JP7530360B2 - Ｔｙｋ２阻害剤およびその使用 - Google Patents

Ｔｙｋ２阻害剤およびその使用 Download PDF

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Publication number
JP7530360B2
JP7530360B2 JP2021530887A JP2021530887A JP7530360B2 JP 7530360 B2 JP7530360 B2 JP 7530360B2 JP 2021530887 A JP2021530887 A JP 2021530887A JP 2021530887 A JP2021530887 A JP 2021530887A JP 7530360 B2 JP7530360 B2 JP 7530360B2
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nitrogen
compound
sulfur
oxygen
independently selected
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Japanese (ja)
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JP2022509260A (ja
JP2022509260A5 (https=
Inventor
ジェレミー ロバート グリーンウッド，
クレッグ イー． マッセ，
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Takeda Pharmaceutical Co Ltd
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Takeda Pharmaceutical Co Ltd
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Priority to JP2025283785A priority patent/JP2026053668A/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2021530887A 2018-11-30 2019-11-27 Ｔｙｋ２阻害剤およびその使用 Active JP7530360B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2024120957A JP2024160253A (ja) 2018-11-30 2024-07-26 Ｔｙｋ２阻害剤およびその使用
JP2025283785A JP2026053668A (ja) 2018-11-30 2025-12-26 Ｔｙｋ２阻害剤およびその使用

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862773620P 2018-11-30 2018-11-30
US62/773,620 2018-11-30
PCT/US2019/063510 WO2020112937A1 (en) 2018-11-30 2019-11-27 Tyk2 inhibitors and uses thereof

Related Child Applications (1)

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JP2024120957A Division JP2024160253A (ja) 2018-11-30 2024-07-26 Ｔｙｋ２阻害剤およびその使用

Publications (3)

Publication Number Publication Date
JP2022509260A JP2022509260A (ja) 2022-01-20
JP2022509260A5 JP2022509260A5 (https=) 2022-12-05
JP7530360B2 true JP7530360B2 (ja) 2024-08-07

Family

ID=70848642

Family Applications (3)

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JP2021530887A Active JP7530360B2 (ja) 2018-11-30 2019-11-27 Ｔｙｋ２阻害剤およびその使用
JP2024120957A Pending JP2024160253A (ja) 2018-11-30 2024-07-26 Ｔｙｋ２阻害剤およびその使用
JP2025283785A Pending JP2026053668A (ja) 2018-11-30 2025-12-26 Ｔｙｋ２阻害剤およびその使用

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2024120957A Pending JP2024160253A (ja) 2018-11-30 2024-07-26 Ｔｙｋ２阻害剤およびその使用
JP2025283785A Pending JP2026053668A (ja) 2018-11-30 2025-12-26 Ｔｙｋ２阻害剤およびその使用

Country Status (8)

Country Link
US (2) US11053241B2 (https=)
EP (1) EP3886843A4 (https=)
JP (3) JP7530360B2 (https=)
CN (1) CN113271938A (https=)
AU (1) AU2019389025B2 (https=)
CA (1) CA3120866A1 (https=)
IL (1) IL283409B1 (https=)
WO (1) WO2020112937A1 (https=)

