CY1112478T1 - Ενωσεις κιναζολινονης ως αντικαρκινικοι παραγοντες - Google Patents

Ενωσεις κιναζολινονης ως αντικαρκινικοι παραγοντες

Info

Publication number
CY1112478T1
CY1112478T1 CY20121100255T CY121100255T CY1112478T1 CY 1112478 T1 CY1112478 T1 CY 1112478T1 CY 20121100255 T CY20121100255 T CY 20121100255T CY 121100255 T CY121100255 T CY 121100255T CY 1112478 T1 CY1112478 T1 CY 1112478T1
Authority
CY
Cyprus
Prior art keywords
compounds
kinazolinone
cancer factors
quinazolinone compounds
alone
Prior art date
Application number
CY20121100255T
Other languages
Greek (el)
English (en)
Inventor
Weibo Wang
Liana M Lagniton
Ryan N Constantine
Manoj C Desai
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CY1112478T1 publication Critical patent/CY1112478T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CY20121100255T 2003-11-25 2012-03-12 Ενωσεις κιναζολινονης ως αντικαρκινικοι παραγοντες CY1112478T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US52505903P 2003-11-25 2003-11-25
EP04812051A EP1689724B1 (en) 2003-11-25 2004-11-24 Quinazolinone compounds as anticancer agents

Publications (1)

Publication Number Publication Date
CY1112478T1 true CY1112478T1 (el) 2015-12-09

Family

ID=34632957

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121100255T CY1112478T1 (el) 2003-11-25 2012-03-12 Ενωσεις κιναζολινονης ως αντικαρκινικοι παραγοντες

Country Status (17)

Country Link
US (2) US7939539B2 (enExample)
EP (1) EP1689724B1 (enExample)
JP (2) JP4778439B2 (enExample)
KR (1) KR20060127413A (enExample)
CN (1) CN1886384A (enExample)
AT (1) ATE538103T1 (enExample)
AU (1) AU2004293464A1 (enExample)
CA (1) CA2546932A1 (enExample)
CY (1) CY1112478T1 (enExample)
DK (1) DK1689724T3 (enExample)
ES (1) ES2376552T3 (enExample)
IL (1) IL175714A0 (enExample)
PL (1) PL1689724T3 (enExample)
PT (1) PT1689724E (enExample)
SG (1) SG148202A1 (enExample)
SI (1) SI1689724T1 (enExample)
WO (1) WO2005051922A1 (enExample)

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Also Published As

Publication number Publication date
SI1689724T1 (sl) 2012-04-30
EP1689724B1 (en) 2011-12-21
KR20060127413A (ko) 2006-12-12
WO2005051922A1 (en) 2005-06-09
US20050209254A1 (en) 2005-09-22
IL175714A0 (en) 2006-09-05
EP1689724A1 (en) 2006-08-16
US20110190293A1 (en) 2011-08-04
ATE538103T1 (de) 2012-01-15
JP2011084570A (ja) 2011-04-28
US7939539B2 (en) 2011-05-10
PT1689724E (pt) 2012-02-06
AU2004293464A1 (en) 2005-06-09
ES2376552T3 (es) 2012-03-14
SG148202A1 (en) 2008-12-31
PL1689724T3 (pl) 2012-05-31
DK1689724T3 (da) 2012-02-27
CA2546932A1 (en) 2005-06-09
JP2007512368A (ja) 2007-05-17
CN1886384A (zh) 2006-12-27
JP4778439B2 (ja) 2011-09-21

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