DE69502539T2 - Sarpogrelat enthaltende opthalmologische Zubereitungen zur Senkung des intraokularen Druckes - Google Patents
Sarpogrelat enthaltende opthalmologische Zubereitungen zur Senkung des intraokularen DruckesInfo
- Publication number
- DE69502539T2 DE69502539T2 DE69502539T DE69502539T DE69502539T2 DE 69502539 T2 DE69502539 T2 DE 69502539T2 DE 69502539 T DE69502539 T DE 69502539T DE 69502539 T DE69502539 T DE 69502539T DE 69502539 T2 DE69502539 T2 DE 69502539T2
- Authority
- DE
- Germany
- Prior art keywords
- intraocular pressure
- sarpogrelate
- ophthalmic
- salts
- solution
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
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- NLJMYIDDQXHKNR-UHFFFAOYSA-K sodium citrate Chemical compound O.O.[Na+].[Na+].[Na+].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O NLJMYIDDQXHKNR-UHFFFAOYSA-K 0.000 description 1
- 235000019259 sodium dehydroacetate Nutrition 0.000 description 1
- 229940079839 sodium dehydroacetate Drugs 0.000 description 1
- 235000019830 sodium polyphosphate Nutrition 0.000 description 1
- DSOWAKKSGYUMTF-GZOLSCHFSA-M sodium;(1e)-1-(6-methyl-2,4-dioxopyran-3-ylidene)ethanolate Chemical compound [Na+].C\C([O-])=C1/C(=O)OC(C)=CC1=O DSOWAKKSGYUMTF-GZOLSCHFSA-M 0.000 description 1
- 239000004334 sorbic acid Substances 0.000 description 1
- 235000010199 sorbic acid Nutrition 0.000 description 1
- 229940075582 sorbic acid Drugs 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
- 235000010356 sorbitol Nutrition 0.000 description 1
- 201000003826 superficial keratitis Diseases 0.000 description 1
- 230000001629 suppression Effects 0.000 description 1
- 229940127230 sympathomimetic drug Drugs 0.000 description 1
- 229940095064 tartrate Drugs 0.000 description 1
- 238000010998 test method Methods 0.000 description 1
- 230000001225 therapeutic effect Effects 0.000 description 1
- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
- 229940033663 thimerosal Drugs 0.000 description 1
- 229960004605 timolol Drugs 0.000 description 1
- 210000001519 tissue Anatomy 0.000 description 1
- 208000008281 urolithiasis Diseases 0.000 description 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
- 229920002554 vinyl polymer Polymers 0.000 description 1
- 230000004382 visual function Effects 0.000 description 1
- 238000005303 weighing Methods 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
- A61K31/225—Polycarboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8717094 | 1994-03-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69502539D1 DE69502539D1 (de) | 1998-06-25 |
| DE69502539T2 true DE69502539T2 (de) | 1998-10-01 |
Family
ID=13907523
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69502539T Expired - Fee Related DE69502539T2 (de) | 1994-03-18 | 1995-03-15 | Sarpogrelat enthaltende opthalmologische Zubereitungen zur Senkung des intraokularen Druckes |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US5652272A (enExample) |
| EP (1) | EP0686393B1 (enExample) |
| KR (1) | KR100338053B1 (enExample) |
| CN (1) | CN1126072A (enExample) |
| AT (1) | ATE166227T1 (enExample) |
| CA (1) | CA2144810A1 (enExample) |
| DE (1) | DE69502539T2 (enExample) |
| ES (1) | ES2116681T3 (enExample) |
| TW (1) | TW309426B (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5998467A (en) * | 1995-10-25 | 1999-12-07 | Mitsubishi Chemical Corporation | Medicine for oculopathy |
| US6960579B1 (en) | 1998-05-19 | 2005-11-01 | Alcon Manufacturing, Ltd. | Serotonergic 5HT7 receptor compounds for treating ocular and CNS disorders |
| TR200100754T2 (tr) | 1998-09-18 | 2001-10-22 | Alcon Laboratories, Inc. | Glausomanın tedavi edilmesi için serotonerjik 5HT2. |
| AU2001230589A1 (en) * | 2000-02-09 | 2001-08-20 | Mitsubishi Pharma Corporation | Therapeutic and/or preventive agents for optic nerve diseases and retinal diseases |
