CR20150610A - Compuestos de pirimidino sustituido y derivados para combatir plagas de animales - Google Patents

Compuestos de pirimidino sustituido y derivados para combatir plagas de animales

Info

Publication number
CR20150610A
CR20150610A CR20150610A CR20150610A CR20150610A CR 20150610 A CR20150610 A CR 20150610A CR 20150610 A CR20150610 A CR 20150610A CR 20150610 A CR20150610 A CR 20150610A CR 20150610 A CR20150610 A CR 20150610A
Authority
CR
Costa Rica
Prior art keywords
derivatives
animal pests
compounds replaced
combat animal
pirimidine
Prior art date
Application number
CR20150610A
Other languages
English (en)
Inventor
Arun Narine
Nina Gertrud Bandur
Joachim Dickhaut
Swetlana Derksen
Raffael Koller
Deyn Wolfgang Von
Jean-Yves Wach
Deborah L Culbertson
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of CR20150610A publication Critical patent/CR20150610A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Abstract

La presente invención provee compuestos novedosos útiles como inhibidores de proteasoma. La invención además provee composiciones farmacéuticas que comprenden los compuestos de la invención y métodos para utilizar las composiciones en el tratamiento de varias enfermedades.
CR20150610A 2013-04-11 2015-11-10 Compuestos de pirimidino sustituido y derivados para combatir plagas de animales CR20150610A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361810746P 2013-04-11 2013-04-11
PCT/EP2014/057344 WO2014167084A1 (en) 2013-04-11 2014-04-11 Substituted pyrimidinium compounds and derivatives for combating animal pests

Publications (1)

Publication Number Publication Date
CR20150610A true CR20150610A (es) 2016-04-12

Family

ID=50478847

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20150610A CR20150610A (es) 2013-04-11 2015-11-10 Compuestos de pirimidino sustituido y derivados para combatir plagas de animales

Country Status (16)

Country Link
US (2) US9730451B2 (es)
EP (1) EP2984089B1 (es)
JP (2) JP6449850B2 (es)
KR (2) KR102223216B1 (es)
CN (1) CN105121441B (es)
AR (1) AR096022A1 (es)
AU (1) AU2014253086B2 (es)
BR (1) BR112015021863B1 (es)
CA (1) CA2901559C (es)
CL (1) CL2015003001A1 (es)
CR (1) CR20150610A (es)
ES (1) ES2913139T3 (es)
MX (1) MX2015014204A (es)
PT (1) PT2984089T (es)
UA (1) UA115904C2 (es)
WO (1) WO2014167084A1 (es)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR096022A1 (es) * 2013-04-11 2015-12-02 Basf Se Compuestos de pirimidinio sustituido, útiles para combatir plagas de animales
ES2639487T3 (es) 2013-06-17 2017-10-26 Basf Se Compuestos de pirimidinio sustituidos y derivados para combatir plagas animales
JP7027329B2 (ja) * 2016-04-01 2022-03-01 ビーエーエスエフ ソシエタス・ヨーロピア 二環式化合物
EP3440062B1 (en) * 2016-04-06 2021-10-06 Boehringer Ingelheim Animal Health USA Inc. Process for the preparation of enantiomerically enriched isoxazoline compounds - crystalline toluene solvate of (s)-afoxolaner
EP3497102B1 (de) 2016-08-15 2022-12-07 Bayer CropScience Aktiengesellschaft Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel
JOP20190086A1 (ar) 2016-10-21 2019-04-18 Novartis Ag مشتقات نافثيريدينون جديدة واستخدامها في معالجة عدم انتظام ضربات القلب
EP3575286B1 (en) 2017-01-26 2022-05-11 Mitsui Chemicals Agro, Inc. Pyridone compound and bactericide for agricultural and horticultural use, which uses said compound as active ingredient
BR112019018126A2 (pt) 2017-03-31 2020-04-07 Basf Se composto, misturas, composição pesticida, métodos de controle de insetos, acarídeos ou nematoides, de proteção de plantas e de proteção de material de propagação vegetal e semente
JP7168556B2 (ja) 2017-04-10 2022-11-09 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
JP7134946B2 (ja) 2017-04-10 2022-09-12 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
RU2765748C2 (ru) 2017-04-11 2022-02-02 Мицуи Кемикалз Агро, Инк. Пиридоны и содержащие их сельскохозяйственные и садовые фунгициды в качестве активных ингредиентов
JP7263250B2 (ja) 2017-04-27 2023-04-24 ビーエーエスエフ ソシエタス・ヨーロピア 光学活性２，３－ジヒドロチアゾロ［３，２－ａ］ピリミジン－４－イウム化合物を製造する方法
WO2018202654A1 (en) 2017-05-03 2018-11-08 Basf Se Process for preparing chiral 2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium compounds
US11117863B2 (en) 2017-06-08 2021-09-14 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
WO2018229202A1 (en) 2017-06-16 2018-12-20 Basf Se Mesoionic imidazolium compounds and derivatives for combating animal pests
BR112019025191B1 (pt) 2017-06-19 2023-11-28 Basf Se Compostos de pirimidínio substituídos, composição, método para proteger culturas, semente revestida, uso dos compostos e uso de um composto
WO2019042932A1 (en) * 2017-08-31 2019-03-07 Basf Se METHOD FOR CONTROLLING RICE PARASITES IN RICE
EP3694852A1 (en) * 2017-10-13 2020-08-19 Basf Se Imidazolidine pyrimidinium compounds for combating animal pests
WO2019086474A1 (en) 2017-10-31 2019-05-09 Syngenta Participations Ag Pesticidally active mesoionics heterocyclic compounds
WO2019115404A1 (en) 2017-12-13 2019-06-20 Syngenta Participations Ag Pesticidally active mesoionic heterocyclic compounds
PL3762368T3 (pl) 2018-03-08 2022-06-06 Incyte Corporation ZWIĄZKI AMINOPIRAZYNODIOLOWE JAKO INHIBITORY PI3K-γ
CN110317200B (zh) * 2018-03-28 2020-09-11 东莞市东阳光农药研发有限公司 嘧啶鎓化合物及其用途
CN110452238B (zh) * 2018-04-18 2020-08-11 东莞市东阳光农药研发有限公司 嘧啶鎓化合物及其用途
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
BR112021003324A2 (pt) 2018-09-19 2021-05-11 Basf Se misturas de pesticidas, composições, métodos de combate ou controle de pragas invertebradas, de proteção de plantas em crescimento e de proteção de material de propagação vegetal, uso de mistura de pesticidas e semente
EP3628158A1 (en) 2018-09-28 2020-04-01 Basf Se Pesticidal mixture comprising a mesoionic compound and a biopesticide
WO2020064492A1 (en) 2018-09-28 2020-04-02 Basf Se Method of controlling pests by seed treatment application of a mesoionic compound or mixture thereof
TWI780230B (zh) * 2018-09-28 2022-10-11 德商巴地斯顏料化工廠 用於製備含硫之嘧啶鎓化合物之方法
EP3628157A1 (en) 2018-09-28 2020-04-01 Basf Se Method of controlling insecticide resistant insects and virus transmission to plants
EP3628156A1 (en) 2018-09-28 2020-04-01 Basf Se Method for controlling pests of sugarcane, citrus, rapeseed, and potato plants
TWI804514B (zh) * 2018-09-28 2023-06-11 德商巴地斯顏料化工廠 用於對抗動物有害生物之嘧啶鎓化合物及其混合物
WO2020126591A1 (en) 2018-12-18 2020-06-25 Basf Se Substituted pyrimidinium compounds for combating animal pests
CN111620867A (zh) * 2019-02-28 2020-09-04 东莞市东阳光农药研发有限公司 介离子杀虫剂
EP3769623A1 (en) 2019-07-22 2021-01-27 Basf Se Mesoionic imidazolium compounds and derivatives for combating animal pests
CN113923987A (zh) 2019-05-29 2022-01-11 巴斯夫欧洲公司 用于防除动物害虫的介离子咪唑鎓化合物和衍生物
EP4032894A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate
EP4032886A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one
EP4032893A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate
EP4032878A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one
EP4063362A1 (en) 2021-03-25 2022-09-28 Basf Se Method for preparing enantiomerically enriched 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one by hydrogenation of the 2-oxo derivative in the presence of a chiral transition metal catalyst

