CS208658B2 - Method of makingthe derivatives of the 3-amino-17aaza-d-homo-5alfaandrostane - Google Patents

Method of makingthe derivatives of the 3-amino-17aaza-d-homo-5alfaandrostane

Info

Publication number
CS208658B2
CS208658B2 CS785347A CS534778A CS208658B2 CS 208658 B2 CS208658 B2 CS 208658B2 CS 785347 A CS785347 A CS 785347A CS 534778 A CS534778 A CS 534778A CS 208658 B2 CS208658 B2 CS 208658B2
Authority
CS
Czechoslovakia
Prior art keywords
alpha
homo
formula
aza
androstane
Prior art date
Application number
CS785347A
Other languages
Czech (cs)
English (en)
Inventor
Zoltan Tuba
Maria Marsai
Sandor Goeroeg
Katalin Biro
Egon Karpati
Laszlo Szporny
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of CS208658B2 publication Critical patent/CS208658B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A63—SPORTS; GAMES; AMUSEMENTS
    • A63H—TOYS, e.g. TOPS, DOLLS, HOOPS OR BUILDING BLOCKS
    • A63H1/00—Tops
    • A63H1/32—Whirling or spinning discs driven by twisted cords

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
CS785347A 1977-08-18 1978-08-16 Method of makingthe derivatives of the 3-amino-17aaza-d-homo-5alfaandrostane CS208658B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU77RI644A HU175287B (hu) 1977-08-18 1977-08-18 Sposob poluchenija novykh proizvodnykh 3-amino-17al'fa-aza-d-gomo-androstana,dalee ikh kislotoaddicionnykh i chetvjortichnykh solej

Publications (1)

Publication Number Publication Date
CS208658B2 true CS208658B2 (en) 1981-09-15

Family

ID=11001041

Family Applications (1)

Application Number Title Priority Date Filing Date
CS785347A CS208658B2 (en) 1977-08-18 1978-08-16 Method of makingthe derivatives of the 3-amino-17aaza-d-homo-5alfaandrostane

Country Status (18)

Country Link
US (1) US4200636A (nl)
JP (1) JPS5448799A (nl)
AT (1) AT364096B (nl)
AU (1) AU519292B2 (nl)
BE (1) BE869834A (nl)
CA (1) CA1110229A (nl)
CS (1) CS208658B2 (nl)
DD (1) DD138323A5 (nl)
DE (1) DE2835987A1 (nl)
DK (1) DK363278A (nl)
FR (1) FR2400525A1 (nl)
GB (1) GB2003479B (nl)
HU (1) HU175287B (nl)
IL (1) IL55352A0 (nl)
NL (1) NL190704C (nl)
PL (1) PL113864B1 (nl)
SE (1) SE436885B (nl)
YU (1) YU40920B (nl)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5140022A (en) * 1990-10-01 1992-08-18 Anaquest, Inc. 3-acyclic or cyclicaminomethyl-17a-lower-alkyl-17a-aza-d-homo-5-alpha-androstanes
US5229511A (en) * 1990-10-01 1993-07-20 Anaquest, Inc. 3-substituted-aminomethyl-3-substituted-oxy-17A-methyl-17A-lower-alkyl-17A-aza-d-homo-5-alpha-androstanes
GB2331988B (en) * 1997-12-04 2003-04-16 Imperial College Polycyclic sulphamate inhibitors or oestrone sulphatase
ES2314760T3 (es) 2001-10-18 2009-03-16 Sterix Limited Compuestos esteroideos para la inhibicion de la sulfatasa esteroidea.
WO2016084790A1 (ja) * 2014-11-25 2016-06-02 第一三共株式会社 ヒドロナフトキノリン誘導体

