CN107007546A - 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物 - Google Patents

用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物 Download PDF

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Publication number
CN107007546A
CN107007546A CN201710280045.2A CN201710280045A CN107007546A CN 107007546 A CN107007546 A CN 107007546A CN 201710280045 A CN201710280045 A CN 201710280045A CN 107007546 A CN107007546 A CN 107007546A
Authority
CN
China
Prior art keywords
cream
oxymetazoline
weight
skin
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN201710280045.2A
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English (en)
Chinese (zh)
Inventor
S·D·尚勒
C·鲍威勒
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EPI Health LLC
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of CN107007546A publication Critical patent/CN107007546A/zh
Pending legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4174—Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Media Introduction/Drainage Providing Device (AREA)
CN201710280045.2A 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物 Pending CN107007546A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161443210P 2011-02-15 2011-02-15
US61/443,210 2011-02-15
CN2012800179627A CN103458897A (zh) 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CN2012800179627A Division CN103458897A (zh) 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物

Publications (1)

Publication Number Publication Date
CN107007546A true CN107007546A (zh) 2017-08-04

Family

ID=45757218

Family Applications (2)

Application Number Title Priority Date Filing Date
CN201710280045.2A Pending CN107007546A (zh) 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物
CN2012800179627A Pending CN103458897A (zh) 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN2012800179627A Pending CN103458897A (zh) 2011-02-15 2012-02-14 用于治疗红斑痤疮的症状的羟甲唑啉药物乳膏组合物

Country Status (11)

Country Link
US (4) US20120208858A1 (enExample)
EP (2) EP3578178A1 (enExample)
JP (3) JP6225030B2 (enExample)
KR (2) KR20190114010A (enExample)
CN (2) CN107007546A (enExample)
AU (3) AU2012217858A1 (enExample)
BR (1) BR112013020770A2 (enExample)
CA (1) CA2827373C (enExample)
ES (1) ES2742273T3 (enExample)
RU (1) RU2648439C2 (enExample)
WO (1) WO2012112566A1 (enExample)

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AU2019390704A1 (en) * 2018-11-26 2021-06-03 Cellix Bio Private Limited Ophthalmic compositions and methods for the treatment of skin diseases and eye diseases
EP3964212A4 (en) * 2019-04-30 2023-01-04 Generos Biopharma Ltd. COMPOUND FOR THE TREATMENT OF INFLAMMATORY AUTOIMMUNEAL DISEASES AND USE THEREOF
CN115368310B (zh) 2021-05-18 2025-06-27 奥库菲尔医药公司 合成甲磺酸酚妥拉明的方法
KR102633256B1 (ko) * 2021-10-08 2024-02-05 (주)우리스마트바이오 참당귀 추출물을 이용한 피부개선용 화장품 조성물, 이를 포함한 피부개선용 화장품 및 피부개선용 화장품 제조방법
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Also Published As

Publication number Publication date
AU2019203993A1 (en) 2019-06-27
CA2827373C (en) 2019-05-14
US11541000B2 (en) 2023-01-03
RU2648439C2 (ru) 2018-03-26
CA2827373A1 (en) 2012-08-23
BR112013020770A2 (pt) 2019-08-27
AU2019203993B2 (en) 2020-05-28
ES2742273T3 (es) 2020-02-13
US20190167566A1 (en) 2019-06-06
KR20140020912A (ko) 2014-02-19
EP2675449B1 (en) 2019-04-24
JP6225030B2 (ja) 2017-11-01
AU2017202726A1 (en) 2017-05-18
AU2017202726B2 (en) 2019-03-07
EP2675449A1 (en) 2013-12-25
US20200276108A1 (en) 2020-09-03
JP2014505733A (ja) 2014-03-06
EP3578178A1 (en) 2019-12-11
CN103458897A (zh) 2013-12-18
US20120208858A1 (en) 2012-08-16
KR102058756B1 (ko) 2020-01-22
US20140113947A1 (en) 2014-04-24
JP2018193399A (ja) 2018-12-06
JP2017066162A (ja) 2017-04-06
JP6389534B2 (ja) 2018-09-12
AU2012217858A1 (en) 2013-09-05
WO2012112566A1 (en) 2012-08-23
KR20190114010A (ko) 2019-10-08
RU2013141845A (ru) 2015-03-27

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Effective date of registration: 20190403

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Applicant before: ALLERGAN, Inc.

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Application publication date: 20170804