CN113271938A - Tyk2抑制剂和其用途 - Google Patents

Tyk2抑制剂和其用途 Download PDF

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Publication number
CN113271938A
CN113271938A CN201980087661.3A CN201980087661A CN113271938A CN 113271938 A CN113271938 A CN 113271938A CN 201980087661 A CN201980087661 A CN 201980087661A CN 113271938 A CN113271938 A CN 113271938A
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CN
China
Prior art keywords
compound
nitrogen
sulfur
oxygen
independently selected
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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CN201980087661.3A
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English (en)
Chinese (zh)
Inventor
J·R·葛林伍德
C·E·玛斯
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
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Nimbus Lakshmi Inc
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Filing date
Publication date
Application filed by Nimbus Lakshmi Inc filed Critical Nimbus Lakshmi Inc
Publication of CN113271938A publication Critical patent/CN113271938A/zh
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CN201980087661.3A 2018-11-30 2019-11-27 Tyk2抑制剂和其用途 Pending CN113271938A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862773620P 2018-11-30 2018-11-30
US62/773,620 2018-11-30
PCT/US2019/063510 WO2020112937A1 (en) 2018-11-30 2019-11-27 Tyk2 inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
CN113271938A true CN113271938A (zh) 2021-08-17

Family

ID=70848642

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201980087661.3A Pending CN113271938A (zh) 2018-11-30 2019-11-27 Tyk2抑制剂和其用途

Country Status (8)

Country Link
US (2) US11053241B2 (https=)
EP (1) EP3886843A4 (https=)
JP (3) JP7530360B2 (https=)
CN (1) CN113271938A (https=)
AU (1) AU2019389025B2 (https=)
CA (1) CA3120866A1 (https=)
IL (1) IL283409B1 (https=)
WO (1) WO2020112937A1 (https=)

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CN117342955A (zh) * 2023-10-08 2024-01-05 盐城师范学院 一种制备4’-甲基-联苯-2-胺的方法

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TW202425965A (zh) * 2022-09-30 2024-07-01 日商科研製藥股份有限公司 縮環化合物及含有其之醫藥
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Publication number Priority date Publication date Assignee Title
US20180037570A1 (en) * 2016-08-08 2018-02-08 Merck Patent Gmbh Tlr7/8 antagonists and uses thereof
WO2018071794A1 (en) * 2016-10-14 2018-04-19 Nimbus Lakshmi, Inc. Tyk2 inhibitors and uses thereof
WO2018089695A1 (en) * 2016-11-11 2018-05-17 Dynavax Technologies Corporation Toll-like receptor antagonist compounds and methods of use

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117342955A (zh) * 2023-10-08 2024-01-05 盐城师范学院 一种制备4’-甲基-联苯-2-胺的方法

Also Published As

Publication number Publication date
JP7530360B2 (ja) 2024-08-07
EP3886843A4 (en) 2022-08-31
IL283409A (en) 2021-07-29
IL283409B1 (en) 2026-03-01
AU2019389025B2 (en) 2025-07-24
US11834449B2 (en) 2023-12-05
CA3120866A1 (en) 2020-06-04
JP2026053668A (ja) 2026-03-25
AU2019389025A1 (en) 2021-06-17
US11053241B2 (en) 2021-07-06
EP3886843A1 (en) 2021-10-06
US20220106306A1 (en) 2022-04-07
JP2022509260A (ja) 2022-01-20
WO2020112937A1 (en) 2020-06-04
US20200172540A1 (en) 2020-06-04
JP2024160253A (ja) 2024-11-13

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Effective date of registration: 20231129

Address after: Osaka, Japan

Applicant after: TAKEDA PHARMACEUTICAL Co.,Ltd.

Address before: Massachusetts

Applicant before: NIMBUS LAKSHMI, Inc.

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