| CA2397203A1 (en) * | 2000-03-31 | 2001-10-11 | Sandra C. Tobias | Phosphoramidate prodrugs |
| CA2460777A1 (en) * | 2001-09-26 | 2003-04-03 | Mitsubishi Pharma Corporation | Thrombus/thrombogenesis inhibitors |
| JP2005511764A (ja) * | 2001-12-14 | 2005-04-28 | アルコン，インコーポレイテッド | 緑内障の処置のためのアミノアルキルベンゾフラン−５−オール化合物 |
| TW593302B (en) * | 2001-12-20 | 2004-06-21 | Alcon Inc | Novel benzodifuranimidazoline and benzofuranimidazoline derivatives and their use for the treatment of glaucoma |
| WO2004019874A2 (en) * | 2002-08-30 | 2004-03-11 | Alcon, Inc. | Substituted 5-chroman-5-yl-ethylamine compounds and their use for the treatment of glaucoma |
| EP1581209A4 (en) * | 2002-12-13 | 2009-03-11 | Alcon Inc | NEW BENZOPYRAN ANALOGUE AND ITS USE FOR THE TREATMENT OF GLAUKOM |
| US7947295B2 (en) * | 2003-06-13 | 2011-05-24 | Alcon, Inc. | Ophthalmic compositions containing a synergistic combination of two polymers |
| US7914803B2 (en) | 2003-06-13 | 2011-03-29 | Alcon, Inc. | Ophthalmic compositions containing a synergistic combination of three polymers |
| TWI336257B (en) * | 2003-06-13 | 2011-01-21 | Alcon Inc | Ophthalmic compositions containing a synergistic combination of three polymers |
| CA2839930C (en) * | 2003-06-13 | 2016-07-05 | Alcon, Inc. | Ophthalmic compositions containing a synergistic combination of two polymers |
| WO2005053688A1 (en) * | 2003-11-26 | 2005-06-16 | Alcon, Inc. | Substituted furo[2,3-g] indazoles for the treatment of glaucoma |
| US7338972B1 (en) | 2003-12-15 | 2008-03-04 | Alcon, Inc. | Substituted 1-alkylamino-1H-indazoles for the treatment of glaucoma |
| WO2005058911A2 (en) * | 2003-12-15 | 2005-06-30 | Alcon, Inc. | Substituted [1,4]oxazino[2,3-g]indazoles for the treatment of glaucoma |
| US7129257B1 (en) | 2003-12-15 | 2006-10-31 | Alcon, Inc. | Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma |
| US7425572B2 (en) | 2004-12-08 | 2008-09-16 | Alcon, Inc. | Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma |
| TW200744567A (en) * | 2005-09-23 | 2007-12-16 | Alcon Inc | Phenylethylamine analogs and their use for treating glaucoma |
| WO2007149728A2 (en) * | 2006-06-20 | 2007-12-27 | Alcon Research, Ltd. | Aryl and heteroaryl tetrahydrobenzazepine derivatives and their use for treating glaucoma |
| ZA200904917B (en) * | 2007-02-09 | 2010-09-29 | Alcon Inc | Ophthalmic compositions containing a synergistic combination of three polymers |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH02304022A (ja) * | 1989-05-18 | 1990-12-17 | Mitsubishi Kasei Corp | セロトニン拮抗剤 |
-
1995
- 1995-03-15 AT AT95301727T patent/ATE166227T1/de not_active IP Right Cessation
- 1995-03-15 US US08/404,315 patent/US5652272A/en not_active Expired - Fee Related
- 1995-03-15 DE DE69502539T patent/DE69502539T2/de not_active Expired - Fee Related
- 1995-03-15 TW TW084102465A patent/TW309426B/zh active
- 1995-03-15 EP EP95301727A patent/EP0686393B1/en not_active Expired - Lifetime
- 1995-03-15 ES ES95301727T patent/ES2116681T3/es not_active Expired - Lifetime
- 1995-03-16 CA CA002144810A patent/CA2144810A1/en not_active Abandoned
- 1995-03-17 CN CN95103537A patent/CN1126072A/zh active Pending
- 1995-03-17 KR KR1019950005633A patent/KR100338053B1/ko not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2144810A1 (en) | 1995-09-19 |
| KR950031062A (ko) | 1995-12-18 |
| CN1126072A (zh) | 1996-07-10 |
| DE69502539D1 (de) | 1998-06-25 |
| TW309426B (enExample) | 1997-07-01 |
| KR100338053B1 (ko) | 2002-11-23 |
| US5652272A (en) | 1997-07-29 |
| ES2116681T3 (es) | 1998-07-16 |
| EP0686393B1 (en) | 1998-05-20 |
| EP0686393A1 (en) | 1995-12-13 |
| ATE166227T1 (de) | 1998-06-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition | ||
| 8327 | Change in the person/name/address of the patent owner |
Owner name: SENJU PHARMACEUTICAL CO., LTD., OSAKA, JP MITSUBIS |
|
| 8339 | Ceased/non-payment of the annual fee |