DE60022523D1 - Aminopiperidinderivate als antibakterielles arzneimittel - Google Patents

Aminopiperidinderivate als antibakterielles arzneimittel

Info

Publication number
DE60022523D1
DE60022523D1 DE60022523T DE60022523T DE60022523D1 DE 60022523 D1 DE60022523 D1 DE 60022523D1 DE 60022523 T DE60022523 T DE 60022523T DE 60022523 T DE60022523 T DE 60022523T DE 60022523 D1 DE60022523 D1 DE 60022523D1
Authority
DE
Germany
Prior art keywords
antibacterial drug
aminopiperidine derivatives
derivatives
aminopiperidine
antibacterial
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60022523T
Other languages
English (en)
Other versions
DE60022523T2 (de
Inventor
David Thomas Davies
Andrew Lightfoot
Roger Edward Markwell
Neil David Pearson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Application granted granted Critical
Publication of DE60022523D1 publication Critical patent/DE60022523D1/de
Publication of DE60022523T2 publication Critical patent/DE60022523T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
DE60022523T 1999-07-23 2000-07-17 Aminopiperidinderivate als antibakterielles arzneimittel Expired - Fee Related DE60022523T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9917408 1999-07-23
GBGB9917408.8A GB9917408D0 (en) 1999-07-23 1999-07-23 Compounds
PCT/EP2000/006938 WO2001007432A2 (en) 1999-07-23 2000-07-17 Aminopiperidine derivatives as antibacterials

Publications (2)

Publication Number Publication Date
DE60022523D1 true DE60022523D1 (de) 2005-10-13
DE60022523T2 DE60022523T2 (de) 2006-06-29

Family

ID=10857877

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60022523T Expired - Fee Related DE60022523T2 (de) 1999-07-23 2000-07-17 Aminopiperidinderivate als antibakterielles arzneimittel

Country Status (9)

Country Link
US (2) US7001913B1 (de)
EP (1) EP1214314B1 (de)
JP (1) JP2003505455A (de)
AT (1) ATE304006T1 (de)
AU (1) AU5986200A (de)
DE (1) DE60022523T2 (de)
ES (1) ES2246244T3 (de)
GB (1) GB9917408D0 (de)
WO (1) WO2001007432A2 (de)

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JP2008528604A (ja) * 2005-01-25 2008-07-31 グラクソ グループ リミテッド 抗菌剤
US7709472B2 (en) 2005-01-25 2010-05-04 Glaxo Group Limited Antibacterial agents
WO2006081264A1 (en) 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
MY150958A (en) 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
JO2952B1 (en) * 2005-08-03 2016-03-15 جانسين فارماسوتيكا ان. في Quinoline derivatives acting as antibacterial agents
CA2635126A1 (en) 2006-01-26 2007-08-02 Actelion Pharmaceuticals Ltd Tetrahydropyrane antibiotics
JP2009532504A (ja) 2006-04-06 2009-09-10 グラクソ グループ リミテッド 抗菌薬
KR100760148B1 (ko) 2006-07-19 2007-09-18 주식회사 엘지생활건강 알파-리포산을 안정화시킨 화장료 조성물
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AU2008212999A1 (en) 2007-02-06 2008-08-14 Boehringer Ingelheim International Gmbh Bicyclic heterocycles, drugs containing said compounds, use thereof, and method for production thereof
GB0707706D0 (en) * 2007-04-20 2007-05-30 Glaxo Group Ltd Compounds
EP2005995A1 (de) * 2007-06-22 2008-12-24 Glaxo Group Limited Heterocyclische Verbindungen für die Behandlung von Tuberkulose
CA2711582A1 (en) 2008-02-07 2009-08-13 Boehringer Ingelheim International Gmbh Spirocyclic heterocycles, formulations containing said compounds, use thereof and processes for the preparation thereof
JP2011518149A (ja) 2008-04-15 2011-06-23 アクテリオン ファーマシューティカルズ リミテッド 三環式抗菌剤
JP5739802B2 (ja) 2008-05-13 2015-06-24 アストラゼネカ アクチボラグ ４−（３−クロロ−２−フルオロアニリノ）−７−メトキシ−６−｛［１−（ｎ−メチルカルバモイルメチル）ピペリジン−４−イル］オキシ｝キナゾリンのフマル酸塩
JP5539351B2 (ja) 2008-08-08 2014-07-02 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング シクロヘキシルオキシ置換ヘテロ環、これらの化合物を含有する医薬、およびそれらを生成するための方法
EP2332939A1 (de) 2009-11-26 2011-06-15 Æterna Zentaris GmbH Neuartige Naphthyridinderivate und ihre Verwendung als Kinasehemmer
EP3927703B1 (de) 2019-02-19 2023-04-05 Univerza V Ljubljani Antibakterielle substanzen auf basis monocyclischer fragmente, die mit aminopiperidin-naphthyridin-gerüst gekoppelt sind

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Also Published As

Publication number Publication date
US20060079546A1 (en) 2006-04-13
DE60022523T2 (de) 2006-06-29
ATE304006T1 (de) 2005-09-15
GB9917408D0 (en) 1999-09-22
US7001913B1 (en) 2006-02-21
WO2001007432A8 (en) 2001-09-07
ES2246244T3 (es) 2006-02-16
WO2001007432A3 (en) 2001-05-25
AU5986200A (en) 2001-02-13
JP2003505455A (ja) 2003-02-12
EP1214314B1 (de) 2005-09-07
WO2001007432A2 (en) 2001-02-01
EP1214314A2 (de) 2002-06-19

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee