CN105960239A - 利用含有噻吩并三唑并二氮杂*化合物的药物制剂治疗白血病的方法 - Google Patents

利用含有噻吩并三唑并二氮杂*化合物的药物制剂治疗白血病的方法 Download PDF

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Publication number
CN105960239A
CN105960239A CN201480065213.0A CN201480065213A CN105960239A CN 105960239 A CN105960239 A CN 105960239A CN 201480065213 A CN201480065213 A CN 201480065213A CN 105960239 A CN105960239 A CN 105960239A
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compound
thienotriazolodiazepine
formula
solid dispersion
carbons
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CN201480065213.0A
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Chinese (zh)
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马里亚·E·里韦罗
埃里克·雷蒙德
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Oncoethix GmbH
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Oncoethix GmbH
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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CN201480065213.0A 2013-11-27 2014-11-26 利用含有噻吩并三唑并二氮杂*化合物的药物制剂治疗白血病的方法 Pending CN105960239A (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201361909702P 2013-11-27 2013-11-27
US61/909,702 2013-11-27
US201462012128P 2014-06-13 2014-06-13
US62/012,128 2014-06-13
US201462080804P 2014-11-17 2014-11-17
US62/080,804 2014-11-17
PCT/EP2014/075709 WO2015078929A1 (en) 2013-11-27 2014-11-26 Method of treating leukemia using pharmaceutical formulation containing thienotriazolodiazepine compounds

Publications (1)

Publication Number Publication Date
CN105960239A true CN105960239A (zh) 2016-09-21

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CN201480065213.0A Pending CN105960239A (zh) 2013-11-27 2014-11-26 利用含有噻吩并三唑并二氮杂*化合物的药物制剂治疗白血病的方法

Country Status (6)

Country Link
US (1) US9757385B2 (enExample)
EP (1) EP3074018A1 (enExample)
JP (1) JP2016538310A (enExample)
KR (1) KR20160079823A (enExample)
CN (1) CN105960239A (enExample)
WO (1) WO2015078929A1 (enExample)

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CN108743591A (zh) * 2018-07-17 2018-11-06 苏州大学 用于治疗癌症的药物组合物及其应用
CN116098870A (zh) * 2023-04-10 2023-05-12 上海赛默罗生物科技有限公司 α5-GABAA受体调节剂的固体分散体及其制备方法

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EP3137086A4 (en) * 2014-05-02 2017-12-27 Oncoethix GmbH Method of treating resistant non-hodgkin lymphoma, medulloblastoma, and/or alk+non-small cell lung cancer using thienotriazolodiazepine compounds
EP3185871A1 (en) * 2014-08-28 2017-07-05 Oncoethix GmbH Methods of treating acute myeloid leukemia or acute lymphoid leukemia using pharmaceutical compositions containing thienotriazolodiazepine compounds
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JP6885629B2 (ja) 2016-07-29 2021-06-16 オンターナル セラピューティック インコーポレイテッドＯｎｃｔｅｒｎａｌ Ｔｈｅｒａｐｅｕｔｉｃｓ， Ｉｎｃ． インドリノン化合物の使用
CN110099685A (zh) * 2016-10-20 2019-08-06 赛尔基因光迪斯研究公司 溴结构域抑制剂
EA202092635A1 (ru) 2018-06-13 2021-03-23 Дибли Аг Получение конденсированных производных триазепина и их применение в качестве ингибиторов bet
US12162870B2 (en) 2021-06-08 2024-12-10 The Regents Of The University Of California Anticancer compounds
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