CY1105796T1 - Θepαπεια οξεωσης της μεγαλης κοιλιας των μηρυκαστικων με αναστολεις αλφα-αμυλασης - Google Patents

Θepαπεια οξεωσης της μεγαλης κοιλιας των μηρυκαστικων με αναστολεις αλφα-αμυλασης

Info

Publication number
CY1105796T1
CY1105796T1 CY20061101681T CY061101681T CY1105796T1 CY 1105796 T1 CY1105796 T1 CY 1105796T1 CY 20061101681 T CY20061101681 T CY 20061101681T CY 061101681 T CY061101681 T CY 061101681T CY 1105796 T1 CY1105796 T1 CY 1105796T1
Authority
CY
Cyprus
Prior art keywords
ruminant
amylase
bacterial
glucosidase
acidosis
Prior art date
Application number
CY20061101681T
Other languages
English (en)
Inventor
Bernard Joseph Banks
Mark Andrew Haxell
Graham Lunn
Michael Stephen Pacey
Lee Richard Roberts
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0012760A external-priority patent/GB0012760D0/en
Priority claimed from GB0012793A external-priority patent/GB0012793D0/en
Priority claimed from GB0017495A external-priority patent/GB0017495D0/en
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of CY1105796T1 publication Critical patent/CY1105796T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/702Oligosaccharides, i.e. having three to five saccharide radicals attached to each other by glycosidic linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K10/00Animal feeding-stuffs
    • A23K10/10Animal feeding-stuffs obtained by microbiological or biochemical processes
    • A23K10/12Animal feeding-stuffs obtained by microbiological or biochemical processes by fermentation of natural products, e.g. of vegetable material, animal waste material or biomass
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/163Sugars; Polysaccharides
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K50/00Feeding-stuffs specially adapted for particular animals
    • A23K50/10Feeding-stuffs specially adapted for particular animals for ruminants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7016Disaccharides, e.g. lactose, lactulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Polymers & Plastics (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Animal Husbandry (AREA)
  • Food Science & Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biotechnology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Sustainable Development (AREA)
  • Biomedical Technology (AREA)
  • Microbiology (AREA)
  • Physiology (AREA)
  • Birds (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Fodder In General (AREA)
  • Saccharide Compounds (AREA)
  • Feed For Specific Animals (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Η εφεύρεση που περιγράφεται εδώ αφορά: τη χρήση ενός αποτελεσματικού αναστολέα μιας βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης στη βιομηχανική κατασκευή μιας σύνθεσης για τη θεραπεία οξέωσης, μέθοδο θεραπείας οξέωσης της μεγάλης κοιλίας των μηρυκαστικών, που περιλαμβάνει χορήγηση αποτελεσματικής ποσότητας ενός αποτελεσματικού αναστολέα μιας βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης σε ένα μηρυκαστικό, συνταγοποίηση κατάλληλη για τη θεραπεία οξέωσης σε ένα ζώο, που περιλαμβάνει αποτελεσματικό αναστολέα μιας βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης σε ανάμιξη με ένα κατάλληλο έκδοχο, διαλύτη ή φορέα, που επιλέγεται σε σχέση με τον επιδιωκόμενο τρόπο χορήγησης και την πρότυπη φαρμακευτική/κτηνιατρική/αγροκτήματος πρακτική, μεθόδους λεπτομερούς εξέτασης χρήσιμες στην πιστοποίηση ενός κατάλληλου αναστολέα μιας βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης για τη θεραπεία οξέωσης σε ένα μηρυκαστικό, μέθοδο για βελτίωση της ποιότητας γάλακτος ή/και της ποσότητας μηρυκαστικού, που περιλαμβάνει θεραπεία ενός μηρυκαστικού με μια αποτελεσματική ποσότητα ενός αναστολέα βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης, μια ένωση του τύπου I:ή κτηνιατρικώς αποδεκτό άλας, διαλύτωμα (συμπεριλαμβανομένου υδρίτη) ή προφαρμάκου αυτής και μεθόδους για να κατασκευάζεται ένας αποτελεσματικός αναστολέας μιας βακτηριακής α-αμυλάσης ή/και α-γλυκοσιδάσης χρήσιμος για τη θεραπεία οξέωσης σε ένα μηρυκαστικό.
CY20061101681T 2000-05-24 2006-11-17 Θepαπεια οξεωσης της μεγαλης κοιλιας των μηρυκαστικων με αναστολεις αλφα-αμυλασης CY1105796T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0012760A GB0012760D0 (en) 2000-05-24 2000-05-24 Treatment
GB0012793A GB0012793D0 (en) 2000-05-24 2000-05-24 Treatment
GB0017495A GB0017495D0 (en) 2000-07-17 2000-07-17 Treatment

Publications (1)

Publication Number Publication Date
CY1105796T1 true CY1105796T1 (el) 2011-02-02

Family

ID=27255738

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20061101681T CY1105796T1 (el) 2000-05-24 2006-11-17 Θepαπεια οξεωσης της μεγαλης κοιλιας των μηρυκαστικων με αναστολεις αλφα-αμυλασης

Country Status (17)

