DE602006020273D1 - Substituierte heteroarylamidmodulatoren der aktivität des glucokortikoidrezeptors, von ap-1 und/oder von nfkb und anwendung davon - Google Patents

Substituierte heteroarylamidmodulatoren der aktivität des glucokortikoidrezeptors, von ap-1 und/oder von nfkb und anwendung davon

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Publication number
DE602006020273D1
DE602006020273D1 DE602006020273T DE602006020273T DE602006020273D1 DE 602006020273 D1 DE602006020273 D1 DE 602006020273D1 DE 602006020273 T DE602006020273 T DE 602006020273T DE 602006020273 T DE602006020273 T DE 602006020273T DE 602006020273 D1 DE602006020273 D1 DE 602006020273D1
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Germany
Prior art keywords
sup
receptor
corticide
nfkb
modulators
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DE602006020273T
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Inventor
James E Sheppeck
Murali T G Dhar
Arthur M P Doweyko
Lidia M Doweyko
John L Gilmore
David S Weinstein
Hai-Yun Xiao
Bingwei Vera Yang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of DE602006020273D1 publication Critical patent/DE602006020273D1/de
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DE602006020273T 2005-01-13 2006-01-13 Substituierte heteroarylamidmodulatoren der aktivität des glucokortikoidrezeptors, von ap-1 und/oder von nfkb und anwendung davon Active DE602006020273D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US64350905P 2005-01-13 2005-01-13
US11/330,553 US7361654B2 (en) 2005-01-13 2006-01-12 Substituted heteroaryl amide modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
PCT/US2006/001328 WO2006076632A1 (en) 2005-01-13 2006-01-13 SUBSTITUTED HETEROARYL AMIDE MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NFκB ACTIVITY AND USE THEREOF

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DE602006020273D1 true DE602006020273D1 (de) 2011-04-07

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DE602006020273T Active DE602006020273D1 (de) 2005-01-13 2006-01-13 Substituierte heteroarylamidmodulatoren der aktivität des glucokortikoidrezeptors, von ap-1 und/oder von nfkb und anwendung davon

Country Status (6)

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US (1) US7361654B2 (de)
EP (1) EP1896434B1 (de)
JP (1) JP2008526993A (de)
AT (1) ATE499349T1 (de)
DE (1) DE602006020273D1 (de)
WO (1) WO2006076632A1 (de)

Families Citing this family (19)

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Publication number Priority date Publication date Assignee Title
US7253283B2 (en) * 2004-01-16 2007-08-07 Bristol-Myers Squibb Company Tricyclic modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
US7569689B2 (en) * 2004-01-16 2009-08-04 Bristol-Myers Squibb Company Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
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