CO6270185A2 - Derivados de isotiazol y pirazol como fungicidas - Google Patents

Derivados de isotiazol y pirazol como fungicidas

Info

Publication number
CO6270185A2
CO6270185A2 CO10001339A CO10001339A CO6270185A2 CO 6270185 A2 CO6270185 A2 CO 6270185A2 CO 10001339 A CO10001339 A CO 10001339A CO 10001339 A CO10001339 A CO 10001339A CO 6270185 A2 CO6270185 A2 CO 6270185A2
Authority
CO
Colombia
Prior art keywords
compound
heteroaryl
optionally substituted
hydrogen
alkyl
Prior art date
Application number
CO10001339A
Other languages
English (en)
Inventor
Peter Ackermann
Carla Bobbio
Camilla Corsi
Josef Ehrenfreund
Ann Monica Mcginley
Andreas Verras
Ruud Titulaer
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of CO6270185A2 publication Critical patent/CO6270185A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Abstract

1.- Un compuesto de Formula I:donde X es S, N o NR5 e Y es N o NR5, con la condicion de que uno de X o Y, pero no ambos, sea N; R1 y R3 son, independientemente, hidrogeno, o alquilo, alquenilo, alquinilo, heterociclilo, trialquilsililo, arilalquilo, ariloxialquilo, ariltioalquilo, arilo o heteroarilo, sustituido en forma opcional, con la condicion de que no sean ambos hidrogeno; R2 es alquilo, alquenilo, alquinilo, heterociclilo, arilalquilo, arilo o heteroarilo, sustituido en forma opcional; R4 es hidrogeno o un grupo que en condiciones biologicas puede disociarse para formar un alcohol en esta posicion; R5 es hidrogeno o alquilo, alquenilo, alquinilo, heterociclilo, trialquilsililo, arilalquilo, ariloxialquilo, ariltioalquilo, arilo o heteroarilo, sustituido en forma opcional; o una sal o N-oxido del mismo. 2.- El compuesto de la reivindicacion 1, donde X es S e Y es N. 3.- El compuesto de la reivindicacion 1, donde X es NR5 e Y es N. 4.- El compuesto de la reivindicacion 1, donde X es N e Y es NR5. 5.- El compuesto de cualquiera de las reivindicaciones 1 a 4, donde R1 y R3 son, independientemente, hidrogeno o alquilo, ariloxialquilo, ariltioalquilo, arilo o heteroarilo, sustituido en forma opcional. 6.- El compuesto de cualquiera de las reivindicaciones 1 a 4, donde R1 y R3 son, independientemente, hidrogeno o alquilo, fenilo o heteroarilo de 5 o 6 miembros sustituido en forma opcional.7.- El compuesto de cualquiera de las reivindicaciones precedentes, donde R2 es heteroarilo sustituido en forma opcional.
CO10001339A 2007-07-11 2010-01-07 Derivados de isotiazol y pirazol como fungicidas CO6270185A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0713479.4A GB0713479D0 (en) 2007-07-11 2007-07-11 Substituted aromatic heterocyclic compounds as fungicides

Publications (1)

Publication Number Publication Date
CO6270185A2 true CO6270185A2 (es) 2011-04-20

Family

ID=38461415

Family Applications (1)

Application Number Title Priority Date Filing Date
CO10001339A CO6270185A2 (es) 2007-07-11 2010-01-07 Derivados de isotiazol y pirazol como fungicidas

Country Status (21)