Also Published As

Publication number Publication date
AU3896678A (en) 1980-02-21
YU40920B (en) 1986-08-31
DK363278A (da) 1979-02-19
CA1110229A (en) 1981-10-06
FR2400525A1 (fr) 1979-03-16
GB2003479B (en) 1982-05-26
FR2400525B1 (nl) 1982-06-11
US4200636A (en) 1980-04-29
YU197078A (en) 1982-10-31
JPS5448799A (en) 1979-04-17
NL190704C (nl) 1994-07-01
SE436885B (sv) 1985-01-28
PL113864B1 (en) 1981-01-31
SE7808703L (sv) 1979-02-19
NL190704B (nl) 1994-02-01
BE869834A (fr) 1978-12-18
IL55352A0 (en) 1978-10-31
HU175287B (hu) 1980-06-28
DD138323A5 (de) 1979-10-24
AU519292B2 (en) 1981-11-19
PL209122A1 (pl) 1979-06-04
GB2003479A (en) 1979-03-14
NL7808543A (nl) 1979-02-20
DE2835987A1 (de) 1979-03-01
AT364096B (de) 1981-09-25
ATA597078A (de) 1981-02-15

Similar Documents

Publication Publication Date Title
IL49786A (en) Furo(orthieno)(3,2-c)pyridinium derivatives their preparation and pharmaceutical compositions containing them
JPS6049192B2 (ja) 新規置換ベンズアミド、その製造方法及びこれを有効成分とする向精神薬
BG61324B2 (bg) Азабициклононил-индазол-карбоксамид,притежаващ 5-нт активност като антагонист
US3987177A (en) Vincaminic acid esters
AU2018302026A1 (en) TLR7/8 antagonists and uses thereof
US4234584A (en) Substituted phenylpiperazine derivatives
TW202146400A (zh) 酞嗪酮類化合物及其製備方法和醫藥用途
CN112839944B (zh) 用于治疗狂犬病的化合物及其方法
CS207666B2 (en) Method of making the 2-bromergosin and the additive salts thereof with the acid
CS208658B2 (en) Method of makingthe derivatives of the 3-amino-17aaza-d-homo-5alfaandrostane
DE2718707A1 (de) Isothiazolopyridine, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeparate
DK164551B (da) Analogifremgangsmaade til fremstilling af cyclohexylthienyleddikesyreamider eller fysiologisk taalelige syreadditionssalte deraf
EP0279707A2 (en) Aryloxymethyl derivatives of nitrogenous heterocyclic methanols and ethers thereof having cardiovascular activity
CZ20014458A3 (cs) Polymorfní formy krystalického (2-benzhydryl-l-azabicyklo[2,2,2]okt-3-yl)-(5-isopropyl-2-methoxybenzyl) amoniumchloridu jako antagonisté receptoru NK-1
CS219885B2 (en) Method of making the n-lallyl-2-pyrolidylmethyl/-2,3-dimethoxy-5-sulphamoylbenzamide
US2807617A (en) Acylpiperazines and methods of preparing the same
GB2069480A (en) Process for the separation of the two optical isomers of moprolol and pharmaceutical compositions of the levorotatory antipode thereof
CS241475B2 (en) Method of 1,2-bis/(nicotinamido/)-propane preparation
Taborsky et al. Synthesis and preliminary pharmacology of some 1-methylindoles
SK281980B6 (sk) Kryštallický (+)l-hydrogenvínan, spôsob jeho prípravy, farmaceutický prostriedok s jeho obsahom a jeho použitie
KR20000029564A (ko) 5ＨＴ2ｃ길항제및Ｄ2길항제를함유하는약제학적조성물
PT85822B (pt) Processo para a preparacao de derivados de indolo-pirazino-benzodiazepina
US3671537A (en) Certain 3-(2,6-dichlorophenyl)-2-iminothiazolidines
SK695188A3 (en) Enolether amide 1,1-dioxo-6-chloro-4-hydroxy-2-methyl-n-(2- -pyridyl)-2h-thieno (2,3-e)-1,2-thiazine-3-carboxylic acid, method of its production and pharmaceutical agent
PT92494B (pt) Processo para a preparacao de novos derivados do indol