DE60001182D1 - Erythromycin-Derivate, ihr Verfahren zur Herstellung und ihre Verwendung als Arzneimittel - Google Patents
Erythromycin-Derivate, ihr Verfahren zur Herstellung und ihre Verwendung als ArzneimittelInfo
- Publication number
- DE60001182D1 DE60001182D1 DE60001182T DE60001182T DE60001182D1 DE 60001182 D1 DE60001182 D1 DE 60001182D1 DE 60001182 T DE60001182 T DE 60001182T DE 60001182 T DE60001182 T DE 60001182T DE 60001182 D1 DE60001182 D1 DE 60001182D1
- Authority
- DE
- Germany
- Prior art keywords
- erythromycin derivatives
- medicines
- manufacturing process
- halo
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Oncology (AREA)
- Dermatology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9901292A FR2789392B1 (fr) | 1999-02-04 | 1999-02-04 | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60001182D1 true DE60001182D1 (de) | 2003-02-20 |
DE60001182T2 DE60001182T2 (de) | 2003-10-09 |
Family
ID=9541593
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60001182T Expired - Lifetime DE60001182T2 (de) | 1999-02-04 | 2000-02-03 | Erythromycin-Derivate, ihr Verfahren zur Herstellung und ihre Verwendung als Arzneimittel |
Country Status (8)
Country | Link |
---|---|
US (1) | US6313101B1 (de) |
EP (1) | EP1026170B1 (de) |
JP (2) | JP5019665B2 (de) |
AT (1) | ATE231160T1 (de) |
DE (1) | DE60001182T2 (de) |
DK (1) | DK1026170T3 (de) |
ES (1) | ES2186615T3 (de) |
FR (1) | FR2789392B1 (de) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69933897T2 (de) * | 1998-12-10 | 2007-03-15 | Pfizer Products Inc., Groton | Carbamat- und Carbazatketolid-Antibiotika |
WO2000044761A2 (en) | 1999-01-27 | 2000-08-03 | Pfizer Products Inc. | Ketolide antibiotics |
CZ20013733A3 (cs) | 1999-05-24 | 2002-11-13 | Pfizer Products Inc. | Deriváty 13-methylerythromycinu |
DE19948417A1 (de) * | 1999-10-07 | 2001-04-19 | Morphochem Ag | Imidazol-Derivate und ihre Verwendung als Arzneimittel |
ES2222966T3 (es) | 2000-06-30 | 2005-02-16 | Pfizer Products Inc. | Macrolidos antibioticos. |
US20080287376A1 (en) * | 2004-07-28 | 2008-11-20 | Mohammad Salman | Ketolide Derivatives as Antibacterial Agents |
WO2006046112A2 (en) * | 2004-10-25 | 2006-05-04 | Ranbaxy Laboratories Limited | Ketolide derivatives as antibacterial agents |
CN101917850B (zh) | 2007-10-25 | 2016-01-13 | 森普拉制药公司 | 大环内酯类抗菌剂的制备方法 |
CN102245195B (zh) | 2008-10-24 | 2016-01-13 | 森普拉制药公司 | 使用含三唑的大环内酯的生物防御 |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
JP5914335B2 (ja) | 2009-09-10 | 2016-05-11 | センプラ ファーマシューティカルズ,インコーポレイテッド | マラリア、結核、及びmac病の治療方法 |
KR20130120458A (ko) * | 2010-09-10 | 2013-11-04 | 셈프라 파마슈티컬스, 인크. | 질환을 치료하기 위한 수소결합 형성 플루오로 케토라이드 |
AU2013239696C1 (en) | 2012-03-27 | 2018-11-29 | Cempra Pharmaceuticals, Inc. | Parenteral formulations for administering macrolide antibiotics |
EP2968801B1 (de) | 2013-03-14 | 2018-09-26 | Cempra Pharmaceuticals, Inc. | Verfahren zur behandlung von atemwegserkrankungen und formulierungen dafür |
EP2968384A4 (de) | 2013-03-15 | 2017-02-15 | Cempra Pharmaceuticals, Inc. | Konvergente verfahren zur herstellung antibakterieller makrolidmittel |
CN104860943B (zh) * | 2015-05-18 | 2017-11-17 | 上海毕路得医药科技有限公司 | 5,7‑二氯‑1h‑咪唑并[4,5‑b]吡啶的合成方法 |
CN106432383A (zh) * | 2016-09-14 | 2017-02-22 | 重庆两江药物研发中心有限公司 | 索利霉素及其中间体的制备方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5527780A (en) * | 1992-11-05 | 1996-06-18 | Roussel Uclaf | Erythromycin derivatives |
FR2718450B1 (fr) * | 1994-04-08 | 1997-01-10 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2719587B1 (fr) * | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
FR2732023B1 (fr) * | 1995-03-22 | 1997-04-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2732684B1 (fr) * | 1995-04-06 | 1997-04-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2742757B1 (fr) * | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
-
1999
- 1999-02-04 FR FR9901292A patent/FR2789392B1/fr not_active Expired - Fee Related
-
2000
- 2000-01-31 JP JP2000021454A patent/JP5019665B2/ja not_active Expired - Lifetime
- 2000-02-03 AT AT00400286T patent/ATE231160T1/de not_active IP Right Cessation
- 2000-02-03 DK DK00400286T patent/DK1026170T3/da active
- 2000-02-03 EP EP00400286A patent/EP1026170B1/de not_active Expired - Lifetime
- 2000-02-03 ES ES00400286T patent/ES2186615T3/es not_active Expired - Lifetime
- 2000-02-03 US US09/497,651 patent/US6313101B1/en not_active Expired - Lifetime
- 2000-02-03 DE DE60001182T patent/DE60001182T2/de not_active Expired - Lifetime
-
2010
- 2010-12-08 JP JP2010273652A patent/JP5222348B2/ja not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
FR2789392B1 (fr) | 2001-10-05 |
JP2000229993A (ja) | 2000-08-22 |
FR2789392A1 (fr) | 2000-08-11 |
DK1026170T3 (da) | 2003-05-05 |
EP1026170A1 (de) | 2000-08-09 |
ATE231160T1 (de) | 2003-02-15 |
JP2011136990A (ja) | 2011-07-14 |
ES2186615T3 (es) | 2003-05-16 |
JP5222348B2 (ja) | 2013-06-26 |
EP1026170B1 (de) | 2003-01-15 |
US6313101B1 (en) | 2001-11-06 |
JP5019665B2 (ja) | 2012-09-05 |
DE60001182T2 (de) | 2003-10-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8328 | Change in the person/name/address of the agent |
Representative=s name: PFENNING MEINIG & PARTNER GBR, 80339 MUENCHEN |
|
8328 | Change in the person/name/address of the agent |
Representative=s name: MAIWALD PATENTANWALTSGESELLSCHAFT MBH, 80335 MUENC |