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
TWI468407B (zh) * 2008-02-06 2015-01-11 Du Pont 中離子農藥
UA110924C2 (uk) * 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
UA107804C2 (en) * 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
MX2012001646A (es) * 2009-08-05 2012-03-21 Du Pont Pesticidas mesoionicos.
TWI528899B (zh) * 2010-12-29 2016-04-11 杜邦股份有限公司 中離子性殺蟲劑
CN103582639A (zh) 2011-04-06 2014-02-12 巴斯夫欧洲公司 用于防治动物害虫的取代嘧啶鎓化合物
AR096022A1 (es) * 2013-04-11 2015-12-02 Basf Se Compuestos de pirimidinio sustituido, útiles para combatir plagas de animales
ES2639487T3 (es) 2013-06-17 2017-10-26 Basf Se Compuestos de pirimidinio sustituidos y derivados para combatir plagas animales

Also Published As

Publication number Publication date
JP6449850B2 (ja) 2019-01-09
CN105121441B (zh) 2018-04-20
CA2901559C (en) 2021-11-02
US9730451B2 (en) 2017-08-15
ES2913139T3 (es) 2022-05-31
US11019820B2 (en) 2021-06-01
AU2014253086A1 (en) 2015-10-22
KR20150142025A (ko) 2015-12-21
CA2901559A1 (en) 2014-10-16
CN105121441A (zh) 2015-12-02
KR20210024256A (ko) 2021-03-04
WO2014167084A1 (en) 2014-10-16
KR102223216B1 (ko) 2021-03-04
AR096022A1 (es) 2015-12-02
US20180007905A1 (en) 2018-01-11
UA115904C2 (uk) 2018-01-10
BR112015021863A2 (pt) 2017-07-18
AU2014253086B2 (en) 2018-01-18
CL2015003001A1 (es) 2016-04-22
JP2016521264A (ja) 2016-07-21
EP2984089B1 (en) 2022-03-09
US20160058009A1 (en) 2016-03-03
MX2015014204A (es) 2015-12-11
BR112015021863A8 (pt) 2019-11-26
BR112015021863B1 (pt) 2020-08-18
EP2984089A1 (en) 2016-02-17
PT2984089T (pt) 2022-03-31
JP2019059759A (ja) 2019-04-18

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