Country Link
US (1) US20050233983A1 (el)
EP (2) EP1157696B1 (el)
JP (2) JP3798261B2 (el)
KR (1) KR100643946B1 (el)
AT (1) ATE343391T1 (el)
AU (1) AU785303B2 (el)
CA (1) CA2348245C (el)
CY (1) CY1105796T1 (el)
DE (1) DE60124030T2 (el)
DK (1) DK1157696T3 (el)
ES (1) ES2272418T3 (el)
HU (1) HUP0102159A3 (el)
IL (2) IL186223A0 (el)
MY (1) MY136145A (el)
NZ (1) NZ511877A (el)
PT (1) PT1157696E (el)
TW (1) TWI298021B (el)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60124030T2 (de) * 2000-05-24 2007-04-12 Pfizer Inc. Behandlung von Pansenacidose mit Amylasehemmern
US7906128B2 (en) * 2002-10-21 2011-03-15 Wyeth Llc Use of neuronal sodium channel antagonists for the control of ectoparasites in homeothermic animals
US7108869B2 (en) * 2002-11-07 2006-09-19 Access Business Group International Llc Nutritional supplement containing alpha-glucosidase and alpha-amylase inhibitors
CN1296050C (zh) * 2003-12-10 2007-01-24 浙江海正药业股份有限公司 阿卡波糖肠溶片及制备方法
CN101235061B (zh) * 2007-09-11 2011-03-30 南开大学 一类新的α-淀粉酶抑制剂阿卡他定系列化合物及其应用
US8791245B2 (en) * 2008-10-03 2014-07-29 Glycan Bioscience LLC Anionic conjugates of glycosylated bacterial metabolite
DE102009015558B4 (de) * 2009-03-30 2017-04-27 Ulf-Michael Stumpe Bollus zum Eingeben in die Vormägen von Wiederkäuern zur Verbesserung der Vormagenaktivität und Vormagengesundheit
US20130164275A1 (en) * 2009-10-26 2013-06-27 Pharmachem Laboratories, Inc. Method for treating acidosis in ruminants
CN102212089A (zh) * 2011-04-12 2011-10-12 天津医科大学 一类新的α-淀粉酶抑制剂阿卡他定家族新化合物及其应用
EP3375453A1 (de) * 2017-03-13 2018-09-19 Basf Se Verwendung einer pansengeschützen alpha-amylase
WO2020118345A1 (en) * 2018-12-14 2020-06-18 ProAgni Pty Ltd Animal feed composition
CN110899293A (zh) * 2019-10-15 2020-03-24 上海交通大学 一种对阿卡波糖废渣减量化处理的方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4062950A (en) * 1973-09-22 1977-12-13 Bayer Aktiengesellschaft Amino sugar derivatives
DE2658562A1 (de) * 1976-12-23 1978-10-12 Bayer Ag Aminozuckerderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
US4175123A (en) * 1976-12-23 1979-11-20 Bayer Aktiengesellschaft Amino-sugar derivatives, process for their preparation and pharmaceutical composition thereof
CA1121290A (en) * 1978-02-14 1982-04-06 Yasuji Suhara Amino sugar derivatives
EP0173950A3 (de) * 1984-09-04 1987-10-28 Hoechst Aktiengesellschaft Neuer alpha-Glukosidase Inhibitor, Verfahren zur seiner Herstellung, seine Verwendung und pharmazeutische Präparate
DE3543999A1 (de) * 1985-12-13 1987-06-19 Bayer Ag Hochreine acarbose
US4885361A (en) * 1987-07-31 1989-12-05 Hoffmann-La Roche Inc. Sulfated oligosaccharides
US5021427A (en) * 1988-12-23 1991-06-04 The Board Of Regents, The University Of Texas System Novel pyrrolizidine alkaloid
WO1999026606A2 (en) * 1997-11-25 1999-06-03 Bayer Aktiengesellschaft SUSTAINED RELEASE FORMULATIONS COMPRISING α-GLUCOSIDASE-INHIBITORS
US7022684B2 (en) * 2000-05-24 2006-04-04 Pfizer Inc. Treatment of rumen acidosis with α-amylase inhibitors
DE60124030T2 (de) * 2000-05-24 2007-04-12 Pfizer Inc. Behandlung von Pansenacidose mit Amylasehemmern

Also Published As

Publication number Publication date
DK1157696T3 (da) 2007-02-12
EP1745790A3 (en) 2007-03-21
KR100643946B1 (ko) 2006-11-10
CA2348245C (en) 2007-12-11
IL143225A0 (en) 2002-04-21
KR20010107661A (ko) 2001-12-07
PT1157696E (pt) 2007-01-31
MY136145A (en) 2008-08-29
HUP0102159A2 (hu) 2002-01-28
EP1745790A2 (en) 2007-01-24
ATE343391T1 (de) 2006-11-15
JP2005336192A (ja) 2005-12-08
IL186223A0 (en) 2008-01-20
DE60124030T2 (de) 2007-04-12
IL143225A (en) 2008-03-20
EP1157696A2 (en) 2001-11-28
AU4619201A (en) 2001-11-29
AU785303B2 (en) 2007-01-04
HU0102159D0 (en) 2001-08-28
US20050233983A1 (en) 2005-10-20
DE60124030D1 (de) 2006-12-07
EP1157696B1 (en) 2006-10-25
CA2348245A1 (en) 2001-11-24
EP1157696A3 (en) 2002-02-13
ES2272418T3 (es) 2007-05-01
TWI298021B (en) 2008-06-21
NZ511877A (en) 2002-11-26
JP2002047209A (ja) 2002-02-12
JP3798261B2 (ja) 2006-07-19
HUP0102159A3 (en) 2004-01-28

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