DD159074A5 - Verfahren zur herstellung von dioxidverbindungen - Google Patents

Verfahren zur herstellung von dioxidverbindungen Download PDF

Info

Publication number
DD159074A5
DD159074A5 DD81230153A DD23015381A DD159074A5 DD 159074 A5 DD159074 A5 DD 159074A5 DD 81230153 A DD81230153 A DD 81230153A DD 23015381 A DD23015381 A DD 23015381A DD 159074 A5 DD159074 A5 DD 159074A5
Authority
DD
German Democratic Republic
Prior art keywords
group
formula
compounds
acid
salt
Prior art date
Application number
DD81230153A
Other languages
German (de)
English (en)
Inventor
Peter Schneider
Riccardo Scartazzini
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DD159074A5 publication Critical patent/DD159074A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
DD81230153A 1980-05-22 1981-05-21 Verfahren zur herstellung von dioxidverbindungen DD159074A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH401780 1980-05-22

Publications (1)

Publication Number Publication Date
DD159074A5 true DD159074A5 (de) 1983-02-16

Family

ID=4268255

Family Applications (1)

Application Number Title Priority Date Filing Date
DD81230153A DD159074A5 (de) 1980-05-22 1981-05-21 Verfahren zur herstellung von dioxidverbindungen

Country Status (13)

Country Link
EP (1) EP0041047A3 (instruction)
JP (1) JPS5718685A (instruction)
KR (1) KR830006304A (instruction)
AU (1) AU7091181A (instruction)
DD (1) DD159074A5 (instruction)
DK (1) DK224281A (instruction)
FI (1) FI811532L (instruction)
GB (1) GB2076812A (instruction)
GR (1) GR75639B (instruction)
IL (1) IL62912A0 (instruction)
NO (1) NO811740L (instruction)
PT (1) PT73067B (instruction)
ZA (1) ZA8103408D (instruction)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
GR77151B (instruction) * 1982-01-11 1984-09-07 Prizer
US4503040A (en) * 1984-02-27 1985-03-05 Pfizer Inc. 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors
DE3586021D1 (de) * 1984-07-30 1992-06-17 Merck & Co Inc Penicillin-derivate als entzuendungshemmende und degenerierungskaempfende arzneimittel.
US4591459A (en) * 1984-12-03 1986-05-27 Pfizer Inc. Intermediates for 6-(aminoacyloxymethyl) penicillanic acid 1,1-dioxides
GB2206579B (en) * 1987-07-10 1991-05-29 Erba Farmitalia 6a and 6b-(substituted methyl)-penicillanic acid derivatives
WO1999033838A1 (en) 1997-12-29 1999-07-08 Research Corporation Technologies, Inc. 2-β-SUBSTITUTED-6-ALKYLIDENE PENICILLANIC ACID DERIVATIVES AS β-LACTAMASE INHIBITORS
AU2624600A (en) * 1999-01-26 2000-08-07 American Cyanamid Company 3,6-disubstituted penam sulfone derivatives as antibacterials
US6395726B1 (en) 1999-01-26 2002-05-28 American Cyanamid Company 3,6-disubstituted penam sulfone derivatives
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
ES2272795T3 (es) 2001-07-24 2007-05-01 Southern Methodist University Foundation For Research 7-alquildieno-3-sustituidos-3-cefem-4-carboxilatos como inhibidores de beta-lactamasa.
JP2005525399A (ja) 2002-04-04 2005-08-25 アラムクス エルエルシー セリンおよびメタロ−β−ラクタマーゼの阻害剤
PA8579701A1 (es) * 2002-08-23 2005-05-24 Pfizer Prod Inc Profarmaco inhibidor de beta-lactamasa
WO2004108733A1 (en) * 2003-06-05 2004-12-16 Pfizer Products Inc. Beta-lactamase inhibitor prodrug

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1102308A (en) * 1975-09-26 1981-06-02 John C. Sheehan Carbon and oxygen analogs of cephalosporins
US4207323A (en) * 1975-11-21 1980-06-10 Merck & Co., Inc. 6-Substituted methyl penicillins, derivatives and analogues thereof
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

Also Published As

Publication number Publication date
FI811532A7 (fi) 1981-11-23
EP0041047A2 (de) 1981-12-02
DK224281A (da) 1981-11-23
PT73067B (en) 1983-02-08
JPS5718685A (en) 1982-01-30
PT73067A (en) 1981-06-01
GB2076812A (en) 1981-12-09
AU7091181A (en) 1981-11-26
IL62912A0 (en) 1981-07-31
FI811532L (fi) 1981-11-23
KR830006304A (ko) 1983-09-20
EP0041047A3 (de) 1982-04-07
ZA8103408D (en) 1982-06-30
GR75639B (instruction) 1984-03-02
NO811740L (no) 1981-11-23

Similar Documents

Publication Publication Date Title
DE3005164A1 (de) Antibiotisch wirksame beta -lactamverbindungen, verfahren zu deren herstellung und sie enthaltendes arzneimittel
DD159074A5 (de) Verfahren zur herstellung von dioxidverbindungen
DD201906A5 (de) Verfahren zur herstellung von 7 beta-aminothiadiazolylacetylamino-3 ammoniomethyl-3-cephem-4-carbonsaeureverbindungen
EP0009008A2 (de) Cephalosporinderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
DD215551A5 (de) Verfahren zur herstellung von 6-hydroxyniederalkyl-penem-verbindungen
DD152788A5 (de) Verfahren zur herstellung von polyazathiaverbindungen
EP0246187A2 (de) 2-Pyridyl-penem-Verbindungen
DE69625910T2 (de) Penamsulfone als beta-laktamase inhibitoren
DE2153554A1 (de) Thiaheterocyclische Verbindungen
DD211562A5 (de) Verfahren zur herstellung von 2-heterocyclylniederalkyl-2-penem-verbindungen
EP0022245A2 (de) Amino-thiadiazolyl-Verbindungen, Verfahren zu ihrer Herstellung, sie enthaltende pharmazeutische Präparate; Ausgangsverbindungen und Verfahren zu ihrer Herstellung
EP0199675A1 (de) Heterocyclyl-penem-Verbindungen
CH620444A5 (en) Process for the preparation of bicyclic unsaturated thiaaza compounds
DE4037841A1 (de) Neue 3-substituierte cephalosporine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DE2448582A1 (de) Verfahren zur herstellung von cephalosporinen
DE3431980A1 (de) Aminomethyl-verbindungen
EP0015240A1 (de) Azacyclyl (thio) ureidoacetyl-Verbindungen und Verfahren zu ihrer Herstellung
DE2736071C2 (de) α-Methoxy-cephalosporinderivate, Verfahren zu ihrer Herstellung sowie diese als Wirkstoffe enthaltende pharmazeutische Zubereitungen
DD204256A5 (de) Verfahren zur herstellung von aminooxazolylverbindungen
EP0201459A1 (de) Acylaminomethylpenemverbindungen, ihre Herstellung und sie enthaltende pharmazeutische Präparate
EP0112283A1 (de) Heterocyclylthioverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verwendung von letzteren
EP0037797A2 (de) Cephalosporinverbindungen, Verfahren zu ihrer Herstellung, sie enthaltende pharmazeutische Zusammensetzungen und ihre Verwendung
DE3518848A1 (de) Aminoaethylthioverbindungen
DE3326194A1 (de) Aminoimidazolyl-verbindungen, verfahren zu ihrer herstellung, pharmazeutische praeparate, welche diese vrbindungen enthalten, und verwendung von letzteren
EP0031794A2 (de) Cephalosporinderivative, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Zusammensetzungen