CN1221254C - 新的作为药用配制品的血清素激动剂(5ht2)和拮抗剂(5ht6)复合剂 - Google Patents
新的作为药用配制品的血清素激动剂(5ht2)和拮抗剂(5ht6)复合剂 Download PDFInfo
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- CN1221254C CN1221254C CNB018131549A CN01813154A CN1221254C CN 1221254 C CN1221254 C CN 1221254C CN B018131549 A CNB018131549 A CN B018131549A CN 01813154 A CN01813154 A CN 01813154A CN 1221254 C CN1221254 C CN 1221254C
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SE0002754A SE0002754D0 (sv) | 2000-07-21 | 2000-07-21 | New pharmaceutical combination formulation and method of treatment with the combination |
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WO (1) | WO2002008178A1 (sh) |
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Cited By (1)
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CN107628981A (zh) * | 2017-10-31 | 2018-01-26 | 威海市妇女儿童医院 | 一种肉桂酰基吲哚啉化合物及其制备青光眼药物的应用 |
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US7034029B2 (en) | 2000-11-02 | 2006-04-25 | Wyeth | 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands |
HUP0303756A3 (en) * | 2000-11-02 | 2009-08-28 | Wyeth Corp | 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands and process for their preparation and pharmaceutical compositions containing them |
CN1321110C (zh) * | 2001-06-15 | 2007-06-13 | 弗·哈夫曼-拉罗切有限公司 | 具有5-ht6受体亲和力的4-哌嗪基吲哚衍生物 |
JP2005501019A (ja) * | 2001-06-15 | 2005-01-13 | エフ.ホフマン−ラ ロシュ アーゲー | 5−ht6レセプター親和性を有する4−ピペラジニルインドール誘導体 |
US6825198B2 (en) | 2001-06-21 | 2004-11-30 | Pfizer Inc | 5-HT receptor ligands and uses thereof |
GB0202679D0 (en) * | 2002-02-05 | 2002-03-20 | Glaxo Group Ltd | Novel compounds |
PT1497266E (pt) | 2002-03-27 | 2008-09-10 | Glaxo Group Ltd | Derivados de quinolina e sua utilização como ligandos 5-ht6 |
CL2004000826A1 (es) * | 2003-04-25 | 2005-03-04 | Pfizer | Uso de un agonista para el receptor 5-ht2c para preparar un medicamento util en el tratamiento de la incontinencia urinaria provocada por estres, con la condicion de que el agonista no sea 1-[6-cloro-5-(trifluorometil)-2-piridinil]piperazina (org-129 |
MXPA06000795A (es) | 2003-07-22 | 2006-08-23 | Arena Pharm Inc | Derivados de diaril y arilheteroaril urea como moduladores del receptor 5-ht2a de serotonina utiles para la profilaxis y tratamiento de desordenes relacionados con el mismo. |
EP2400300A1 (en) | 2004-08-25 | 2011-12-28 | Takeda Pharmaceutical Company Limited | Method of screening preventives/remedies for stress urinary incontinence |
US7713954B2 (en) | 2004-09-30 | 2010-05-11 | Roche Palo Alto Llc | Compositions and methods for treating cognitive disorders |
WO2007076875A2 (en) * | 2006-01-06 | 2007-07-12 | Aarhus Universitet | Compounds acting on the serotonin transporter |
US8158617B2 (en) | 2006-05-16 | 2012-04-17 | Takeda Pharmaceutical Company Limited | Fused heterocyclic compound and use thereof |
WO2007149728A2 (en) * | 2006-06-20 | 2007-12-27 | Alcon Research, Ltd. | Aryl and heteroaryl tetrahydrobenzazepine derivatives and their use for treating glaucoma |
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DZ2376A1 (fr) * | 1996-12-19 | 2002-12-28 | Smithkline Beecham Plc | Dérivés de sulfonamides nouveaux procédé pour leurpréparation et compositions pharmaceutiques les c ontenant. |
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US6100291A (en) * | 1998-03-16 | 2000-08-08 | Allelix Biopharmaceuticals Inc. | Pyrrolidine-indole compounds having 5-HT6 affinity |
US6251893B1 (en) * | 1998-06-15 | 2001-06-26 | Nps Allelix Corp. | Bicyclic piperidine and piperazine compounds having 5-HT6 receptor affinity |
GB9819035D0 (en) * | 1998-09-01 | 1998-10-28 | Cerebrus Res Ltd | Chemical compounds VII |
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CN107628981A (zh) * | 2017-10-31 | 2018-01-26 | 威海市妇女儿童医院 | 一种肉桂酰基吲哚啉化合物及其制备青光眼药物的应用 |
CN107628981B (zh) * | 2017-10-31 | 2019-07-30 | 威海市妇女儿童医院 | 一种肉桂酰基吲哚啉化合物及其制备青光眼药物的应用 |
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ZA200210234B (en) | 2004-03-18 |
IL154057A0 (en) | 2003-07-31 |
AU8273401A (en) | 2002-02-05 |
BR0112661A (pt) | 2003-06-24 |
KR100845450B1 (ko) | 2008-07-10 |
EA006604B1 (ru) | 2006-02-24 |
CN1443162A (zh) | 2003-09-17 |
AU2001282734B2 (en) | 2006-10-12 |
NZ523216A (en) | 2005-05-27 |
KR20030036599A (ko) | 2003-05-09 |
HUP0301346A2 (hu) | 2003-08-28 |
CA2411192A1 (en) | 2002-01-31 |
HK1057536A1 (en) | 2004-04-08 |
MXPA03000548A (es) | 2004-04-05 |
SE0002754D0 (sv) | 2000-07-21 |
HUP0301346A3 (en) | 2005-05-30 |
EA200300183A1 (ru) | 2003-08-28 |
JP2004504376A (ja) | 2004-02-12 |
PL360309A1 (en) | 2004-09-06 |
NO20030304L (no) | 2003-03-12 |
NO20030304D0 (no) | 2003-01-20 |
EP1301476A1 (en) | 2003-04-16 |
WO2002008178A1 (en) | 2002-01-31 |
YU2603A (sh) | 2006-05-25 |
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