CS250680B2 - Method of 2-oxindole-1-carboxamides production - Google Patents

Method of 2-oxindole-1-carboxamides production Download PDF

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Publication number
CS250680B2
CS250680B2 CS851921A CS192185A CS250680B2 CS 250680 B2 CS250680 B2 CS 250680B2 CS 851921 A CS851921 A CS 851921A CS 192185 A CS192185 A CS 192185A CS 250680 B2 CS250680 B2 CS 250680B2
Authority
CS
Czechoslovakia
Prior art keywords
alkyl
group
carbon atoms
hydrogen
formula
Prior art date
Application number
CS851921A
Other languages
Czech (cs)
English (en)
Inventor
Thomas Ch Crawford
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS250680B2 publication Critical patent/CS250680B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/34—Oxygen atoms in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/38—Oxygen atoms in positions 2 and 3, e.g. isatin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CS851921A 1984-03-19 1985-03-19 Method of 2-oxindole-1-carboxamides production CS250680B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59066784A 1984-03-19 1984-03-19
US68488984A 1984-12-21 1984-12-21

Publications (1)

Publication Number Publication Date
CS250680B2 true CS250680B2 (en) 1987-05-14

Family

ID=27080914

Family Applications (1)

Application Number Title Priority Date Filing Date
CS851921A CS250680B2 (en) 1984-03-19 1985-03-19 Method of 2-oxindole-1-carboxamides production

Country Status (29)

Country Link
EP (1) EP0155828B1 (de)
JP (1) JPH03178963A (de)
KR (1) KR860001874B1 (de)
AR (1) AR247885A1 (de)
AU (1) AU552119B2 (de)
BG (1) BG44203A3 (de)
CA (1) CA1250832A (de)
CS (1) CS250680B2 (de)
CY (1) CY1667A (de)
DE (1) DE3579716D1 (de)
DK (2) DK163662C (de)
EG (1) EG17274A (de)
ES (1) ES541373A0 (de)
FI (1) FI85265C (de)
GR (1) GR850669B (de)
HK (1) HK75992A (de)
HU (1) HU194825B (de)
IE (1) IE57741B1 (de)
IL (1) IL74630A (de)
MA (1) MA20379A1 (de)
NO (1) NO168639C (de)
NZ (1) NZ211487A (de)
OA (1) OA07967A (de)
PH (1) PH20843A (de)
PL (1) PL145873B1 (de)
PT (1) PT80116B (de)
RO (1) RO90953B (de)
YU (1) YU43869B (de)
ZW (1) ZW4885A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE63543T1 (de) * 1984-02-07 1991-06-15 Pfizer 2-oxindolzwischenprodukte.
US4686224A (en) * 1984-10-31 1987-08-11 Pfizer Inc. Oxindole antiinflammatory agents
DE3621761A1 (de) * 1986-06-28 1988-01-07 Bayer Ag Indolylpropionsaeuren
RO105052B1 (en) * 1987-02-02 1994-12-01 Pfizer Producing process for the crystalline sodium salt, anhydre, of 5-chlorine-3-(2-tenoil)-2-oxindol-1-carboxamide
GB8720693D0 (en) * 1987-09-03 1987-10-07 Glaxo Group Ltd Chemical compounds
US4952703A (en) * 1989-05-25 1990-08-28 Pfizer Inc. Intermediates for making 2-oxindole-1-carboxamides
HUP9600855A3 (en) * 1996-04-03 1998-04-28 Egyt Gyogyszervegyeszeti Gyar Process for producing tenidap
US7186745B2 (en) 2001-03-06 2007-03-06 Astrazeneca Ab Indolone derivatives having vascular damaging activity

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3767653A (en) * 1971-06-28 1973-10-23 Squibb & Sons Inc Thiazines

Also Published As

Publication number Publication date
IL74630A (en) 1988-04-29
DE3579716D1 (de) 1990-10-25
HUT37397A (en) 1985-12-28
HK75992A (en) 1992-10-09
NO168639B (no) 1991-12-09
NO851059L (no) 1985-09-20
PH20843A (en) 1987-05-08
AU4005885A (en) 1985-09-26
PT80116B (pt) 1987-10-20
RO90953B (ro) 1987-02-28
GR850669B (de) 1985-07-25
JPH0525875B2 (de) 1993-04-14
DK64591D0 (da) 1991-04-11
KR850006174A (ko) 1985-10-02
RO90953A (ro) 1987-02-27
ES8603409A1 (es) 1985-12-16
CA1253490C (de) 1989-05-02
EG17274A (en) 1989-06-30
AR247885A1 (es) 1995-04-28
FI85265B (fi) 1991-12-13
PT80116A (en) 1985-04-01
DK64591A (da) 1991-04-11
IE850683L (en) 1985-09-19
EP0155828A3 (en) 1986-02-05
DK165179B (da) 1992-10-19
EP0155828A2 (de) 1985-09-25
ES541373A0 (es) 1985-12-16
MA20379A1 (fr) 1985-10-01
PL252433A1 (en) 1985-12-03
DK163662C (da) 1992-08-31
FI851068A0 (fi) 1985-03-18
BG44203A3 (en) 1988-10-14
DK121485D0 (da) 1985-03-18
JPH03178963A (ja) 1991-08-02
YU42885A (en) 1987-10-31
NO168639C (no) 1992-03-18
DK121485A (da) 1985-09-20
HU194825B (en) 1988-03-28
EP0155828B1 (de) 1990-09-19
FI851068L (fi) 1985-09-20
AU552119B2 (en) 1986-05-22
DK163662B (da) 1992-03-23
ZW4885A1 (en) 1985-06-26
PL145873B1 (en) 1988-11-30
IE57741B1 (en) 1993-03-24
CA1250832A (en) 1989-03-07
OA07967A (fr) 1987-01-31
DK165179C (da) 1993-03-01
YU43869B (en) 1989-12-31
IL74630A0 (en) 1985-06-30
NZ211487A (en) 1988-11-29
KR860001874B1 (ko) 1986-10-24
CY1667A (en) 1993-05-14
FI85265C (fi) 1992-03-25

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