DE69609192T2 - Imidazo(1,2-a)quinoxalin-4-amine als adenosin-antagonisten, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen - Google Patents

Imidazo(1,2-a)quinoxalin-4-amine als adenosin-antagonisten, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen

Info

Publication number
DE69609192T2
DE69609192T2 DE69609192T DE69609192T DE69609192T2 DE 69609192 T2 DE69609192 T2 DE 69609192T2 DE 69609192 T DE69609192 T DE 69609192T DE 69609192 T DE69609192 T DE 69609192T DE 69609192 T2 DE69609192 T2 DE 69609192T2
Authority
DE
Germany
Prior art keywords
quinoxalin
pharmaceutical compositions
compositions containing
pct
imidazo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69609192T
Other languages
English (en)
Other versions
DE69609192D1 (de
Inventor
Stefano Ceccarelli
Sergio Zanarella
Maria Altobelli
Alessandro Alessandra D
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Biomedica Foscama Industria Chimico Farmaceutica SpA
Original Assignee
Biomedica Foscama Industria Chimico Farmaceutica SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biomedica Foscama Industria Chimico Farmaceutica SpA filed Critical Biomedica Foscama Industria Chimico Farmaceutica SpA
Application granted granted Critical
Publication of DE69609192D1 publication Critical patent/DE69609192D1/de
Publication of DE69609192T2 publication Critical patent/DE69609192T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE69609192T 1995-11-24 1996-11-22 Imidazo(1,2-a)quinoxalin-4-amine als adenosin-antagonisten, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen Expired - Fee Related DE69609192T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT95MI002446A IT1276167B1 (it) 1995-11-24 1995-11-24 Imidazo(1,2-alfa)chinossalin-4-ammine attivi come antagonisti adenosinici,procedimento per la loro preparazione e loro composizioni
PCT/IB1996/001291 WO1997019079A1 (en) 1995-11-24 1996-11-22 IMIDAZO[1,2-a]QUINOXALIN-4-AMINES ACTIVE AS ADENOSINE ANTAGONISTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF

Publications (2)

Publication Number Publication Date
DE69609192D1 DE69609192D1 (de) 2000-08-10
DE69609192T2 true DE69609192T2 (de) 2001-03-22

Family

ID=11372590

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69609192T Expired - Fee Related DE69609192T2 (de) 1995-11-24 1996-11-22 Imidazo(1,2-a)quinoxalin-4-amine als adenosin-antagonisten, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen

Country Status (9)

Country Link
US (1) US6124287A (de)
EP (1) EP0865442B1 (de)
AT (1) ATE194347T1 (de)
DE (1) DE69609192T2 (de)
ES (1) ES2149504T3 (de)
GR (1) GR3034354T3 (de)
IT (1) IT1276167B1 (de)
PT (1) PT865442E (de)
WO (1) WO1997019079A1 (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6635626B1 (en) 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
WO1999045009A1 (en) * 1998-03-04 1999-09-10 Bristol-Myers Squibb Company Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
WO2002028860A2 (en) 2000-10-03 2002-04-11 Bristol-Myers Squibb Company Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
US6869956B2 (en) 2000-10-03 2005-03-22 Bristol-Myers Squibb Company Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
CN100386326C (zh) * 2003-10-22 2008-05-07 中国人民解放军军事医学科学院毒物药物研究所 1-羟甲基咪唑并[1，2-a]喹喔啉化合物及其应用
ATE539079T1 (de) * 2006-03-23 2012-01-15 Novartis Ag Imidazochinoxalinverbindungen als immunmodulatoren
DE102006039912A1 (de) * 2006-08-25 2008-03-20 Bayer Healthcare Ag Substituierte Spirotetronsäuren und ihre Verwendung
KR101563103B1 (ko) * 2006-12-13 2015-10-23 아스카 세이야쿠 가부시키가이샤 퀴녹살린 유도체
EP1972629A1 (de) 2007-03-23 2008-09-24 Mutabilis SA Neue Imidazoloheteroarylderivate mit antibakteriellen Eigenschaften
ITMI20072230A1 (it) * 2007-11-23 2009-05-24 Campagnolo Srl Dispositivo di comando per bicicletta con manubrio ricurvo
WO2017037604A1 (en) * 2015-08-28 2017-03-09 Bheema Rao Paraselli Novel fyn kinase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4229452A (en) * 1977-01-07 1980-10-21 Westwood Pharmaceuticals, Inc. Treatment of inflammatory disorders with 4-trifluoromethylimidazo[1,2-a]quinoxaline
US4780464A (en) * 1986-12-08 1988-10-25 Warner-Lambert Company (1,2,4)triazolo(4,3-a)quinoxaline-4-amines
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
BR9406034A (pt) * 1993-03-31 1996-01-02 Basf Ag Derivados de imidazoloquinoxalinonas como antagonistas de eaa.

Also Published As

Publication number Publication date
ES2149504T3 (es) 2000-11-01
US6124287A (en) 2000-09-26
DE69609192D1 (de) 2000-08-10
PT865442E (pt) 2000-10-31
ITMI952446A1 (it) 1997-05-24
ITMI952446A0 (de) 1995-11-24
WO1997019079A1 (en) 1997-05-29
EP0865442A1 (de) 1998-09-23
IT1276167B1 (it) 1997-10-27
EP0865442B1 (de) 2000-07-05
ATE194347T1 (de) 2000-07-15
GR3034354T3 (en) 2000-12-29

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee