CR20110225A - Composición estabilizada para el tratamiento de la psoriasis - Google Patents

Composición estabilizada para el tratamiento de la psoriasis

Info

Publication number
CR20110225A
CR20110225A CR20110225A CR20110225A CR20110225A CR 20110225 A CR20110225 A CR 20110225A CR 20110225 A CR20110225 A CR 20110225A CR 20110225 A CR20110225 A CR 20110225A CR 20110225 A CR20110225 A CR 20110225A
Authority
CR
Costa Rica
Prior art keywords
psoriasis
treatment
stabilized composition
alkyl
carboxylic ester
Prior art date
Application number
CR20110225A
Other languages
English (en)
Inventor
William Shifeng Wei
Yiping Wang
Jianzhen Pan
Sung Hi Jo
Original Assignee
Nexmed Holdings Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nexmed Holdings Inc filed Critical Nexmed Holdings Inc
Publication of CR20110225A publication Critical patent/CR20110225A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/59Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/221Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having an amino group, e.g. acetylcholine, acetylcarnitine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/3533,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A61K31/355Tocopherols, e.g. vitamin E
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Un ungüento estable al almacenamiento del presente invento que comprende un compuesto de vitamina D, un corticosteroide, y un alquilamino substituido de N,N-di(C1-C8) , un éster carboxílico(C2-C18) alquilo de (C4-C18) un éster carboxílico (C8-C22) alquilo de-(C1-C4)-en una base de ungüento de petrolato y opcionalmente conteniendo aceite mineral, y/o tocoferol.
CR20110225A 2008-10-03 2011-04-29 Composición estabilizada para el tratamiento de la psoriasis CR20110225A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19512608P 2008-10-03 2008-10-03

Publications (1)

Publication Number Publication Date
CR20110225A true CR20110225A (es) 2011-07-18

Family

ID=42073781

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20110225A CR20110225A (es) 2008-10-03 2011-04-29 Composición estabilizada para el tratamiento de la psoriasis

Country Status (18)

Country Link
US (2) US9220701B2 (es)
EP (1) EP2343978A4 (es)
JP (1) JP5667060B2 (es)
KR (1) KR20110067145A (es)
CN (1) CN102202509A (es)
AU (1) AU2009300331A1 (es)
BR (1) BRPI0920728A2 (es)
CA (1) CA2739376A1 (es)
CL (1) CL2011000722A1 (es)
CR (1) CR20110225A (es)
EC (1) ECSP11011022A (es)
IL (1) IL212062A0 (es)
MX (1) MX2011003568A (es)
NZ (1) NZ592300A (es)
PE (1) PE20110849A1 (es)
RU (1) RU2526162C2 (es)
WO (1) WO2010039251A1 (es)
ZA (1) ZA201103061B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ592300A (en) * 2008-10-03 2013-01-25 Nexmed Holdings Inc Stabilized composition for treating psoriasis
US11957753B2 (en) 2010-11-22 2024-04-16 Bausch Health Ireland Limited Pharmaceutical formulations containing corticosteroids for topical administration
US8809307B2 (en) * 2010-11-22 2014-08-19 Dow Pharmaceutical Sciences, Inc. Pharmaceutical formulations containing corticosteroids for topical administration
WO2014028780A2 (en) * 2012-08-15 2014-02-20 Nexmed Holdings, Inc. Antifungal compounds and methods of use
CN105784902A (zh) * 2016-03-11 2016-07-20 重庆华邦制药有限公司 低浓度丁酸氯倍他松的检测方法
EP3456314A1 (en) 2017-09-14 2019-03-20 Tiofarma B.V. Topical formulation comprising 17-ketolic corticosteroid
US20210196631A1 (en) * 2018-08-28 2021-07-01 Glenmark Pharmaceuticals Limited Container system and pharmaceutical foam composition comprising betamethasone

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4980378A (en) * 1988-06-01 1990-12-25 Odontex, Inc. Biodegradable absorption enhancers
US6046244A (en) 1997-11-05 2000-04-04 Nexmed Holdings, Inc. Topical compositions for prostaglandin E1 delivery
US6414028B1 (en) 1997-11-05 2002-07-02 Nexmed Holdings, Inc. Topical compositions containing prostaglandin E1
US8263580B2 (en) * 1998-09-11 2012-09-11 Stiefel Research Australia Pty Ltd Vitamin formulation
TR200101790T2 (tr) 1998-12-23 2001-10-22 Idea Ag. Yayılgan olmayan in vivo topik uygulamalar için geliştirilmiş formül
HU230045B1 (hu) 1999-04-23 2015-06-29 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) Bőrgyógyászati alkalmazásra szolgáló nem vizes gyógyszerkészítmény
JP2006511545A (ja) 2002-12-17 2006-04-06 ガルデルマ・ソシエテ・アノニム カルシトリオール及びプロピオン酸クロベタゾールの組み合わせ物を含む医薬組成物
DK1635770T3 (da) * 2003-03-21 2009-08-03 Nexmed Holdings Inc Antifungal neglelak og anvendelsesmetode
US20080069779A1 (en) * 2003-08-04 2008-03-20 Foamix Ltd. Foamable vehicle and vitamin and flavonoid pharmaceutical compositions thereof
FR2871696B1 (fr) * 2004-06-17 2006-11-10 Galderma Sa Composition topique pour le traitement du psoriasis
US20060057075A1 (en) * 2004-08-02 2006-03-16 Moshe Arkin Pharmaceutical and cosmeceutical wash-off mousse shampoo compositions, processes for preparing the same and uses thereof
CA2633489C (en) * 2005-12-14 2013-09-24 Zars Pharma, Inc. Compositions and methods for treating dermatological conditions
US7560489B2 (en) 2006-10-11 2009-07-14 Nexmed Holdings, Inc. Stabilized prostaglandin E composition
NZ592300A (en) * 2008-10-03 2013-01-25 Nexmed Holdings Inc Stabilized composition for treating psoriasis

Also Published As

Publication number Publication date
CL2011000722A1 (es) 2012-01-20
ZA201103061B (en) 2012-04-25
RU2011117230A (ru) 2012-11-10
US20110237558A1 (en) 2011-09-29
US9220701B2 (en) 2015-12-29
KR20110067145A (ko) 2011-06-21
NZ592300A (en) 2013-01-25
ECSP11011022A (es) 2011-06-30
BRPI0920728A2 (pt) 2015-08-18
JP2012504607A (ja) 2012-02-23
US20160067266A1 (en) 2016-03-10
PE20110849A1 (es) 2011-12-02
CN102202509A (zh) 2011-09-28
AU2009300331A1 (en) 2010-04-08
IL212062A0 (en) 2011-06-30
RU2526162C2 (ru) 2014-08-20
EP2343978A1 (en) 2011-07-20
CA2739376A1 (en) 2010-04-08
MX2011003568A (es) 2011-06-09
EP2343978A4 (en) 2013-11-27
WO2010039251A1 (en) 2010-04-08
JP5667060B2 (ja) 2015-02-12

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