYSA-N 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 238000000746 purification Methods 0.000 abstract 1
- 239000003306 quinoline derived antiinfective agent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8719498P | 1998-05-29 | 1998-05-29 | |
US87194P | 1998-05-29 | ||
US10184898P | 1998-09-25 | 1998-09-25 | |
US101848P | 1998-09-25 | ||
PCT/US1999/011739 WO1999061420A1 (en) | 1998-05-29 | 1999-05-27 | 3-[(1--n-methylamino)ethyl-n-benzyl] pyrrolidine monomethanesulfonate |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69911203D1 true DE69911203D1 (de) | 2003-10-16 |
DE69911203T2 DE69911203T2 (de) | 2004-07-15 |
Family
ID=26776704
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69911203T Expired - Fee Related DE69911203T2 (de) | 1998-05-29 | 1999-05-27 | 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidin-monomethanesulfonat |
Country Status (10)
Country | Link |
---|---|
US (1) | US6127400A (de) |
EP (1) | EP1082300B1 (de) |
JP (1) | JP2002516308A (de) |
AT (1) | ATE249432T1 (de) |
AU (1) | AU4211799A (de) |
DE (1) | DE69911203T2 (de) |
DK (1) | DK1082300T3 (de) |
ES (1) | ES2207229T3 (de) |
PT (1) | PT1082300E (de) |
WO (1) | WO1999061420A1 (de) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9820405D0 (en) * | 1998-09-18 | 1998-11-11 | Smithkline Beecham Plc | Process |
GB9920917D0 (en) | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel process |
GB9920919D0 (en) | 1999-09-03 | 1999-11-10 | Sb Pharmco Inc | Novel compound |
KR100517638B1 (ko) | 2002-04-08 | 2005-09-28 | 주식회사 엘지생명과학 | 게미플록사신 산염의 새로운 제조방법 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3390180A (en) * | 1965-04-05 | 1968-06-25 | Celanese Corp | Purification of bis (ortho-diamino-phenyl) compounds |
US3436420A (en) * | 1967-05-02 | 1969-04-01 | Millmaster Onyx Corp | Process of making aliphatic amines |
US3927102A (en) * | 1974-08-21 | 1975-12-16 | Texaco Inc | Separation and recovery of secondary alkyl primary amines |
DE3685157D1 (de) * | 1985-06-26 | 1992-06-11 | Daiichi Seiyaku Co | Pyridoncarbonsaeurederivate. |
US5258528A (en) * | 1990-11-30 | 1993-11-02 | Warner-Lambert Company | Individual stereoisomers of pyrrolidine methanamines substituted on the ring nitrogen by a 1-phenylethyl group |
US5130490A (en) * | 1991-11-25 | 1992-07-14 | Occidental Chemical Corporation | Purification of 3,5-diaminobenzotrifluoride by selective precipitation of the hydrochloride salt |
CA2160124A1 (en) * | 1993-05-06 | 1994-11-24 | William W. Mcwhorter | Optically active 3-(1-(alkylamino)) alkyl pyrrolidines |
IL116281A (en) * | 1995-12-07 | 1999-06-20 | Chemagis Ltd | Process for the purification of (rr,ss)-2-dimethylaminomethyl-1-(3-methoxyphenyl) cyclohexanol and its salts |
JPH10204058A (ja) * | 1997-01-24 | 1998-08-04 | Takasago Internatl Corp | 光学活性ピロリジン誘導体の製造方法 |
-
1999
- 1999-05-27 US US09/320,939 patent/US6127400A/en not_active Expired - Fee Related
- 1999-05-27 AU AU42117/99A patent/AU4211799A/en not_active Abandoned
- 1999-05-27 JP JP2000550826A patent/JP2002516308A/ja active Pending
- 1999-05-27 PT PT99925929T patent/PT1082300E/pt unknown
- 1999-05-27 EP EP99925929A patent/EP1082300B1/de not_active Expired - Lifetime
- 1999-05-27 WO PCT/US1999/011739 patent/WO1999061420A1/en active IP Right Grant
- 1999-05-27 AT AT99925929T patent/ATE249432T1/de not_active IP Right Cessation
- 1999-05-27 DE DE69911203T patent/DE69911203T2/de not_active Expired - Fee Related
- 1999-05-27 ES ES99925929T patent/ES2207229T3/es not_active Expired - Lifetime
- 1999-05-27 DK DK99925929T patent/DK1082300T3/da active
Also Published As
Publication number | Publication date |
---|---|
EP1082300B1 (de) | 2003-09-10 |
DK1082300T3 (da) | 2003-12-15 |
AU4211799A (en) | 1999-12-13 |
DE69911203T2 (de) | 2004-07-15 |
EP1082300A1 (de) | 2001-03-14 |
WO1999061420A1 (en) | 1999-12-02 |
US6127400A (en) | 2000-10-03 |
JP2002516308A (ja) | 2002-06-04 |
ATE249432T1 (de) | 2003-09-15 |
ES2207229T3 (es) | 2004-05-16 |
PT1082300E (pt) | 2004-02-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |