CN110072539A - 抗微生物肽 - Google Patents
抗微生物肽 Download PDFInfo
- Publication number
- CN110072539A CN110072539A CN201780076612.0A CN201780076612A CN110072539A CN 110072539 A CN110072539 A CN 110072539A CN 201780076612 A CN201780076612 A CN 201780076612A CN 110072539 A CN110072539 A CN 110072539A
- Authority
- CN
- China
- Prior art keywords
- alkyl
- aryl
- optionally
- heteroaryl
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662433567P | 2016-12-13 | 2016-12-13 | |
| US62/433,567 | 2016-12-13 | ||
| PCT/EP2017/082697 WO2018109042A2 (en) | 2016-12-13 | 2017-12-13 | Antimicrobial peptides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN110072539A true CN110072539A (zh) | 2019-07-30 |
Family
ID=60788591
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201780076612.0A Pending CN110072539A (zh) | 2016-12-13 | 2017-12-13 | 抗微生物肽 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20200216493A1 (es) |
| EP (1) | EP3554528A2 (es) |
| JP (1) | JP2020500943A (es) |
| KR (1) | KR20190093600A (es) |
| CN (1) | CN110072539A (es) |
| AR (1) | AR110514A1 (es) |
| AU (1) | AU2017375034A1 (es) |
| BR (1) | BR112019011010A2 (es) |
| CA (1) | CA3047043A1 (es) |
| MX (1) | MX2019006768A (es) |
| RU (1) | RU2019120181A (es) |
| TW (1) | TW201827415A (es) |
| WO (1) | WO2018109042A2 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017181179A1 (en) * | 2016-04-15 | 2017-10-19 | The Regents Of The University Of California | Antimicrobial compositions |
| KR20190126838A (ko) * | 2017-03-09 | 2019-11-12 | 유니버시티 오브 링컨 | 새로운 항생제 생성물 |
| JP2021510148A (ja) * | 2018-01-03 | 2021-04-15 | バーシテック リミテッドＶｅｒｓｉｔｅｃｈ Ｌｉｍｉｔｅｄ | 新規抗生物質およびその使用方法 |
| US20220273760A1 (en) * | 2019-07-24 | 2022-09-01 | Sunshine Lake Pharma Co., Ltd. | A teixobactin analogue and use thereof |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS50160492A (es) * | 1974-06-22 | 1975-12-25 | ||
| GB9724859D0 (en) * | 1997-11-26 | 1998-01-21 | Univ Nottingham | Compounds and their use as antibacterial agents |
| AU769791B2 (en) * | 1998-06-24 | 2004-02-05 | New York University | Novel Staphylococcus peptides for bacterial interference |
| CN102405053B (zh) * | 2009-01-06 | 2015-07-29 | C3剑股份有限公司 | 靶向抗微生物部分 |
| TW202138383A (zh) * | 2012-12-03 | 2021-10-16 | 美商諾維生物製藥有限公司 | 新穎縮肽及其用途 |
| US9605026B2 (en) * | 2013-01-19 | 2017-03-28 | New York University | Hydrogen-bond surrogate peptides and peptidomimetics for p53 reactivation |
| WO2017181179A1 (en) * | 2016-04-15 | 2017-10-19 | The Regents Of The University Of California | Antimicrobial compositions |
| CN106632604B (zh) * | 2016-12-22 | 2021-03-19 | 深圳先进技术研究院 | 一种Teixobactin类似物及其制备方法和应用 |
| CN107266531B (zh) * | 2017-07-28 | 2020-04-07 | 北京大学深圳研究生院 | Teixobactin及其制备方法 |
-
2017
- 2017-12-13 KR KR1020197018910A patent/KR20190093600A/ko unknown
- 2017-12-13 JP JP2019551749A patent/JP2020500943A/ja active Pending
- 2017-12-13 BR BR112019011010A patent/BR112019011010A2/pt not_active Application Discontinuation
- 2017-12-13 CN CN201780076612.0A patent/CN110072539A/zh active Pending
- 2017-12-13 AR ARP170103485A patent/AR110514A1/es unknown
- 2017-12-13 WO PCT/EP2017/082697 patent/WO2018109042A2/en unknown
- 2017-12-13 MX MX2019006768A patent/MX2019006768A/es unknown
- 2017-12-13 EP EP17818515.3A patent/EP3554528A2/en not_active Withdrawn
- 2017-12-13 TW TW106143830A patent/TW201827415A/zh unknown
- 2017-12-13 RU RU2019120181A patent/RU2019120181A/ru not_active Application Discontinuation
- 2017-12-13 CA CA3047043A patent/CA3047043A1/en not_active Abandoned
- 2017-12-13 AU AU2017375034A patent/AU2017375034A1/en not_active Abandoned
- 2017-12-13 US US16/468,900 patent/US20200216493A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| BR112019011010A2 (pt) | 2019-10-08 |
| MX2019006768A (es) | 2019-08-01 |
| WO2018109042A3 (en) | 2018-07-26 |
| JP2020500943A (ja) | 2020-01-16 |
| EP3554528A2 (en) | 2019-10-23 |
| US20200216493A1 (en) | 2020-07-09 |
| AR110514A1 (es) | 2019-04-03 |
| KR20190093600A (ko) | 2019-08-09 |
| RU2019120181A (ru) | 2021-01-18 |
| AU2017375034A1 (en) | 2019-06-13 |
| CA3047043A1 (en) | 2018-06-21 |
| TW201827415A (zh) | 2018-08-01 |
| WO2018109042A2 (en) | 2018-06-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PB01 | Publication | ||
| PB01 | Publication | ||
| WD01 | Invention patent application deemed withdrawn after publication |
Application publication date: 20190730 |
|
| WD01 | Invention patent application deemed withdrawn after publication |