CO2022001663A2 - Composiciones medicinales y/o farmacéuticas para la instilación intravesical, preparación y uso de las mismas - Google Patents

Composiciones medicinales y/o farmacéuticas para la instilación intravesical, preparación y uso de las mismas

Info

Publication number
CO2022001663A2
CO2022001663A2 CONC2022/0001663A CO2022001663A CO2022001663A2 CO 2022001663 A2 CO2022001663 A2 CO 2022001663A2 CO 2022001663 A CO2022001663 A CO 2022001663A CO 2022001663 A2 CO2022001663 A2 CO 2022001663A2
Authority
CO
Colombia
Prior art keywords
advantageously
composition
salt
urethra
bladder
Prior art date
Application number
CONC2022/0001663A
Other languages
English (en)
Inventor
Sándor Lovász
Gábor Rényi
János Giber
Péter Birinyi
Original Assignee
Lovasz Sandor
Renyi Gabor
Giber Janos
Birinyi Peter
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from HU2000094A external-priority patent/HUP2000094A1/hu
Application filed by Lovasz Sandor, Renyi Gabor, Giber Janos, Birinyi Peter filed Critical Lovasz Sandor
Publication of CO2022001663A2 publication Critical patent/CO2022001663A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/726—Glycosaminoglycans, i.e. mucopolysaccharides
    • A61K31/727—Heparin; Heparan
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/726—Glycosaminoglycans, i.e. mucopolysaccharides
    • A61K31/728—Hyaluronic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/737—Sulfated polysaccharides, e.g. chondroitin sulfate, dermatan sulfate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención se refiere a nuevas composiciones medicinales y/o farmacéuticas indicadas como composición A y composición B en forma líquida para usarse a manera de una composición medicinal o medicamento para la instilación intravesical, en el tratamiento local simultáneo de enfermedades de la uretra y/o la vejiga, en donde las composiciones A y B son para usarse ventajosamente en el tratamiento contra el síndrome de dolor vesical (cistitis intersticial), en la uretra, y mediante la reposición de la capa GAG en la superficie interna de la vejiga; además, ventajosamente la composición A es para usarse en el tratamiento analgésico y anestésico local de la uretra y/o la vejiga, y además, de manera ventajosa en el tratamiento contra la inflamación de la uretra y/o la vejiga, y su preparación. De acuerdo con el uso de las composiciones del tema de la invención, el tratamiento contra IC/BPS se implementa en dos etapas usando la primera composición A y en segundo lugar la composición B para la instilación intravesical a través de la uretra. También se optimizan la osmolaridad y el pH de las composiciones. De acuerdo con la el tema de la invención, la composición A comprende los siguientes componentes: El anestésico local, ventajosamente lidocaína o una sal adecuada de la misma, un corticosteroide, ventajosamente dexametasona-disodio-difosfato o agente antiinflamatorio no esteroideo, ventajosamente sal de diclofenaco, en donde además, ventajosamente el anestésico local y el agente antiinflamatorio no esteroideo y las formas ventajosas de los mismos están incrustados en el liposoma o además, ventajosamente están componiendo complejos con un agente de composición de complejos; alcalino básico, ventajosamente hidróxido de sodio; agua destilada estéril; sal alcalina, de manera ventajosa cloruro de sodio. De acuerdo con la materia de la invención, adicionalmente la composición B comprende los siguientes componentes: Ácido hialurónico o una sal alcalina adecuada del mismo, ventajosamente hialuronato de sodio, sal alcalina de sulfato de condroitina, ventajosamente condroitina-sulfato de sodio, heparina, ventajosamente sal sódica de heparina; básico alcalino, ventajosamente hidróxido de sodio o bicarbonato de sodio, agua destilada estéril, sal alcalina, ventajosamente cloruro de sodio y sal de metal alcalinotérreo, ventajosamente cloruro de calcio.
CONC2022/0001663A 2019-07-18 2022-02-17 Composiciones medicinales y/o farmacéuticas para la instilación intravesical, preparación y uso de las mismas CO2022001663A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
HUP1900257 2019-07-18
HU2000094A HUP2000094A1 (hu) 2020-03-12 2020-03-12 Gyógyászati és/vagy gyógyszerkészítmény intravezikális instillációra, elõállításuk és alkalmazásuk
PCT/HU2020/000026 WO2021009525A1 (en) 2019-07-18 2020-09-15 Medicinal and/or pharmaceutical compositions for intravesical instillation, preparation and use thereof

Publications (1)

Publication Number Publication Date
CO2022001663A2 true CO2022001663A2 (es) 2022-07-19

Family

ID=89666444

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2022/0001663A CO2022001663A2 (es) 2019-07-18 2022-02-17 Composiciones medicinales y/o farmacéuticas para la instilación intravesical, preparación y uso de las mismas

Country Status (8)

Country Link
US (1) US20220273698A1 (es)
EP (1) EP3999028A1 (es)
JP (1) JP2022540702A (es)
AU (1) AU2020314184A1 (es)
CA (1) CA3147879A1 (es)
CO (1) CO2022001663A2 (es)
IL (1) IL289943A (es)
WO (1) WO2021009525A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020252003A1 (en) 2019-06-13 2020-12-17 Hollister Incorporated Reusable urinary catheter products
US12440644B2 (en) 2019-06-25 2025-10-14 Hollister Incorporated Reusable urinary catheter products
GB2639834A (en) * 2024-03-22 2025-10-08 Remicine Ip B V Composition and method of treatment

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6083933A (en) * 1999-04-19 2000-07-04 Stellar International Inc. Treatment of cystitis-like symptoms with chondroitin sulfate following administration of a challenge solution
CN1557290A (zh) * 2004-01-19 2004-12-29 江苏扬子江药业集团有限公司 复方双氯芬酸钾注射液制剂
SI1708722T1 (sl) * 2004-01-28 2014-10-30 The Regents Of The University Of California Nova intersticijska terapija za takojšnje simptome sprostitve in kronična terapija pri intersticijskem cistitisu
WO2007073397A1 (en) * 2005-12-19 2007-06-28 Urigen, Inc. Kits and improved compositions for treating lower urinary tract discorders
US9849086B2 (en) * 2012-03-19 2017-12-26 Nanologix Research, Inc. Method and composition for treating cystitis
EP3400950B1 (de) * 2017-05-12 2019-11-13 Farco-Pharma GmbH Blaseninstillationszusammensetzung enthaltend chondoitinsulfat (20 mg/ml), hyaluronsäure (16 mg/ml) und phosphatpuffer (ph 6,1 bis 7,9) mit erhöhter lagerstabiliät zur behandlung von cystitis
CN109568333A (zh) * 2018-12-26 2019-04-05 江西润泽药业有限公司 一种治疗鼻炎的滴鼻液及其制备方法

Also Published As

Publication number Publication date
JP2022540702A (ja) 2022-09-16
US20220273698A1 (en) 2022-09-01
WO2021009525A1 (en) 2021-01-21
CA3147879A1 (en) 2021-01-21
AU2020314184A1 (en) 2022-03-10
IL289943A (en) 2022-03-01
EP3999028A1 (en) 2022-05-25

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