DE3235565A1 - Piperidinderivate, ihre herstellung und verwendung - Google Patents

Piperidinderivate, ihre herstellung und verwendung

Info

Publication number
DE3235565A1
DE3235565A1 DE19823235565 DE3235565A DE3235565A1 DE 3235565 A1 DE3235565 A1 DE 3235565A1 DE 19823235565 DE19823235565 DE 19823235565 DE 3235565 A DE3235565 A DE 3235565A DE 3235565 A1 DE3235565 A1 DE 3235565A1
Authority
DE
Germany
Prior art keywords
formula
compounds
alkyl
hydrogen
arylmethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19823235565
Other languages
German (de)
English (en)
Inventor
Wolfram Dr. 6507 Ingelheim Gaida
Wolfgang Dr. 6200 Wiesbaden Hoefke
Anton Dr. 6503 Mainz-Kastel Mentrup
Ernst-Otto Dr. Renth
Kurt Dr. 6507 Ingelheim Schromm
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim GmbH
Original Assignee
Boehringer Ingelheim GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim GmbH filed Critical Boehringer Ingelheim GmbH
Priority to DE19823235565 priority Critical patent/DE3235565A1/de
Priority to EP83108375A priority patent/EP0104445A3/de
Priority to SU833641410A priority patent/SU1187720A3/ru
Priority to US06/531,842 priority patent/US4539323A/en
Priority to FI833292A priority patent/FI833292A7/fi
Priority to PH29564A priority patent/PH20015A/en
Priority to JP58174020A priority patent/JPS5978187A/ja
Priority to IL69777A priority patent/IL69777A/xx
Priority to CS836919A priority patent/CS235342B2/cs
Priority to GR72505A priority patent/GR78973B/el
Priority to CA000437468A priority patent/CA1215981A/en
Priority to YU01921/83A priority patent/YU192183A/xx
Priority to PL1983243878A priority patent/PL139590B1/pl
Priority to AU19396/83A priority patent/AU561118B2/en
Priority to NO833423A priority patent/NO833423L/no
Priority to DD83255091A priority patent/DD212517A5/de
Priority to DK436583A priority patent/DK436583A/da
Priority to ES525876A priority patent/ES8501762A1/es
Priority to NZ205716A priority patent/NZ205716A/xx
Priority to HU833307A priority patent/HU191637B/hu
Priority to PT77380A priority patent/PT77380B/pt
Priority to ZA837081A priority patent/ZA837081B/xx
Priority to KR1019830004475A priority patent/KR840006222A/ko
Publication of DE3235565A1 publication Critical patent/DE3235565A1/de
Priority to ES534351A priority patent/ES8504182A1/es
Priority to ES534349A priority patent/ES8504180A1/es
Priority to ES534350A priority patent/ES534350A0/es
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DE19823235565 1982-09-25 1982-09-25 Piperidinderivate, ihre herstellung und verwendung Withdrawn DE3235565A1 (de)

Priority Applications (26)

Application Number Priority Date Filing Date Title
DE19823235565 DE3235565A1 (de) 1982-09-25 1982-09-25 Piperidinderivate, ihre herstellung und verwendung
EP83108375A EP0104445A3 (de) 1982-09-25 1983-08-25 Piperidinochinoxalin-Derivate, ihre Herstellung und Verwendung
SU833641410A SU1187720A3 (ru) 1982-09-25 1983-09-13 Способ получени производных пиперидина или их кислотноаддитивных солей
US06/531,842 US4539323A (en) 1982-09-25 1983-09-14 N-[1-(4-Amino-6,7-dialkoxy-2-quinazolinyl)-4-piperidyl]-oxazolidine-2,4-diones
FI833292A FI833292A7 (fi) 1982-09-25 1983-09-15 Piperidiinijohdokset, niiden valmistus ja käyttö.
PH29564A PH20015A (en) 1982-09-25 1983-09-20 N-(1-(4-amino-6,7-dialkoxy-2-quinazolinyl)-4-piperidyl)-oxazolidine-2,4-diones
JP58174020A JPS5978187A (ja) 1982-09-25 1983-09-20 新規ピペリジン誘導体
IL69777A IL69777A (en) 1982-09-25 1983-09-21 N-(1-(4-amino-6,7-dialkoxy-2-quinazolinyl)-4-piperidyl)-oxozolidine-2,4-diones,their preparation and pharmaceutical compositions containing them
CS836919A CS235342B2 (en) 1982-09-25 1983-09-22 Method of piperidine derivatives production
GR72505A GR78973B (forum.php) 1982-09-25 1983-09-22
AU19396/83A AU561118B2 (en) 1982-09-25 1983-09-23 Quinazolinyl-piperidyl-oxazolidine diones
HU833307A HU191637B (en) 1982-09-25 1983-09-23 Process for producing piperidine derivatives
PL1983243878A PL139590B1 (en) 1982-09-25 1983-09-23 Process for preparing novel derivatives of piperidine
CA000437468A CA1215981A (en) 1982-09-25 1983-09-23 Piperidine derivatives, the preparation and use thereof
NO833423A NO833423L (no) 1982-09-25 1983-09-23 Fremgangsmaate for fremstilling av piperidinderivater for anvendelse ved hjerte/kretsloepforstyrrelser.
DD83255091A DD212517A5 (de) 1982-09-25 1983-09-23 Verfahren zur herstellung von neuen piperidinderivaten
DK436583A DK436583A (da) 1982-09-25 1983-09-23 Fremgangsmaade til fremstilling af piperidinderivater
ES525876A ES8501762A1 (es) 1982-09-25 1983-09-23 Procedimiento para preparar nuevos derivados de piperidina
NZ205716A NZ205716A (en) 1982-09-25 1983-09-23 Piperidine derivatives and pharmaceutical compositions
YU01921/83A YU192183A (forum.php) 1982-09-25 1983-09-23
PT77380A PT77380B (de) 1982-09-25 1983-09-23 Piperidinderivate ihre herstellung und verwendung
ZA837081A ZA837081B (en) 1982-09-25 1983-09-23 Piperidine derivatives,processes for their preparation and pharmaceutical compositions containing them
KR1019830004475A KR840006222A (ko) 1982-09-25 1983-09-24 피페리딘 유도체의 제조방법
ES534351A ES8504182A1 (es) 1982-09-25 1984-07-16 Procedimiento para preparar nuevos derivados de piperidina
ES534349A ES8504180A1 (es) 1982-09-25 1984-07-16 Procedimiento para preparar nuevos derivados de piperidina
ES534350A ES534350A0 (es) 1982-09-25 1984-07-16 Procedimiento para preparar nuevos derivados de piperidina