Country Link
US (1) US8377953B2 (es)
EP (1) EP2162448A1 (es)
JP (1) JP2010532775A (es)
KR (1) KR20100045435A (es)
CN (2) CN103012393A (es)
AR (1) AR066160A1 (es)
AU (1) AU2008274558B8 (es)
BR (1) BRPI0814623A2 (es)
CA (1) CA2692374C (es)
CL (1) CL2008002014A1 (es)
CO (1) CO6270185A2 (es)
CR (1) CR11197A (es)
EC (1) ECSP109862A (es)
EG (1) EG26050A (es)
GB (1) GB0713479D0 (es)
GT (1) GT200800139A (es)
IL (1) IL202811A0 (es)
RU (1) RU2010104397A (es)
TW (1) TW200918529A (es)
WO (1) WO2009007098A1 (es)
ZA (1) ZA200909222B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0823000D0 (en) * 2008-12-17 2009-01-28 Syngenta Participations Ag Isothiazole and pyrazole derivatives with plant growth regulating properties
BR112013001237A2 (pt) * 2010-07-19 2016-05-17 Syngenta Participations Ag compostos de isoxazola, isoatiazola, furano e tiofeno como microbicidas
TW201245155A (en) 2010-09-01 2012-11-16 Du Pont Fungicidal pyrazoles
WO2015171392A1 (en) * 2014-05-06 2015-11-12 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
CN112979633B (zh) * 2019-12-12 2024-02-02 东莞市东阳光农药研发有限公司 新的肟类衍生物及其制备方法和应用
EP4173485A1 (en) * 2021-10-27 2023-05-03 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Protein aggregation inhibiting compounds for plant disease control

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH069313A (ja) * 1992-06-29 1994-01-18 Mitsui Toatsu Chem Inc イソチアゾールカルボン酸アニリド誘導体を有効成分とするイネいもち病防除剤
JP3964478B2 (ja) * 1995-06-30 2007-08-22 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ環含有カルボン酸誘導体及びそれを含有する医薬
JP3966933B2 (ja) * 1996-11-28 2007-08-29 株式会社エス・ディー・エス バイオテック 置換ピラゾール誘導体、その製造方法およびそれを有効成分とする農園芸用殺菌剤
DE19838708A1 (de) * 1998-08-26 2000-03-02 Bayer Ag Verwendung von 5-Amino-pyrazol-Derivaten zur Bekämpfung von Mikroorganismen
DE10034129A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Pyrazolylbenzylether
AU3034801A (en) * 2000-01-28 2001-08-07 Syngenta Limited Isothiazole derivatives and their use as pesticides
GB0024795D0 (en) * 2000-10-10 2000-11-22 Hoffmann La Roche Pyrazole derivatives for the treatment of viral diseases
WO2002040473A1 (fr) * 2000-11-17 2002-05-23 Ishihara Sangyo Kaisha, Ltd. Composes de pyrimidine ou leurs sels, herbicides contenant ces composes ou ces sels, leur procede d'utilisation dans l'elimination des mauvaises herbes
SE0300119D0 (sv) * 2003-01-17 2003-01-17 Astrazeneca Ab Novel compounds
EP1794167A4 (en) 2004-09-10 2009-10-21 Syngenta Ltd SUBSTITUTED ISOXAZOLE AS FUNGICIDES
GB0823000D0 (en) * 2008-12-17 2009-01-28 Syngenta Participations Ag Isothiazole and pyrazole derivatives with plant growth regulating properties

Also Published As

Publication number Publication date
CN103012393A (zh) 2013-04-03
WO2009007098A1 (en) 2009-01-15
RU2010104397A (ru) 2011-08-20
CA2692374C (en) 2013-08-27
CA2692374A1 (en) 2009-01-15
US20110224241A1 (en) 2011-09-15
CL2008002014A1 (es) 2008-11-14
TW200918529A (en) 2009-05-01
CN101687845A (zh) 2010-03-31
AU2008274558A1 (en) 2009-01-15
ZA200909222B (en) 2010-09-29
EP2162448A1 (en) 2010-03-17
EG26050A (en) 2013-01-15
AU2008274558B8 (en) 2013-08-01
CR11197A (es) 2010-03-23
GB0713479D0 (en) 2007-08-22
GT200800139A (es) 2009-04-29
BRPI0814623A2 (pt) 2015-01-27
JP2010532775A (ja) 2010-10-14
US8377953B2 (en) 2013-02-19
ECSP109862A (es) 2010-02-26
IL202811A0 (en) 2010-06-30
AR066160A1 (es) 2009-07-29
AU2008274558B2 (en) 2013-07-18
KR20100045435A (ko) 2010-05-03
WO2009007098A8 (en) 2010-05-06

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