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TWI707852B (zh) 2015-09-02 2020-10-21 美商林伯士拉克許米公司 Tyk2 抑制劑及其用途
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CN113271940A (zh) 2018-10-15 2021-08-17 林伯士拉克许米公司 Tyk2抑制剂和其用途
CA3120866A1 (en) 2018-11-30 2020-06-04 Nimbus Lakshmi, Inc. Tyk2 inhibitors and uses thereof
JP2024501507A (ja) * 2020-12-25 2024-01-12 スーチュアン ハイスーク ファーマシューティカル カンパニー リミテッド ケトヘキソキナーゼ阻害剤及びその用途
CA3213816A1 (en) 2021-03-16 2022-09-22 Anrui Biomedical Technology (Guangzhou) Co., Ltd. Amino heteroaryl compounds and compositions
EP4423086A1 (en) 2021-10-25 2024-09-04 Kymera Therapeutics, Inc. Tyk2 degraders and uses thereof
TW202425965A (zh) * 2022-09-30 2024-07-01 日商科研製藥股份有限公司 縮環化合物及含有其之醫藥
CN115974751A (zh) * 2022-12-13 2023-04-18 山东能源集团新材料有限公司 一种吡拉西坦制备方法及系统
CN120752237A (zh) * 2022-12-22 2025-10-03 普罗泰克特治疗有限公司 吡咯并吡啶和吡咯并哒嗪类化合物及其作为pkr抑制剂的用途
WO2025010294A2 (en) * 2023-07-03 2025-01-09 Blossomhill Therapeutics, Inc. Macrocyclic compounds and use as tyk2 inhibitors
US11891394B1 (en) 2023-09-06 2024-02-06 King Faisal University Pyrrolo[2,3-c][1,6]naphthyridine-8-carboxylic acid compounds as CK2 inhibitors
US11878978B1 (en) 2023-09-06 2024-01-23 King Faisal University Pyrrolo[2,3-c]quinoline compounds as CK2 inhibitors
US11858935B1 (en) 2023-09-06 2024-01-02 King Faisal University Pyrrolo[2,3-c][1,7]naphthyridine-2-carboxylic acid compounds as CK2 inhibitors
CN117342955A (zh) * 2023-10-08 2024-01-05 盐城师范学院 一种制备4’-甲基-联苯-2-胺的方法
WO2025222103A1 (en) * 2024-04-19 2025-10-23 Raythera, Inc. Stat6 modulators and methods of uses thereof
WO2025264818A1 (en) * 2024-06-20 2025-12-26 Raythera, Inc. Stat6 modulators and methods of uses thereof

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WO2006011670A1 (ja) 2004-07-28 2006-02-02 Takeda Pharmaceutical Company Limited ピロロ［２，３－ｃ］ピリジン化合物、その製造方法および用途
JP2017514838A (ja) 2014-05-01 2017-06-08 ノバルティス アーゲー Ｔｏｌｌ様受容体７アゴニストとしての化合物および組成物
WO2018031434A1 (en) 2016-08-08 2018-02-15 Merck Patent Gmbh Tlr7/8 antagonists and uses thereof
WO2018089695A1 (en) 2016-11-11 2018-05-17 Dynavax Technologies Corporation Toll-like receptor antagonist compounds and methods of use

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JP2001512729A (ja) 1997-08-05 2001-08-28 ファイザー・プロダクツ・インク 神経ペプチドＹ受容体アンタゴニストとしての４−アミノピロ−ル（３，２−ｄ）ピリミジン
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JP2017514838A (ja) 2014-05-01 2017-06-08 ノバルティス アーゲー Ｔｏｌｌ様受容体７アゴニストとしての化合物および組成物
WO2018031434A1 (en) 2016-08-08 2018-02-15 Merck Patent Gmbh Tlr7/8 antagonists and uses thereof
WO2018089695A1 (en) 2016-11-11 2018-05-17 Dynavax Technologies Corporation Toll-like receptor antagonist compounds and methods of use

Also Published As

Publication number Publication date
JP2026053668A (ja) 2026-03-25
JP2022509260A (ja) 2022-01-20
AU2019389025A1 (en) 2021-06-17
US11053241B2 (en) 2021-07-06
IL283409B1 (en) 2026-03-01
WO2020112937A1 (en) 2020-06-04
IL283409A (en) 2021-07-29
AU2019389025B2 (en) 2025-07-24
EP3886843A4 (en) 2022-08-31
US20200172540A1 (en) 2020-06-04
JP2024160253A (ja) 2024-11-13
US11834449B2 (en) 2023-12-05
CN113271938A (zh) 2021-08-17
US20220106306A1 (en) 2022-04-07
EP3886843A1 (en) 2021-10-06
CA3120866A1 (en) 2020-06-04

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