CN120661512A - 治疗克罗恩病和溃疡性结肠炎的方法 - Google Patents

治疗克罗恩病和溃疡性结肠炎的方法

Info

Publication number
CN120661512A
CN120661512A CN202510812764.9A CN202510812764A CN120661512A CN 120661512 A CN120661512 A CN 120661512A CN 202510812764 A CN202510812764 A CN 202510812764A CN 120661512 A CN120661512 A CN 120661512A
Authority
CN
China
Prior art keywords
weeks
patient
pharmaceutically acceptable
acceptable salt
tinib
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN202510812764.9A
Other languages
English (en)
Chinese (zh)
Inventor
R·B·萨卡
S·容格维尔特
A·P·马哈多德拉塞尔达
A·M·罗宾逊
J·J·V·埃内霍萨
A·L·潘根
M-E·穆罕默德
A·奥特曼
B·克吕恩德
A·D·阿利安
T·B·波尔查德特
F·L·诺尔斯特隆
A·Y·谢赫
M·M·马尔赫恩
J·加延特
P·J·马罗姆
P·T·迈尔
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AbbVie Inc
Original Assignee
AbbVie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=61750557&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN120661512(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by AbbVie Inc filed Critical AbbVie Inc
Publication of CN120661512A publication Critical patent/CN120661512A/zh
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CN202510812764.9A 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法 Pending CN120661512A (zh)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US201762469337P 2017-03-09 2017-03-09
US62/469337 2017-03-09
US201762470565P 2017-03-13 2017-03-13
US62/470565 2017-03-13
US201762483289P 2017-04-07 2017-04-07
US62/483289 2017-04-07
US201762593629P 2017-12-01 2017-12-01
US62/593629 2017-12-01
PCT/US2018/021800 WO2018165581A1 (en) 2017-03-09 2018-03-09 Methods of treating crohn's disease and ulcerative colitis
CN201880016862.XA CN110392572A (zh) 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CN201880016862.XA Division CN110392572A (zh) 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法

Publications (1)

Publication Number Publication Date
CN120661512A true CN120661512A (zh) 2025-09-19

Family

ID=61750557

Family Applications (2)

Application Number Title Priority Date Filing Date
CN202510812764.9A Pending CN120661512A (zh) 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法
CN201880016862.XA Pending CN110392572A (zh) 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN201880016862.XA Pending CN110392572A (zh) 2017-03-09 2018-03-09 治疗克罗恩病和溃疡性结肠炎的方法

Country Status (9)

Country Link
US (3) US20190046527A1 (https=)
EP (2) EP3592353A1 (https=)
JP (3) JP2020510016A (https=)
CN (2) CN120661512A (https=)
AU (2) AU2018230500B2 (https=)
BR (1) BR112019018576A2 (https=)
MX (2) MX2019010733A (https=)
TW (2) TWI851536B (https=)
WO (2) WO2018165581A1 (https=)

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CN114206878B (zh) 2020-07-08 2024-04-19 苏州科睿思制药有限公司 乌帕替尼的晶型及其制备方法和用途
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CN114380837B (zh) * 2021-12-27 2023-06-30 上海邈金医药科技有限公司 一种具有Janus激酶抑制活性的化合物、包括该化合物的组合物及其应用
MX2024008557A (es) * 2022-01-13 2024-09-11 Abbvie Inc Método de administración de upadacitinib para evitar interacciones farmacologicas y efectos adversos.
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Also Published As

Publication number Publication date
WO2018165581A1 (en) 2018-09-13
TW201840318A (zh) 2018-11-16
US20220233527A1 (en) 2022-07-28
CN110392572A (zh) 2019-10-29
WO2022178492A1 (en) 2022-08-25
US20210361647A1 (en) 2021-11-25
EP4487908A2 (en) 2025-01-08
JP2024009963A (ja) 2024-01-23
JP2026041823A (ja) 2026-03-10
AU2018230500A1 (en) 2019-09-19
US11607411B2 (en) 2023-03-21
TW202517269A (zh) 2025-05-01
AU2018230500B2 (en) 2024-03-07
EP3592353A1 (en) 2020-01-15
MX2022015499A (es) 2023-01-24
AU2024203642A1 (en) 2024-06-20
TWI851536B (zh) 2024-08-11
AU2024203642B2 (en) 2025-08-21
JP2020510016A (ja) 2020-04-02
CA3052873A1 (en) 2018-09-13
BR112019018576A2 (pt) 2020-04-14
EP4487908A3 (en) 2025-01-15
MX2019010733A (es) 2019-11-01
US20190046527A1 (en) 2019-02-14

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