DE602004020488D1 - Mikroemulsionen von retinoiden und diese enthaltende pharmazeutische zusammensetzungen - Google Patents

Mikroemulsionen von retinoiden und diese enthaltende pharmazeutische zusammensetzungen

Info

Publication number
DE602004020488D1
DE602004020488D1 DE602004020488T DE602004020488T DE602004020488D1 DE 602004020488 D1 DE602004020488 D1 DE 602004020488D1 DE 602004020488 T DE602004020488 T DE 602004020488T DE 602004020488 T DE602004020488 T DE 602004020488T DE 602004020488 D1 DE602004020488 D1 DE 602004020488D1
Authority
DE
Germany
Prior art keywords
microemulsions
retinoids
pharmaceutical compositions
compositions containing
retinoid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602004020488T
Other languages
English (en)
Inventor
Enea Menegatti
Rita Cortesi
Elisabetta Esposito
Pierangelo Bellato
Giovanni Gennari
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fidia Farmaceutici SpA
Original Assignee
Fidia Farmaceutici SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia Farmaceutici SpA filed Critical Fidia Farmaceutici SpA
Publication of DE602004020488D1 publication Critical patent/DE602004020488D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/07—Retinol compounds, e.g. vitamin A
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
DE602004020488T 2003-10-17 2004-10-08 Mikroemulsionen von retinoiden und diese enthaltende pharmazeutische zusammensetzungen Active DE602004020488D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT002019A ITMI20032019A1 (it) 2003-10-17 2003-10-17 Microemulsioni di retinoidi e composizioni farmaceutiche che le contengono
PCT/EP2004/011236 WO2005039532A1 (en) 2003-10-17 2004-10-08 Microemulsions of retinoids, and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
DE602004020488D1 true DE602004020488D1 (de) 2009-05-20

Family

ID=34509450

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602004020488T Active DE602004020488D1 (de) 2003-10-17 2004-10-08 Mikroemulsionen von retinoiden und diese enthaltende pharmazeutische zusammensetzungen

Country Status (12)

Country Link
US (1) US7781489B2 (de)
EP (1) EP1673065B1 (de)
JP (1) JP2007508339A (de)
AT (1) ATE427737T1 (de)
AU (1) AU2004283432B2 (de)
CA (1) CA2542663C (de)
DE (1) DE602004020488D1 (de)
ES (1) ES2322472T3 (de)
IT (1) ITMI20032019A1 (de)
PL (1) PL1673065T3 (de)
SI (1) SI1673065T1 (de)
WO (1) WO2005039532A1 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1592420B1 (de) 2003-01-24 2014-01-01 Stiefel Research Australia Pty Ltd Clindamycinphosphat-schaum
FR2865651B1 (fr) * 2004-01-29 2007-09-28 Fabre Pierre Dermo Cosmetique Compositions topiques associant des fragments de hyaluronate de sodium et un retinoide utiles en dermatologie cosmetique et medicale
FR2894827B1 (fr) * 2005-12-21 2010-10-29 Galderma Res & Dev Preparations pharmaceutiques ou cosmetiques pour application topique et/ou parenterale, leurs procedes de preparation,et leurs utilisations
CA2680606C (en) 2006-03-29 2014-08-05 Wayne State University Liposomal nanoparticles and other formulations of fenretinide for use in therapy and drug delivery
EP1967180A1 (de) * 2007-03-06 2008-09-10 Almirall Hermal GmbH Topische Zusammensetzung enthaltend einen Retinoid-Rezeptor-Agonist
CA2686558A1 (fr) * 2007-05-11 2008-12-11 Galderma Research & Development Preparations pharmaceutiques ou cosmetiques pour application topique et/ou parenterale, leurs procedes de preparation, et leurs utilisations
DE102008034944B4 (de) * 2008-07-26 2017-03-16 Arivine Pharma Ag Mikroemulsion
EP2344198B1 (de) * 2008-09-27 2020-11-04 Jina Pharmaceuticals Inc. Pharmazeutische präparate auf lipidbasis zur topischen verabreichung
CN102438590B (zh) 2009-02-25 2013-07-10 施泰福研究澳大利亚有限公司 局部泡沫组合物
WO2013142247A1 (en) * 2012-03-22 2013-09-26 Precision Dermatology, Inc. Cyclodextrin-based microemulsions, and dermatological uses thereof
US10702604B2 (en) * 2012-06-01 2020-07-07 Galderma Research & Development Lipid nanocapsules comprising a retinoid, nanodispersion and composition containing the same, process for preparing the same and use thereof in dermatology
EP2882865B1 (de) 2012-08-10 2017-09-27 Galderma Research & Development Verfahren zur diagnose von rosacea
US10857080B2 (en) 2013-12-04 2020-12-08 Galderma Research & Development Lipid microcapsules preferably comprising a lipophilic active substance and composition containing same, method for the production thereof, and use of same in dermatology and in cosmetics
WO2016193588A1 (fr) 2015-05-29 2016-12-08 Galderma Research & Development Compositions comprenant au moins un principe actif disperse et des microcapsules lipidiques
EP3308766B1 (de) 2016-10-11 2019-12-25 Ionia Azure AG Kosmetische wasser-in-öl-mikroemulsion