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19823235565 DE3235565A1 (de) 1982-09-25 1982-09-25 Piperidinderivate, ihre herstellung und verwendung

Publications (1)

Publication Number Publication Date
DE3235565A1 true DE3235565A1 (de) 1984-03-29

Family

ID=6174159

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19823235565 Withdrawn DE3235565A1 (de) 1982-09-25 1982-09-25 Piperidinderivate, ihre herstellung und verwendung

Country Status (23)

Country Link
US (1) US4539323A (forum.php)
EP (1) EP0104445A3 (forum.php)
JP (1) JPS5978187A (forum.php)
KR (1) KR840006222A (forum.php)
AU (1) AU561118B2 (forum.php)
CA (1) CA1215981A (forum.php)
CS (1) CS235342B2 (forum.php)
DD (1) DD212517A5 (forum.php)
DE (1) DE3235565A1 (forum.php)
DK (1) DK436583A (forum.php)
ES (4) ES8501762A1 (forum.php)
FI (1) FI833292A7 (forum.php)
GR (1) GR78973B (forum.php)
HU (1) HU191637B (forum.php)
IL (1) IL69777A (forum.php)
NO (1) NO833423L (forum.php)
NZ (1) NZ205716A (forum.php)
PH (1) PH20015A (forum.php)
PL (1) PL139590B1 (forum.php)
PT (1) PT77380B (forum.php)
SU (1) SU1187720A3 (forum.php)
YU (1) YU192183A (forum.php)
ZA (1) ZA837081B (forum.php)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4601897A (en) * 1985-11-06 1986-07-22 Pfizer Inc. Prazosin-pirbuterol combination for bronchodilation
JPS62212385A (ja) * 1986-03-13 1987-09-18 Kotobuki Seiyaku Kk キナゾリン誘導体並びに血圧降下剤及びその製法
EP1317258B1 (en) * 2000-06-28 2009-02-11 Merck & Co., Inc. Use of allopurinol for the treatment of hypertension
ATE397669T1 (de) 2002-07-01 2008-06-15 Tibotec Pharm Ltd Mit phänotypischer medikamentenresistenz korrelierte mutationsprofile in hiv-1-reverse- transkriptase
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0009465A1 (de) * 1978-09-20 1980-04-02 Ciba-Geigy Ag N-(1-(4-Amino-2-chinazolinyl)-3- oder -4-piperidyl-lactame, Verfahren zu ihrer Herstellung, sowie pharmazeutische Präparate enthaltend diese Verbindungen
US4309541A (en) * 1978-09-20 1982-01-05 Ciba-Geigy Corporation Piperidinyl-lactams
FR2483920A1 (fr) * 1980-06-09 1981-12-11 Synthelabo Nouveaux derives de quinazoline, leur procede de preparation et leur application en therapeutique

Also Published As

Publication number Publication date
ES534351A0 (es) 1985-04-01
PT77380B (de) 1986-03-20
US4539323A (en) 1985-09-03
ES534349A0 (es) 1985-04-01
HU191637B (en) 1987-03-30
PL243878A1 (en) 1985-01-02
AU1939683A (en) 1984-03-29
CS235342B2 (en) 1985-05-15
IL69777A (en) 1986-09-30
KR840006222A (ko) 1984-11-22
ES8504181A1 (es) 1985-04-01
ES534350A0 (es) 1985-04-01
FI833292A0 (fi) 1983-09-15
YU192183A (forum.php) 1986-12-31
PT77380A (de) 1983-10-01
DD212517A5 (de) 1984-08-15
FI833292L (fi) 1984-03-26
DK436583D0 (da) 1983-09-23
ES8504180A1 (es) 1985-04-01
ZA837081B (en) 1985-05-29
PL139590B1 (en) 1987-02-28
EP0104445A2 (de) 1984-04-04
JPS5978187A (ja) 1984-05-04
CA1215981A (en) 1986-12-30
ES8504182A1 (es) 1985-04-01
EP0104445A3 (de) 1985-07-10
PH20015A (en) 1986-08-28
ES525876A0 (es) 1984-12-01
NO833423L (no) 1984-03-26
NZ205716A (en) 1985-08-30
SU1187720A3 (ru) 1985-10-23
AU561118B2 (en) 1987-04-30
GR78973B (forum.php) 1984-10-02
ES8501762A1 (es) 1984-12-01
DK436583A (da) 1984-03-26
FI833292A7 (fi) 1984-03-26

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Legal Events

Date Code Title Description
8139 Disposal/non-payment of the annual fee