CO2022002493A2 - Nanoemulsion de ácido 18p-glicirretínico - Google Patents

Nanoemulsion de ácido 18p-glicirretínico

Info

Publication number
CO2022002493A2
CO2022002493A2 CONC2022/0002493A CO2022002493A CO2022002493A2 CO 2022002493 A2 CO2022002493 A2 CO 2022002493A2 CO 2022002493 A CO2022002493 A CO 2022002493A CO 2022002493 A2 CO2022002493 A2 CO 2022002493A2
Authority
CO
Colombia
Prior art keywords
glycyrrhetinic acid
formulation
nanoemulsion
treatment
acid nanoemulsion
Prior art date
Application number
CONC2022/0002493A
Other languages
English (en)
Inventor
Hernández Ulises Zendejas
Original Assignee
Atso Corp Affairs S A De C V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Atso Corp Affairs S A De C V filed Critical Atso Corp Affairs S A De C V
Publication of CO2022002493A2 publication Critical patent/CO2022002493A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Formulación farmacéutica que comprende ácidβ 18 -glicirretínico, siendo dicha formulación una nanoemulsión con el objeto de potenciar la biodisponibilidad del principio activo, método de preparación de la formulación y su uso en el tratamiento de infecciones causadas por el virus del papiloma humano. Está pensada para la aplicación en la zona vaginal y del cérvix para el tratamiento de infecciones causadas por el virus del papiloma humano, como el cáncer cervicouterino.
CONC2022/0002493A 2019-08-08 2022-03-01 Nanoemulsion de ácido 18p-glicirretínico CO2022002493A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
MX2019009482A MX2019009482A (es) 2019-08-08 2019-08-08 FORMAS FARMACEUTICAS DEL ACIDO 18ß-GLICIRRETINICO.
PCT/MX2020/050025 WO2021025550A1 (es) 2019-08-08 2020-08-07 Nanoemulsion de ácido 18p-glicirretínico

Publications (1)

Publication Number Publication Date
CO2022002493A2 true CO2022002493A2 (es) 2022-04-29

Family

ID=74503526

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2022/0002493A CO2022002493A2 (es) 2019-08-08 2022-03-01 Nanoemulsion de ácido 18p-glicirretínico

Country Status (9)

Country Link
US (1) US20220296544A1 (es)
EP (1) EP4023219A4 (es)
CN (1) CN114450001A (es)
BR (1) BR112022002176A2 (es)
CA (1) CA3147206A1 (es)
CO (1) CO2022002493A2 (es)
MX (1) MX2019009482A (es)
WO (1) WO2021025550A1 (es)
ZA (1) ZA202202125B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023159476A1 (en) 2022-02-25 2023-08-31 L'oreal Composition for caring for keratin materials

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2072014B (en) * 1980-03-08 1984-02-15 Kanebo Ltd Cosmetics containing 18-glycyrrhizins
LU86396A1 (fr) * 1986-04-18 1986-09-02 Pharma Roche Posay Lab Compositions pour le traitement de la calvitie et des alopecies
MX351117B (es) * 2011-02-25 2017-10-03 Desarrollos Vph S A De C V Formulacion de la sal acido glicirricinico en gel termorreversible y acido tricloroacetico para su aplicacion en el tracto genital de mujeres y varones con lesiones causadas por el virus del papiloma humano y cancer en los mismos.
RU2493852C1 (ru) * 2012-04-12 2013-09-27 Леонид Леонидович Клопотенко Композиция, содержащая фермент дезоксирибонуклеазу и/или стеарилглицирретинат или глицирризиновую кислоту или ее соли: глицирризинат аммония, или дикалия, или тринатрия
CN105342987A (zh) * 2015-12-04 2016-02-24 亚飞(上海)生物医药科技有限公司 一种凝胶及其制备方法和应用
ITUB20159218A1 (it) * 2015-12-21 2017-06-21 Valitudo Pharma Srls Composizione, per uso topico, utile per favorire la cicatrizzazione di lesioni sulla pelle.
MX2017010806A (es) * 2017-08-22 2018-01-18 Atso Corp Affairs S A De C V Formulacion de acido 18-beta-glicirretinico en combinacion con revesterol y metformina, usos y metodo de fabricacion.

Also Published As

Publication number Publication date
EP4023219A1 (en) 2022-07-06
CA3147206A1 (en) 2021-02-11
WO2021025550A1 (es) 2021-02-11
BR112022002176A2 (pt) 2022-05-03
CN114450001A (zh) 2022-05-06
MX2019009482A (es) 2021-02-09
US20220296544A1 (en) 2022-09-22
ZA202202125B (en) 2023-11-29
EP4023219A4 (en) 2023-04-26

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