CO5160321A1 - Novedosas composiciones de tipranavir y ritonavir - Google Patents

Novedosas composiciones de tipranavir y ritonavir

Info

Publication number
CO5160321A1
CO5160321A1 CO99069669A CO99069669A CO5160321A1 CO 5160321 A1 CO5160321 A1 CO 5160321A1 CO 99069669 A CO99069669 A CO 99069669A CO 99069669 A CO99069669 A CO 99069669A CO 5160321 A1 CO5160321 A1 CO 5160321A1
Authority
CO
Colombia
Prior art keywords
tipranavir
ritonavir
new compositions
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
CO99069669A
Other languages
English (en)
Inventor
James J Ferry
John R Baldwin
Marie T Borin
Original Assignee
Pharmascia And Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmascia And Upjohn Company filed Critical Pharmascia And Upjohn Company
Publication of CO5160321A1 publication Critical patent/CO5160321A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Abstract

Una novedosa composición que comprende una cantidad terapéuticamente efectiva de tipranavir o una sal farmacéuticamente aceptable del mismo, y una cantidad terapéuticamente efectiva de ritonavir o una sal farmacéuticamente aceptable del mismo para mejorar la farmacocinética del tipranavir o para incrementar los niveles de tipranavir en sangre humana.
CO99069669A 1998-11-04 1999-11-04 Novedosas composiciones de tipranavir y ritonavir CO5160321A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10696398P 1998-11-04 1998-11-04

Publications (1)

Publication Number Publication Date
CO5160321A1 true CO5160321A1 (es) 2002-05-30

Family

ID=22314155

Family Applications (1)

Application Number Title Priority Date Filing Date
CO99069669A CO5160321A1 (es) 1998-11-04 1999-11-04 Novedosas composiciones de tipranavir y ritonavir

Country Status (13)

Country Link
US (1) US6147095A (es)
EP (1) EP1126847A1 (es)
JP (1) JP2002528502A (es)
CN (1) CN1154491C (es)
AU (1) AU762349B2 (es)
BR (1) BR9914940A (es)
CA (1) CA2346131C (es)
CO (1) CO5160321A1 (es)
HK (1) HK1040625B (es)
MY (1) MY118526A (es)
PE (1) PE20001296A1 (es)
TW (1) TW580387B (es)
WO (1) WO2000025784A1 (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9815567D0 (en) * 1998-07-18 1998-09-16 Glaxo Group Ltd Antiviral compound
EE200300201A (et) * 2000-10-31 2003-08-15 Boehringer Ingelheim Pharmaceuticals, Inc. Püranoonsete proteaasi inhibiitorite iseemulgeeruva kompositsiooni oraalne doos
US6500963B2 (en) 2001-02-22 2002-12-31 Boehringer Ingelheim Pharma Kg Process for preparing optically active dihydropyrones
DE10108470A1 (de) * 2001-02-22 2002-09-05 Boehringer Ingelheim Pharma Verfahren zur Herstellung optisch aktiver Dihydropyrone
US20030180279A1 (en) * 2002-03-19 2003-09-25 Tibor Sipos Composition and method to prevent or reduce diarrhea and steatorrhea in HIV patients
US20040197321A1 (en) * 2002-03-19 2004-10-07 Tibor Sipos Composition and method to prevent or reduce diarrhea and steatorrhea in HIV patients
US20040152625A1 (en) * 2002-12-16 2004-08-05 Boehringer Ingelheim International Gmbh Method for improving the pharmacokinetics of an NNRTI
AU2003295940A1 (en) * 2002-12-16 2004-07-29 Boehringer Ingelheim Pharmaceuticals, Inc. Treatment of hiv infection through combined administration of tipranavir and capravirine
WO2004087139A1 (en) * 2003-03-27 2004-10-14 Boehringer Ingelheim International Gmbh Antiviral combination of tipranavir and a further antiretroviral compound
AR045841A1 (es) * 2004-09-28 2005-11-16 Richmond Sa Com Ind Y Financie Una composicion farmaceutica solida que comprende al tiazolil metil ester del acido [5s-(5r*, 8r*, 10r*,11r*)] -10- hidroxi-2- metil-5-(1-metiletil)-1-[2-(1-metiletil)-4-tiazolil]-3,6-dioxo-8,11-bis(fenilmetil)-2,4,7,12- tetraazatridecan-13-oico y un procedimiento para prepararla.
CA2583187A1 (en) * 2004-11-08 2006-05-18 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and etravirine
US20060135562A1 (en) * 2004-11-16 2006-06-22 Boehringer Ingelheim International Gmbh Method for treating HIV infection through co-administration of tipranavir and darunavir
JP2008520701A (ja) * 2004-11-19 2008-06-19 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング チプラナビル及びレバーセットの同時投与を介したhiv感染症の治療方法
WO2006055660A2 (en) * 2004-11-19 2006-05-26 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and uk-427, 857
US20060160859A1 (en) * 2004-12-01 2006-07-20 Boehringer Ingelheim International Gmbh Method for treating HIV infection through co-administration of tipranavir and GW873140
EP1819335A1 (en) * 2004-12-01 2007-08-22 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and sch-417690
CA2586501A1 (en) * 2004-12-01 2006-06-08 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and gw695634
US8598364B2 (en) 2007-03-12 2013-12-03 Nektar Therapeutics Oligomer-protease inhibitor conjugates
WO2009114151A1 (en) * 2008-03-12 2009-09-17 Nektar Therapeutics Oligomer-amino acid and olgomer-atazanavir conjugates
US20100021505A1 (en) * 2008-07-28 2010-01-28 Tibor Sipos Composition and method to prevent or reduce diarrhea and steatorrhea in HIV patients
WO2010144869A2 (en) 2009-06-12 2010-12-16 Nektar Therapeutics Protease inhibitors
MA34215B1 (fr) * 2010-04-02 2013-05-02 Phivco 1 Llc Traitement d'association comprenant un antagoniste du récepteur ccr5, un inhibiteur de la protéase du vih-1 et un accélérateur pharmacocinétique
WO2012166795A1 (en) * 2011-05-30 2012-12-06 String Therapeutics Inc. Methods and compositions for therapeutic drug monitoring and dosing by point-of-care pharmacokinetic profiling

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5608085A (en) * 1995-02-27 1997-03-04 The University Of Tennessee Research Corporation Synthesis of optically active calanolides A and B and enantiomers and related compounds
US6037157A (en) * 1995-06-29 2000-03-14 Abbott Laboratories Method for improving pharmacokinetics
US5932570A (en) * 1996-11-08 1999-08-03 Dupont Pharmaceuticals Company 1-(3-aminoindazol-5-yl)-3-phenylmethyl-cyclic ureas useful as HIV protease inhibitors
ZA9710071B (en) * 1996-11-21 1998-05-25 Abbott Lab Pharmaceutical composition.

Also Published As

Publication number Publication date
JP2002528502A (ja) 2002-09-03
CN1154491C (zh) 2004-06-23
TW580387B (en) 2004-03-21
HK1040625A1 (en) 2002-06-21
MY118526A (en) 2004-11-30
CA2346131A1 (en) 2000-05-11
PE20001296A1 (es) 2000-11-23
CN1324237A (zh) 2001-11-28
AU762349B2 (en) 2003-06-26
WO2000025784A1 (en) 2000-05-11
EP1126847A1 (en) 2001-08-29
CA2346131C (en) 2013-01-15
BR9914940A (pt) 2001-07-10
US6147095A (en) 2000-11-14
AU1440400A (en) 2000-05-22
HK1040625B (zh) 2005-04-01

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