CO4480739A1 - Formas zwitterionicas de trovafloxacina - Google Patents

Formas zwitterionicas de trovafloxacina

Info

Publication number
CO4480739A1
CO4480739A1 CO96046149A CO96046149A CO4480739A1 CO 4480739 A1 CO4480739 A1 CO 4480739A1 CO 96046149 A CO96046149 A CO 96046149A CO 96046149 A CO96046149 A CO 96046149A CO 4480739 A1 CO4480739 A1 CO 4480739A1
Authority
CO
Colombia
Prior art keywords
drying
hygroscopic
hygroscopic polymorph
pentahydrate
treat
Prior art date
Application number
CO96046149A
Other languages
English (en)
Spanish (es)
Inventor
Allen Douglas John Meldrum
Joseph David Bruning
Timothy Norris
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CO4480739A1 publication Critical patent/CO4480739A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Physical Water Treatments (AREA)
  • Processing Of Solid Wastes (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CO96046149A 1995-08-29 1996-08-29 Formas zwitterionicas de trovafloxacina CO4480739A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US297595P 1995-08-29 1995-08-29

Publications (1)

Publication Number Publication Date
CO4480739A1 true CO4480739A1 (es) 1997-07-09

Family

ID=21703460

Family Applications (1)

Application Number Title Priority Date Filing Date
CO96046149A CO4480739A1 (es) 1995-08-29 1996-08-29 Formas zwitterionicas de trovafloxacina

Country Status (30)

Country Link
EP (1) EP0850060A1 (fr)
JP (1) JP3188476B2 (fr)
KR (1) KR100343909B1 (fr)
CN (1) CN1190889A (fr)
AP (1) AP636A (fr)
AR (1) AR003985A1 (fr)
AU (1) AU704115B2 (fr)
BR (1) BR9609998A (fr)
CA (1) CA2229786C (fr)
CO (1) CO4480739A1 (fr)
CZ (1) CZ56698A3 (fr)
DZ (1) DZ2087A1 (fr)
GT (1) GT199600072A (fr)
HR (1) HRP960395B1 (fr)
HU (1) HUP9900170A3 (fr)
IL (1) IL122651A (fr)
MA (1) MA23966A1 (fr)
MY (1) MY113874A (fr)
NO (1) NO309814B1 (fr)
NZ (1) NZ312199A (fr)
OA (1) OA10669A (fr)
PE (1) PE12598A1 (fr)
PL (1) PL325170A1 (fr)
RU (1) RU2144921C1 (fr)
SK (1) SK23898A3 (fr)
TN (1) TNSN96109A1 (fr)
TR (1) TR199800339T1 (fr)
WO (1) WO1997007800A1 (fr)
YU (1) YU48396A (fr)
ZA (1) ZA967282B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (es) 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
US7019142B2 (en) 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
PA8466701A1 (es) * 1998-01-21 2000-09-29 Pfizer Prod Inc Comprimido de mesilato de trovafloxacino
US6114531A (en) * 1998-07-28 2000-09-05 Pfizer Inc. Process for preparing quinolone and naphthyridone carboxylic acids
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.
US6239141B1 (en) 1999-06-04 2001-05-29 Pfizer Inc. Trovafloxacin oral suspensions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids

Also Published As

Publication number Publication date
ZA967282B (en) 1998-03-02
CZ56698A3 (cs) 1999-02-17
AP636A (en) 1998-04-09
BR9609998A (pt) 1999-07-06
SK23898A3 (en) 1999-05-07
DZ2087A1 (fr) 2002-07-22
NZ312199A (en) 1999-06-29
JP3188476B2 (ja) 2001-07-16
YU48396A (sh) 1998-12-23
WO1997007800A1 (fr) 1997-03-06
CA2229786A1 (fr) 1997-03-06
JPH10511692A (ja) 1998-11-10
AU704115B2 (en) 1999-04-15
TR199800339T1 (xx) 1998-06-22
AU6367696A (en) 1997-03-19
CN1190889A (zh) 1998-08-19
HUP9900170A3 (en) 1999-11-29
PE12598A1 (es) 1998-03-20
EP0850060A1 (fr) 1998-07-01
MA23966A1 (fr) 1997-04-01
NO309814B1 (no) 2001-04-02
KR100343909B1 (ko) 2003-04-10
GT199600072A (es) 1998-02-14
AP9600853A0 (en) 1996-10-31
HRP960395B1 (en) 2001-12-31
IL122651A (en) 2000-02-17
MX9801664A (es) 1998-08-30
OA10669A (en) 2000-11-06
HRP960395A2 (en) 1998-06-30
PL325170A1 (en) 1998-07-06
AR003985A1 (es) 1998-09-30
IL122651A0 (en) 1998-08-16
NO980862D0 (no) 1998-02-27
CA2229786C (fr) 2002-02-19
HUP9900170A2 (hu) 1999-05-28
TNSN96109A1 (fr) 2005-03-15
RU2144921C1 (ru) 2000-01-27
NO980862L (no) 1998-02-27
MY113874A (en) 2002-06-29
KR19990044232A (ko) 1999-06-25

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