CN120754111A - 用于治疗IgA肾病的包含布地奈德的药物组合物 - Google Patents

用于治疗IgA肾病的包含布地奈德的药物组合物

Info

Publication number
CN120754111A
CN120754111A CN202510929056.3A CN202510929056A CN120754111A CN 120754111 A CN120754111 A CN 120754111A CN 202510929056 A CN202510929056 A CN 202510929056A CN 120754111 A CN120754111 A CN 120754111A
Authority
CN
China
Prior art keywords
budesonide
composition
dissolution medium
dissolution
minutes
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN202510929056.3A
Other languages
English (en)
Chinese (zh)
Inventor
E·K·里塞尔
L·M·佩尔韦托夫-莫拉斯
K·桑德沃德
C·O·A·佩德森
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kalititas Treatment Co
Original Assignee
Kalititas Treatment Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=85076189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN120754111(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB2217146.6A external-priority patent/GB202217146D0/en
Priority claimed from GBGB2217150.8A external-priority patent/GB202217150D0/en
Application filed by Kalititas Treatment Co filed Critical Kalititas Treatment Co
Priority claimed from CN202380018644.0A external-priority patent/CN118591376A/zh
Publication of CN120754111A publication Critical patent/CN120754111A/zh
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4891Coated capsules; Multilayered drug free capsule shells
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CN202510929056.3A 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物 Pending CN120754111A (zh)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US202263302226P 2022-01-24 2022-01-24
US202263302216P 2022-01-24 2022-01-24
US63/302,216 2022-01-24
US63/302,226 2022-01-24
GB2217150.8 2022-11-16
GBGB2217146.6A GB202217146D0 (en) 2022-11-16 2022-11-16 New pharmaceutical compositions
GB2217146.6 2022-11-16
GBGB2217150.8A GB202217150D0 (en) 2022-11-16 2022-11-16 New pharmaceutical compositions
CN202380018644.0A CN118591376A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
PCT/EP2023/051680 WO2023139285A1 (en) 2022-01-24 2023-01-24 Pharmaceutical composition comprising budesonide for treating iga nephropathy

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CN202380018644.0A Division CN118591376A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物

Publications (1)

Publication Number Publication Date
CN120754111A true CN120754111A (zh) 2025-10-10

Family

ID=85076189

Family Applications (6)

Application Number Title Priority Date Filing Date
CN202510929056.3A Pending CN120754111A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202510935869.3A Pending CN120754112A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202510116905.3A Pending CN120053463A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202510943983.0A Pending CN120754113A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202610075373.8A Pending CN121796407A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202610075378.0A Pending CN121774982A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物

Family Applications After (5)

Application Number Title Priority Date Filing Date
CN202510935869.3A Pending CN120754112A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202510116905.3A Pending CN120053463A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202510943983.0A Pending CN120754113A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202610075373.8A Pending CN121796407A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物
CN202610075378.0A Pending CN121774982A (zh) 2022-01-24 2023-01-24 用于治疗IgA肾病的包含布地奈德的药物组合物

Country Status (14)

Country Link
US (10) US11896719B2 (enExample)
EP (1) EP4469060A1 (enExample)
JP (1) JP2025508321A (enExample)
KR (2) KR20250008979A (enExample)
CN (6) CN120754111A (enExample)
AU (1) AU2023210461A1 (enExample)
CA (1) CA3249575A1 (enExample)
CL (1) CL2024002201A1 (enExample)
CO (1) CO2024009565A2 (enExample)
GE (1) GEAP202416588A (enExample)
IL (1) IL314067A (enExample)
MX (1) MX2024009024A (enExample)
TW (2) TW202547520A (enExample)
WO (1) WO2023139285A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11896719B2 (en) 2022-01-24 2024-02-13 Calliditas Therapeutics Ab Pharmaceutical compositions

Citations (1)

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CN102088962A (zh) * 2008-05-12 2011-06-08 阿基米德开发有限公司 用于皮质类固醇口服给药的组合物

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Also Published As

Publication number Publication date
CA3249575A1 (en) 2023-07-27
US12311057B2 (en) 2025-05-27
US20250381146A1 (en) 2025-12-18
WO2023139285A1 (en) 2023-07-27
IL314067A (en) 2024-09-01
GEAP202416588A (en) 2024-11-25
US20250268835A1 (en) 2025-08-28
US11896719B2 (en) 2024-02-13
US20240173264A1 (en) 2024-05-30
TW202339765A (zh) 2023-10-16
TW202547520A (zh) 2025-12-16
AU2023210461A1 (en) 2024-07-18
US20250381147A1 (en) 2025-12-18
US12171883B2 (en) 2024-12-24
EP4469060A1 (en) 2024-12-04
CN120754113A (zh) 2025-10-10
US20240122863A1 (en) 2024-04-18
US20250255824A1 (en) 2025-08-14
US12171882B2 (en) 2024-12-24
JP2025508321A (ja) 2025-03-26
CN120053463A (zh) 2025-05-30
KR102919268B1 (ko) 2026-01-27
KR20240141771A (ko) 2024-09-27
KR20250008979A (ko) 2025-01-16
MX2024009024A (es) 2024-11-08
US20250312283A1 (en) 2025-10-09
TWI896928B (zh) 2025-09-11
US20250057775A1 (en) 2025-02-20
CN121774982A (zh) 2026-04-03
CL2024002201A1 (es) 2025-01-03
CO2024009565A2 (es) 2024-09-19
CN120754112A (zh) 2025-10-10
US20230293444A1 (en) 2023-09-21
US20250312282A1 (en) 2025-10-09
CN121796407A (zh) 2026-04-07

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