CY1120700T1 - Ενωσεις τριαμινοπυριμιδινης χρησιμες για προληψη ή αγωγη ελονοσιας - Google Patents

Ενωσεις τριαμινοπυριμιδινης χρησιμες για προληψη ή αγωγη ελονοσιας

Info

Publication number
CY1120700T1
CY1120700T1 CY181100997T CY181100997T CY1120700T1 CY 1120700 T1 CY1120700 T1 CY 1120700T1 CY 181100997 T CY181100997 T CY 181100997T CY 181100997 T CY181100997 T CY 181100997T CY 1120700 T1 CY1120700 T1 CY 1120700T1
Authority
CY
Cyprus
Prior art keywords
prevention
treatment
maternity
compounds used
triaminopyrimidine
Prior art date
Application number
CY181100997T
Other languages
Greek (el)
English (en)
Inventor
Peer Mohamed Shahul Hameed
Vikas Patil
Kannan Murugan
Bellale Eknath Vithalrao
Anandkumar Raichurkar
Sudhir Landge
Jayashree Puttur
Choudhury Nilanjana Roy
Gajanan Shanbhag
Krishna Koushik
Pravin Iyer
Sambandamurthy Vasan Kirthika
Suresh Solapure
Shridhar Narayanan
Original Assignee
Medicines For Malaria Venture Mmv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medicines For Malaria Venture Mmv filed Critical Medicines For Malaria Venture Mmv
Publication of CY1120700T1 publication Critical patent/CY1120700T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CY181100997T 2014-04-28 2018-09-27 Ενωσεις τριαμινοπυριμιδινης χρησιμες για προληψη ή αγωγη ελονοσιας CY1120700T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN2142CH2014 2014-04-28
PCT/EP2015/056496 WO2015165660A1 (en) 2014-04-28 2015-03-26 Triaminopyrimidine compounds useful for preventing or treating malaria

Publications (1)

Publication Number Publication Date
CY1120700T1 true CY1120700T1 (el) 2019-12-11

Family

ID=52779638

Family Applications (1)

Application Number Title Priority Date Filing Date
CY181100997T CY1120700T1 (el) 2014-04-28 2018-09-27 Ενωσεις τριαμινοπυριμιδινης χρησιμες για προληψη ή αγωγη ελονοσιας

Country Status (22)

Country Link
US (1) US9957253B2 (https=)
EP (1) EP3137455B1 (https=)
JP (1) JP6529983B2 (https=)
CN (1) CN106255685B (https=)
AP (1) AP2016009570A0 (https=)
BR (1) BR112016024467B1 (https=)
CA (1) CA2946654C (https=)
CY (1) CY1120700T1 (https=)
DK (1) DK3137455T3 (https=)
ES (1) ES2696350T3 (https=)
HR (1) HRP20181816T1 (https=)
HU (1) HUE042043T2 (https=)
LT (1) LT3137455T (https=)
MX (1) MX374458B (https=)
MY (1) MY178971A (https=)
PH (1) PH12016502322B1 (https=)
PL (1) PL3137455T3 (https=)
PT (1) PT3137455T (https=)
RS (1) RS58124B1 (https=)
SI (1) SI3137455T1 (https=)
SM (1) SMT201800588T1 (https=)
WO (1) WO2015165660A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105699584B (zh) * 2016-02-03 2018-02-09 昆药集团股份有限公司 一种蒿甲醚相关物质的检测方法
WO2018079629A1 (ja) 2016-10-26 2018-05-03 カルナバイオサイエンス株式会社 抗マラリア活性を有する新規ピリミジン誘導体
CN106727584A (zh) * 2017-02-08 2017-05-31 于贵庆 一种治疗骨病的药物组合物
JP2020532513A (ja) * 2017-09-05 2020-11-12 カディラ ヘルスケア リミティド トリアミノピリミジン化合物およびその中間体の調製方法
CN117327007B (zh) * 2023-09-26 2024-09-13 上海陶术生物科技有限公司 一种vt107的制备方法
WO2025115034A1 (en) * 2023-11-30 2025-06-05 Zydus Lifesciences Limited A process for the preparation of a triaminopyrimidine compound and novel intermediates thereof
EP4574143A1 (en) 2023-12-21 2025-06-25 Universität Regensburg Inhibitors of plasmodia remodeling enzymes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003286711A1 (en) * 2002-10-25 2004-05-13 Vertex Pharmaceuticals Incorporated Indazolinone compositions useful as kinase inhibitors
RU2405778C2 (ru) * 2004-09-30 2010-12-10 Тиботек Фармасьютикалз Лтд. 5-гетероциклилпиримидины, ингибирующие вич
WO2014058685A1 (en) * 2012-10-08 2014-04-17 Merck Sharp & Dohme Corp. Inhibitors of irak4 activity

Also Published As

Publication number Publication date
AP2016009570A0 (en) 2016-11-30
CA2946654A1 (en) 2015-11-05
MY178971A (en) 2020-10-26
CN106255685B (zh) 2019-08-20
EP3137455A1 (en) 2017-03-08
CN106255685A (zh) 2016-12-21
US20170050951A1 (en) 2017-02-23
RS58124B1 (sr) 2019-02-28
MX374458B (es) 2025-03-06
JP2017514804A (ja) 2017-06-08
PH12016502322B1 (en) 2022-03-23
PL3137455T3 (pl) 2019-01-31
MX2016014166A (es) 2017-02-14
PH12016502322A1 (en) 2017-01-30
BR112016024467B1 (pt) 2022-11-29
LT3137455T (lt) 2018-10-25
CA2946654C (en) 2022-08-23
EP3137455B1 (en) 2018-08-15
BR112016024467A2 (pt) 2017-08-15
WO2015165660A1 (en) 2015-11-05
HK1231478A1 (en) 2017-12-22
SI3137455T1 (sl) 2019-01-31
US9957253B2 (en) 2018-05-01
HRP20181816T1 (hr) 2018-12-28
PT3137455T (pt) 2018-11-21
DK3137455T3 (en) 2018-12-10
SMT201800588T1 (it) 2019-01-11
JP6529983B2 (ja) 2019-06-12
ES2696350T3 (es) 2019-01-15
HUE042043T2 (hu) 2019-06-28

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