DE69606677T2 - Eine Trifluormethylsulfonylphenyl- oder Trifluormethylsulfinylphenylgruppe enthaltende 2-Cyan-3-hydroxy-propenamidderivate, Verfahren zu ihrer Herstellung, ihre Anwendung als Arzneimittel und diese enthaltende pharmazeutische Zusammensetzungen - Google Patents
Eine Trifluormethylsulfonylphenyl- oder Trifluormethylsulfinylphenylgruppe enthaltende 2-Cyan-3-hydroxy-propenamidderivate, Verfahren zu ihrer Herstellung, ihre Anwendung als Arzneimittel und diese enthaltende pharmazeutische ZusammensetzungenInfo
- Publication number
- DE69606677T2 DE69606677T2 DE69606677T DE69606677T DE69606677T2 DE 69606677 T2 DE69606677 T2 DE 69606677T2 DE 69606677 T DE69606677 T DE 69606677T DE 69606677 T DE69606677 T DE 69606677T DE 69606677 T2 DE69606677 T2 DE 69606677T2
- Authority
- DE
- Germany
- Prior art keywords
- cyano
- hydroxy
- trifluoromethylsulfonylphenyl
- medicaments
- processes
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
- C07C317/38—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring with the nitrogen atom of at least one amino group being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfones
- C07C317/40—Y being a hydrogen or a carbon atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9520092.9A GB9520092D0 (en) | 1995-10-02 | 1995-10-02 | Chemical compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69606677D1 DE69606677D1 (de) | 2000-03-23 |
DE69606677T2 true DE69606677T2 (de) | 2000-08-17 |
Family
ID=10781638
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69606677T Expired - Fee Related DE69606677T2 (de) | 1995-10-02 | 1996-10-01 | Eine Trifluormethylsulfonylphenyl- oder Trifluormethylsulfinylphenylgruppe enthaltende 2-Cyan-3-hydroxy-propenamidderivate, Verfahren zu ihrer Herstellung, ihre Anwendung als Arzneimittel und diese enthaltende pharmazeutische Zusammensetzungen |
Country Status (10)
Country | Link |
---|---|
US (1) | US5693844A (de) |
EP (1) | EP0767167B1 (de) |
JP (1) | JPH09132559A (de) |
AT (1) | ATE189810T1 (de) |
DE (1) | DE69606677T2 (de) |
DK (1) | DK0767167T3 (de) |
ES (1) | ES2143159T3 (de) |
GB (1) | GB9520092D0 (de) |
GR (1) | GR3033175T3 (de) |
PT (1) | PT767167E (de) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1325380A (zh) * | 1998-09-11 | 2001-12-05 | 味之素株式会社 | 苯衍生物和它们的药物用途 |
US8686048B2 (en) | 2010-05-06 | 2014-04-01 | Rhizen Pharmaceuticals Sa | Immunomodulator and anti-inflammatory compounds |
US20140031383A1 (en) | 2011-02-08 | 2014-01-30 | Dana-Farber Cancer Institute, Inc. | Methods for treatment of melanoma |
TN2016000197A1 (en) | 2013-11-22 | 2017-10-06 | Genzyme Corp | Novel methods for treating neurodegenerative diseases. |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1116382B (it) * | 1977-11-30 | 1986-02-10 | Sigma Tau Ind Farmaceuti | Metodo di preparazione industriale dell'acido rs-beta-benzoilamino isobutirrico |
IT1097280B (it) * | 1978-06-26 | 1985-08-31 | Montedison Spa | Pigmenti bismetinici |
US4710514A (en) * | 1982-05-04 | 1987-12-01 | Sumitomo Chemical Company, Limited | Fungicidal carbamates and thiolcarbamates |
US4946867A (en) * | 1987-09-07 | 1990-08-07 | Sumitomo Chemical Company, Limited | Cyanoacetamide derivative, and plant disease protectant comprising the same as an active ingredient |
DK0527736T3 (da) * | 1990-05-18 | 1997-10-20 | Hoechst Ag | Isoxazol-4-carboxylsyreamider og hydroxyalkyliden-cyanoacetamider, lægemidler indeholdende disse forbindelser og anvendelsen af disse lægemidler. |
IL99811A (en) * | 1990-10-30 | 1996-03-31 | Roussel Uclaf | 3-Cycloalkyl-propanamides, tautomeric forms of these, their salts, method of preparation, use as drugs and preparations containing them |
IL102790A (en) * | 1991-09-17 | 1996-01-31 | Roussel Uclaf | History of 3-cycloalkyl-prop-2-anamide |
GB9200275D0 (en) * | 1992-01-08 | 1992-02-26 | Roussel Lab Ltd | Chemical compounds |
GB9313365D0 (en) * | 1993-06-29 | 1993-08-11 | Roussel Lab Ltd | Chemical compounds |
-
1995
- 1995-10-02 GB GBGB9520092.9A patent/GB9520092D0/en active Pending
-
1996
- 1996-09-26 US US08/721,500 patent/US5693844A/en not_active Expired - Fee Related
- 1996-10-01 DE DE69606677T patent/DE69606677T2/de not_active Expired - Fee Related
- 1996-10-01 DK DK96402091T patent/DK0767167T3/da active
- 1996-10-01 ES ES96402091T patent/ES2143159T3/es not_active Expired - Lifetime
- 1996-10-01 EP EP96402091A patent/EP0767167B1/de not_active Expired - Lifetime
- 1996-10-01 AT AT96402091T patent/ATE189810T1/de not_active IP Right Cessation
- 1996-10-01 PT PT96402091T patent/PT767167E/pt unknown
- 1996-10-02 JP JP8279859A patent/JPH09132559A/ja not_active Withdrawn
-
2000
- 2000-04-07 GR GR20000400868T patent/GR3033175T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DK0767167T3 (da) | 2000-07-24 |
EP0767167A1 (de) | 1997-04-09 |
JPH09132559A (ja) | 1997-05-20 |
DE69606677D1 (de) | 2000-03-23 |
GR3033175T3 (en) | 2000-08-31 |
EP0767167B1 (de) | 2000-02-16 |
ATE189810T1 (de) | 2000-03-15 |
GB9520092D0 (en) | 1995-12-06 |
US5693844A (en) | 1997-12-02 |
PT767167E (pt) | 2000-06-30 |
ES2143159T3 (es) | 2000-05-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8327 | Change in the person/name/address of the patent owner |
Owner name: AVENTIS PHARMA S.A., ANTONY CEDEX, FR |
|
8339 | Ceased/non-payment of the annual fee |