CN104411301B - 适于改善运动障碍治疗的口服药物配方 - Google Patents

适于改善运动障碍治疗的口服药物配方 Download PDF

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CN104411301B
CN104411301B CN201380031301.4A CN201380031301A CN104411301B CN 104411301 B CN104411301 B CN 104411301B CN 201380031301 A CN201380031301 A CN 201380031301A CN 104411301 B CN104411301 B CN 104411301B
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pharmaceutical composition
activator
acceptor
ht1b
component
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CN104411301A (zh
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J·B·汉森
M·S·汤姆森
J·D·米克尔森
P·G·尼尔森
M·克瑞尔加德
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Psychology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CN201380031301.4A 2012-04-18 2013-04-18 适于改善运动障碍治疗的口服药物配方 Active CN104411301B (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
DKPA201270196 2012-04-18
DKPA201270196 2012-04-18
PCT/DK2012/050190 WO2012163365A1 (en) 2011-06-01 2012-06-01 Combinations of serotonin receptor agonists for treatment of movement disorders
DKPCT/DK2012/050190 2012-06-01
DKPA201270755 2012-12-04
DKPA201270755 2012-12-04
PCT/DK2013/050111 WO2013156035A1 (en) 2012-04-18 2013-04-18 Orally available pharmaceutical formulation suitable for improved management of movement disorders

Publications (2)

Publication Number Publication Date
CN104411301A CN104411301A (zh) 2015-03-11
CN104411301B true CN104411301B (zh) 2018-02-06

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US (1) US10561618B2 (enExample)
EP (1) EP2838517B1 (enExample)
JP (1) JP6216768B2 (enExample)
KR (1) KR102104635B1 (enExample)
CN (1) CN104411301B (enExample)
AU (1) AU2013248685B2 (enExample)
BR (1) BR112014025907B1 (enExample)
CA (1) CA2870123C (enExample)
DK (1) DK2838517T3 (enExample)
ES (1) ES2654787T3 (enExample)
HU (1) HUE037732T2 (enExample)
IL (1) IL235000B (enExample)
IN (1) IN2014DN09571A (enExample)
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MY (1) MY169068A (enExample)
NO (1) NO2838517T3 (enExample)
NZ (1) NZ700474A (enExample)
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PT (1) PT2838517T (enExample)
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PL3160464T3 (pl) * 2014-06-26 2018-12-31 Contera Pharma Aps 6-hydroksybuspiron do stosowania w leczeniu zaburzeń ruchowych
KR102533428B1 (ko) * 2014-07-09 2023-05-16 피에르 파브르 메디카먼트 베피라돌을 이용한 이상운동질환 치료 방법
BR112017015487A2 (pt) 2015-01-20 2018-01-30 Xoc Pharmaceuticals Inc Composto; composição; método de tratamento e/ou prevenção de enxaqueca, als, doença de alzheimer, doença de parkinson, distúrbios extrapirimidais, depressão, náusea, êmese, síndrome das pernas inquietas, insônia, agressão, doença de huntington, doença cardiopulmonar, fibrogênese, hipertensão arterial pulmonar, ansiedade, dependências a drogas, distonia, parassonia ou hiperlactinemia em um indivíduo; métodos de agonização dos receptores d2, 5-ht1d, 5-ht1a e 5-ht2c, em um indivíduo; método de antagonização do receptor d3 em um indivíduo; métodos de agonização seletiva dos receptores 5 -ht1d, e 5-ht2c, método de fornecimento de atividade de antagonista funcional no receptor 5 -ht2b ou no receptor 5-ht7, ou em ambos, em um indivíduo; método de fornecimento de atividade de antagonista funcional nos receptores adrenérgicos em um indivíduo
CA3064274A1 (en) 2017-06-01 2018-12-06 Xoc Pharmaceuticals, Inc. Ergoline derivatives for use in medicine
US11135379B2 (en) 2019-02-15 2021-10-05 Bn Intellectual Properties, Inc. Method of delivering pharmaceutical products
US10758535B1 (en) 2019-04-26 2020-09-01 Sumitomo Dainippon Pharma Co., Ltd. Therapeutic drug for dyskinesia
US11559525B2 (en) 2019-04-26 2023-01-24 Sumitomo Pharma Co., Ltd. Therapeutic drug for dyskinesia
US11364225B2 (en) * 2019-08-21 2022-06-21 Bn Intellectual Properties, Inc. Pharmaceutical formulation for treating symptoms of migraine and cluster headaches, and method of using the same
CN116113402A (zh) 2020-08-31 2023-05-12 住友制药株式会社 帕金森病的运动并发症治疗药
MX2023011240A (es) * 2021-03-25 2024-01-12 Maplight Therapeutics Inc Composiciones farmaceuticas que comprenden zolmitriptan.
WO2025164698A1 (ja) * 2024-01-31 2025-08-07 株式会社ケイファーマ ハンチントン病治療剤及び治療用組成物
CN118308475B (zh) * 2024-03-18 2024-11-26 安徽医科大学第一附属医院 Htr1b作为胚胎发育停滞的诊断标志物和治疗靶点方面的应用
EP4647069A1 (en) 2024-05-07 2025-11-12 Universita' Degli Studi Di Trieste Drugs and compositions for use in the treatment of rett syndrome

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CN101247795A (zh) * 2005-04-06 2008-08-20 埃德莫斯药品有限公司 用于治疗与中枢神经系统（cns）相关疾病的方法和组合物
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