CN105377821A - 酪氨酸激酶抑制剂及其盐的晶体形式 - Google Patents
酪氨酸激酶抑制剂及其盐的晶体形式 Download PDFInfo
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- C07—ORGANIC CHEMISTRY
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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Landscapes
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Applications Claiming Priority (3)
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| US61/801,112 | 2013-03-15 | ||
| PCT/US2014/027591 WO2014152663A1 (en) | 2013-03-15 | 2014-03-14 | Crystalline forms of tyrosine kinase inhibitors and their salts |
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| CN105377821A true CN105377821A (zh) | 2016-03-02 |
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| JP5752601B2 (ja) | 2008-12-08 | 2015-07-22 | ブイエム ファーマ エルエルシー | タンパク質受容体チロシンキナーゼ阻害薬の組成物 |
| US8999992B2 (en) * | 2013-03-15 | 2015-04-07 | Vm Pharma Llc | Crystalline forms of tryosine kinase inhibitors and their salts |
| AU2015318324A1 (en) | 2014-09-17 | 2017-04-06 | Mundipharma International Corporation Limited | Crystalline forms of tyrosine kinase inhibitors and their salts |
| US20180370926A1 (en) * | 2015-08-07 | 2018-12-27 | Purdue Pharma L.P. | Process of preparing tyrosine kinase inhibitor |
| KR102717072B1 (ko) | 2017-10-18 | 2024-10-15 | 인사이트 코포레이션 | Pi3k-감마 저해제로서의 3차 하이드록시기로 치환된 축합된 이미다졸 유도체 |
| WO2019159097A1 (en) * | 2018-02-14 | 2019-08-22 | Sun Pharmaceutical Industries Limited | Crystalline polymorphic forms of acalabrutinib |
| CR20250050A (es) | 2018-09-05 | 2025-03-19 | Incyte Corp | Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165) |
| US12240813B2 (en) | 2020-05-19 | 2025-03-04 | Cybin Irl Limited | Deuterated tryptamine derivatives and methods of use |
| WO2023168023A1 (en) | 2022-03-04 | 2023-09-07 | Reset Pharmaceuticals, Inc. | Co-crystals or salts comprising psilocin |
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| CN102292338A (zh) * | 2008-12-08 | 2011-12-21 | Vm制药有限公司 | 酪氨酸激酶蛋白受体拮抗剂 |
| WO2012119079A1 (en) * | 2011-03-03 | 2012-09-07 | Indiana University Research And Technology Corporation | uPAR-uPA INTERACTION INHIBITORS AND METHODS FOR TREATING CANCER |
| US20150174124A1 (en) * | 2013-03-15 | 2015-06-25 | Vm Pharma Llc | Crystalline forms of tryosine kinase inhibitors and their salts |
| WO2016043975A1 (en) * | 2014-09-17 | 2016-03-24 | Vm Pharma Llc | Crystalline forms of tyrosine kinase inhibitors and their salts |
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2016
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Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102292338A (zh) * | 2008-12-08 | 2011-12-21 | Vm制药有限公司 | 酪氨酸激酶蛋白受体拮抗剂 |
| WO2012119079A1 (en) * | 2011-03-03 | 2012-09-07 | Indiana University Research And Technology Corporation | uPAR-uPA INTERACTION INHIBITORS AND METHODS FOR TREATING CANCER |
| US20150174124A1 (en) * | 2013-03-15 | 2015-06-25 | Vm Pharma Llc | Crystalline forms of tryosine kinase inhibitors and their salts |
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