Family Cites Families (20)

* Cited by examiner, † Cited by third party
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IT1212892B (it) * 1983-10-11 1989-11-30 Della Valle Francesco Acido ialuronico ottenuto per mezzodi filtrazione molecolare sprovvisto di attivita' infiammatoria e sua utilizzazione terapeutica
JPS63500456A (ja) * 1985-08-13 1988-02-18 カリフオルニア　バイオテクノロジ−　インコ−ポレイテツド 薬剤に用いるミクロエマルジョン
US5023271A (en) 1985-08-13 1991-06-11 California Biotechnology Inc. Pharmaceutical microemulsions
JPS6245336A (ja) * 1985-08-21 1987-02-27 Toyo Biyuut Kk 乳化組成物
JPS6295132A (ja) * 1985-10-21 1987-05-01 Nippon Saafuakutanto Kogyo Kk 多価アルコ−ル中油型乳化組成物
US5055303A (en) * 1989-01-31 1991-10-08 Kv Pharmaceutical Company Solid controlled release bioadherent emulsions
JPH03293024A (ja) * 1990-04-11 1991-12-24 Nikko Kemikaruzu Kk レシチンが水相に分散して成る油中水型エマルション
US5110606A (en) * 1990-11-13 1992-05-05 Affinity Biotech, Inc. Non-aqueous microemulsions for drug delivery
GB9214634D0 (en) * 1992-07-09 1992-08-19 Lalvani Kartar S A cosmetic or pharmaceutical preparation
US5744155A (en) * 1993-08-13 1998-04-28 Friedman; Doron Bioadhesive emulsion preparations for enhanced drug delivery
JPH1118697A (ja) * 1997-07-09 1999-01-26 Toyo Beauty Kk 含油ゲル状組成物及び水中油型乳化組成物
TWI241915B (en) * 1998-05-11 2005-10-21 Ciba Sc Holding Ag A method of preparing a pharmaceutical end formulation using a nanodispersion
DE19826503A1 (de) * 1998-06-13 1999-12-16 Beiersdorf Ag Kosmetische und dermatologische Zubereitungen mit einem Gehalt an Chitosan und Phospholipiden
JP2000204011A (ja) 1999-01-13 2000-07-25 Human Limited:Kk 殺菌・制菌・消臭・皮膚保水性向上液の製法
JP2001181180A (ja) * 1999-12-24 2001-07-03 Lion Corp 油中水型乳化組成物
JP4430770B2 (ja) * 2000-01-07 2010-03-10 花王株式会社 皮膚弾力性改善剤
AU1987802A (en) * 2000-11-29 2002-06-11 Lyotropic Therapeutics Llc Solvent systems for pharmaceutical agents
ES2316489T3 (es) 2000-12-05 2009-04-16 Childrens Hospital Los Angeles Composiciones farmaceuticas de fenretinida que tienen biodisponibilidad aumentada y metodos de uso de las mismas.
US6551605B2 (en) * 2001-04-06 2003-04-22 Haarmann & Reimer Diesters or polyesters of naphthalene dicarboxylic acid as solubilizer/stabilizer for retinoids
US7820145B2 (en) * 2003-08-04 2010-10-26 Foamix Ltd. Oleaginous pharmaceutical and cosmetic foam

Also Published As

Publication number Publication date
CA2542663C (en) 2012-11-27
EP1673065A1 (de) 2006-06-28
US20070134276A1 (en) 2007-06-14
PL1673065T3 (pl) 2009-09-30
SI1673065T1 (sl) 2009-08-31
EP1673065B1 (de) 2009-04-08
ITMI20032019A1 (it) 2005-04-18
US7781489B2 (en) 2010-08-24
JP2007508339A (ja) 2007-04-05
CA2542663A1 (en) 2005-05-06
ATE427737T1 (de) 2009-04-15
ES2322472T3 (es) 2009-06-22
AU2004283432B2 (en) 2010-02-11
AU2004283432A1 (en) 2005-05-06
WO2005039532A1 (en) 2005-05-06

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