CN115916744A - 一种稠合三环γ-氨基酸衍生物的缓释药物制剂及其制备方法 - Google Patents
一种稠合三环γ-氨基酸衍生物的缓释药物制剂及其制备方法 Download PDFInfo
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- Inorganic Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
公开了一种稠合三环γ‑氨基酸衍生物的缓释药物制剂及其制备方法。所述稠合三环γ‑氨基酸衍生物为式(I)所示的化合物或者其立体异构体、溶剂化物、前药、代谢产物、药学上可接受的盐或共晶。
Description
PCT国内申请，说明书已公开。
Claims (27)
- PCT国内申请，权利要求书已公开。
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202010695946X | 2020-07-20 | ||
| CN202010695946 | 2020-07-20 | ||
| PCT/CN2021/107286 WO2022017364A1 (zh) | 2020-07-20 | 2021-07-20 | 一种稠合三环γ-氨基酸衍生物的缓释药物制剂及其制备方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN115916744A true CN115916744A (zh) | 2023-04-04 |
Family
ID=79728995
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202180043436.7A Pending CN115916744A (zh) | 2020-07-20 | 2021-07-20 | 一种稠合三环γ-氨基酸衍生物的缓释药物制剂及其制备方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20230320989A1 (zh) |
| EP (1) | EP4183771A4 (zh) |
| JP (1) | JP2023534548A (zh) |
| CN (1) | CN115916744A (zh) |
| TW (1) | TW202214223A (zh) |
| WO (1) | WO2022017364A1 (zh) |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018050046A1 (zh) * | 2016-09-14 | 2018-03-22 | 四川海思科制药有限公司 | 稠合三环γ-氨基酸衍生物及其制备方法和在医药上的应用 |
| WO2019238068A1 (zh) * | 2018-06-13 | 2019-12-19 | 北京泰德制药股份有限公司 | 一种普瑞巴林缓释组合物及其制备方法 |
| WO2020011257A1 (zh) * | 2018-07-12 | 2020-01-16 | 四川海思科制药有限公司 | 一种稠合三环γ-氨基酸衍生物的组合物及其制备 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101120929A (zh) * | 2006-08-07 | 2008-02-13 | 珠海天翼医药技术开发有限公司 | 一种加巴喷丁胃滞留缓释组合物 |
| CN104352460A (zh) * | 2014-10-21 | 2015-02-18 | 齐宏 | 一种加巴喷丁片剂及其制备方法 |
| CN106606495A (zh) * | 2015-10-27 | 2017-05-03 | 四川海思科制药有限公司 | 一种普瑞巴林缓释片药物组合物及其制备方法 |
| WO2017107907A1 (zh) * | 2015-12-25 | 2017-06-29 | 四川海思科制药有限公司 | 稠合环γ-氨基酸衍生物及其制备方法和在医药上的应用 |
| CN106928080B (zh) * | 2015-12-31 | 2020-12-25 | 四川海思科制药有限公司 | 稠合环γ-氨基酸衍生物及其制备方法和在医药上的应用 |
| CN107848952B (zh) * | 2015-12-31 | 2021-04-09 | 四川海思科制药有限公司 | 稠合三环γ-氨基酸衍生物及其制备方法和在医药上的应用 |
| CN111053749B (zh) * | 2018-10-16 | 2022-07-15 | 北京泰德制药股份有限公司 | 一种普瑞巴林缓释组合物及其制备方法 |
| CN111918859B (zh) | 2018-07-12 | 2023-06-30 | 四川海思科制药有限公司 | 稠合三环γ-氨基酸衍生物的盐的晶型及制备和应用 |
| CN112384493B (zh) * | 2018-08-09 | 2023-06-06 | 四川海思科制药有限公司 | 稠合三环γ-氨基酸衍生物的制备方法及中间体 |
-
2021
- 2021-07-20 TW TW110126565A patent/TW202214223A/zh unknown
- 2021-07-20 US US18/006,255 patent/US20230320989A1/en active Pending
- 2021-07-20 CN CN202180043436.7A patent/CN115916744A/zh active Pending
- 2021-07-20 JP JP2023504131A patent/JP2023534548A/ja active Pending
- 2021-07-20 EP EP21845576.4A patent/EP4183771A4/en active Pending
- 2021-07-20 WO PCT/CN2021/107286 patent/WO2022017364A1/zh unknown
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018050046A1 (zh) * | 2016-09-14 | 2018-03-22 | 四川海思科制药有限公司 | 稠合三环γ-氨基酸衍生物及其制备方法和在医药上的应用 |
| WO2019238068A1 (zh) * | 2018-06-13 | 2019-12-19 | 北京泰德制药股份有限公司 | 一种普瑞巴林缓释组合物及其制备方法 |
| WO2020011257A1 (zh) * | 2018-07-12 | 2020-01-16 | 四川海思科制药有限公司 | 一种稠合三环γ-氨基酸衍生物的组合物及其制备 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4183771A1 (en) | 2023-05-24 |
| US20230320989A1 (en) | 2023-10-12 |
| TW202214223A (zh) | 2022-04-16 |
| JP2023534548A (ja) | 2023-08-09 |
| EP4183771A4 (en) | 2024-04-24 |
| WO2022017364A1 (zh) | 2022-01-27 |
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