CN105566291B - 制备甲磺酸伊马替尼晶型的方法 - Google Patents
制备甲磺酸伊马替尼晶型的方法 Download PDFInfo
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- CN105566291B CN105566291B CN201610077381.2A CN201610077381A CN105566291B CN 105566291 B CN105566291 B CN 105566291B CN 201610077381 A CN201610077381 A CN 201610077381A CN 105566291 B CN105566291 B CN 105566291B
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/42—Separation; Purification; Stabilisation; Use of additives
- C07C303/44—Separation; Purification
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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CN201610077381.2A CN105566291B (zh) | 2016-02-02 | 2016-02-02 | 制备甲磺酸伊马替尼晶型的方法 |
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CN201610077381.2A CN105566291B (zh) | 2016-02-02 | 2016-02-02 | 制备甲磺酸伊马替尼晶型的方法 |
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CN105566291A CN105566291A (zh) | 2016-05-11 |
CN105566291B true CN105566291B (zh) | 2018-06-01 |
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Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102250063A (zh) * | 2010-05-19 | 2011-11-23 | 江苏豪森药业股份有限公司 | 甲磺酸伊马替尼的晶型及其制备方法 |
CN102633775A (zh) * | 2012-04-06 | 2012-08-15 | 江南大学 | 一种甲磺酸伊马替尼α晶型的制备方法 |
CN104817536A (zh) * | 2015-04-14 | 2015-08-05 | 江苏豪森药业股份有限公司 | 适合药用的甲磺酸伊马替尼非针状α晶型及其制备方法 |
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- 2016-02-02 CN CN201610077381.2A patent/CN105566291B/zh active Active
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
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CN102250063A (zh) * | 2010-05-19 | 2011-11-23 | 江苏豪森药业股份有限公司 | 甲磺酸伊马替尼的晶型及其制备方法 |
CN102633775A (zh) * | 2012-04-06 | 2012-08-15 | 江南大学 | 一种甲磺酸伊马替尼α晶型的制备方法 |
CN104817536A (zh) * | 2015-04-14 | 2015-08-05 | 江苏豪森药业股份有限公司 | 适合药用的甲磺酸伊马替尼非针状α晶型及其制备方法 |
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TA01 | Transfer of patent application right |
Effective date of registration: 20170519 Address after: 222200 Guanyun City, Jiangsu province Lingang Industrial Zone, the south side of the weft Road, eight Applicant after: Lianyungang Hengyun Pharmaceutical Co. Ltd. Address before: 222200 Jiangsu city of Lianyungang province Guanyun County Harbor Industrial Zone weft seven road No. 1 Applicant before: LIANYUNGANG HENGYUN MEDICAL TECHNOLOGY CO., LTD. |
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Address after: 222200 Guanyun City, Jiangsu province Lingang Industrial Zone, the south side of the weft Road, eight Applicant after: Lianyungang Hengyun Pharmaceutical Co. Ltd. Address before: 222200 Guanyun City, Jiangsu province Lingang Industrial Zone, the south side of the weft Road, eight Applicant before: Lianyungang Hengyun Pharmaceutical Co. Ltd. |
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