CS299191A3 - 4- or 5-substituted pyridine-2-carboxylic acids, process of their preparation as well as their application as medicaments - Google Patents
4- or 5-substituted pyridine-2-carboxylic acids, process of their preparation as well as their application as medicamentsInfo
- Publication number
- CS299191A3 CS299191A3 CS912991A CS299191A CS299191A3 CS 299191 A3 CS299191 A3 CS 299191A3 CS 912991 A CS912991 A CS 912991A CS 299191 A CS299191 A CS 299191A CS 299191 A3 CS299191 A3 CS 299191A3
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- medicaments
- preparation
- well
- application
- carboxylic acids
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Immunology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Transplantation (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4031000A DE4031000A1 (de) | 1990-10-01 | 1990-10-01 | 4- oder 5-substituierte pyridin-2-carbonsaeuren, verfahren zu deren herstellung sowie deren verwendung als arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS299191A3 true CS299191A3 (en) | 1992-06-17 |
Family
ID=6415345
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS912991A CS299191A3 (en) | 1990-10-01 | 1991-09-30 | 4- or 5-substituted pyridine-2-carboxylic acids, process of their preparation as well as their application as medicaments |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP0479177A3 (zh) |
| JP (1) | JPH04247070A (zh) |
| KR (1) | KR920007999A (zh) |
| CN (1) | CN1060655A (zh) |
| AU (1) | AU8485291A (zh) |
| BG (1) | BG95162A (zh) |
| BR (1) | BR9104205A (zh) |
| CA (1) | CA2052510A1 (zh) |
| CS (1) | CS299191A3 (zh) |
| DE (1) | DE4031000A1 (zh) |
| FI (1) | FI914556A (zh) |
| HU (1) | HUT59103A (zh) |
| IE (1) | IE913435A1 (zh) |
| IL (1) | IL99605A0 (zh) |
| MA (1) | MA22313A1 (zh) |
| MX (1) | MX9101347A (zh) |
| NO (1) | NO913834L (zh) |
| PL (1) | PL291881A1 (zh) |
| PT (1) | PT99132A (zh) |
| ZA (1) | ZA917805B (zh) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0617020A1 (en) * | 1992-04-02 | 1994-09-28 | Shudo, Koichi, Prof. Dr. | Carboxylic acid derivatives having retinoic acid-like activity |
| DE4233124A1 (de) * | 1992-10-02 | 1994-04-07 | Hoechst Ag | Acylsulfonamido- und Sulfonamidopyridin-2-carbonsäureester sowie ihre Pyridin-N-oxide, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| WO2006034341A2 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase |
| CA2580857A1 (en) | 2004-09-20 | 2006-09-28 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| JP5094398B2 (ja) | 2004-09-20 | 2012-12-12 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | 複素環式誘導体およびステアロイル−ＣｏＡデサチュラーゼのメディエータとしてのそれらの使用 |
| MX2007003318A (es) | 2004-09-20 | 2007-05-18 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como agentes terapeuticos. |
| TW200626138A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
| WO2006034441A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| WO2006034440A2 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| AU2006343359A1 (en) | 2005-06-03 | 2007-11-15 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3703959A1 (de) * | 1987-02-10 | 1988-08-18 | Hoechst Ag | Pyridin-2,4- und 2,5-dicarbonsaeureamide, verfahren zu ihrer herstellung, verwendung derselben sowie arzneimittel auf basis dieser verbindungen |
| DE3703962A1 (de) * | 1987-02-10 | 1988-08-18 | Hoechst Ag | Pyridin-2,4- und 2,5-dicarbonsaeure-derivate, verfahren zu ihrer herstellung, verwendung derselben sowie arzneimittel auf basis dieser verbindungen |
| DE58908519D1 (de) * | 1988-08-04 | 1994-11-24 | Hoechst Ag | Verbessertes Verfahren zur Herstellung von N,N-Bis(alkoxyalkyl)-pyridin -2,4-dicarbonsäurediamiden. |
-
1990
- 1990-10-01 DE DE4031000A patent/DE4031000A1/de not_active Withdrawn
-
1991
- 1991-09-24 BG BG095162A patent/BG95162A/bg unknown
- 1991-09-27 FI FI914556A patent/FI914556A/fi unknown
- 1991-09-27 IL IL99605A patent/IL99605A0/xx unknown
- 1991-09-30 KR KR1019910017066A patent/KR920007999A/ko not_active Application Discontinuation
- 1991-09-30 CS CS912991A patent/CS299191A3/cs unknown
- 1991-09-30 PL PL29188191A patent/PL291881A1/xx unknown
- 1991-09-30 EP EP19910116632 patent/EP0479177A3/de not_active Withdrawn
- 1991-09-30 BR BR919104205A patent/BR9104205A/pt unknown
- 1991-09-30 JP JP3250719A patent/JPH04247070A/ja active Pending
- 1991-09-30 NO NO91913834A patent/NO913834L/no unknown
- 1991-09-30 HU HU913119A patent/HUT59103A/hu unknown
- 1991-09-30 ZA ZA917805A patent/ZA917805B/xx unknown
- 1991-09-30 IE IE343591A patent/IE913435A1/en not_active Application Discontinuation
- 1991-09-30 CA CA002052510A patent/CA2052510A1/en not_active Abandoned
- 1991-09-30 MX MX9101347A patent/MX9101347A/es unknown
- 1991-09-30 CN CN91109400A patent/CN1060655A/zh active Pending
- 1991-09-30 AU AU84852/91A patent/AU8485291A/en not_active Abandoned
- 1991-10-01 MA MA22593A patent/MA22313A1/fr unknown
- 1991-10-01 PT PT99132A patent/PT99132A/pt not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| HUT59103A (en) | 1992-04-28 |
| HU913119D0 (en) | 1992-01-28 |
| IE913435A1 (en) | 1992-04-08 |
| BG95162A (bg) | 1993-12-24 |
| EP0479177A2 (de) | 1992-04-08 |
| KR920007999A (ko) | 1992-05-27 |
| AU8485291A (en) | 1992-04-02 |
| FI914556A0 (fi) | 1991-09-27 |
| ZA917805B (en) | 1992-05-27 |
| MX9101347A (es) | 1992-06-05 |
| EP0479177A3 (en) | 1992-10-28 |
| PL291881A1 (en) | 1992-06-15 |
| JPH04247070A (ja) | 1992-09-03 |
| NO913834L (no) | 1992-04-02 |
| PT99132A (pt) | 1992-09-30 |
| CN1060655A (zh) | 1992-04-29 |
| DE4031000A1 (de) | 1992-04-09 |
| CA2052510A1 (en) | 1992-04-02 |
| FI914556A (fi) | 1992-04-02 |
| MA22313A1 (fr) | 1992-07-01 |
| IL99605A0 (en) | 1992-08-18 |
| NO913834D0 (no) | 1991-09-30 |
| BR9104205A (pt) | 1992-06-02 |
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