CN104306701A - 化瘀调脂汤 - Google Patents

化瘀调脂汤 Download PDF

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CN104306701A
CN104306701A CN201410528801.5A CN201410528801A CN104306701A CN 104306701 A CN104306701 A CN 104306701A CN 201410528801 A CN201410528801 A CN 201410528801A CN 104306701 A CN104306701 A CN 104306701A
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周峻
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Abstract

本发明公开了一种化瘀调脂汤,包含以下质量份的组分:丹参15,当归15,赤芍15,川芎15,制玉竹10,葛根15,生山楂15,制黄精15,荷叶15,熟地黄10,菊花10,赤芍15,怀牛膝15,枸杞子15,制何首乌10。本发明的化瘀调脂汤可以有效纠正脂代谢紊乱,降低血脂,同时具有降低血粘度的功效,并且对治疗脑梗死合并颈动脉粥样硬化斑块有较好的疗效。

Description

化瘀调脂汤
技术领域
本发明涉及一种重要汤剂,具体涉及一种化瘀调脂汤。
背景技术
脑梗死又称缺血性脑卒中,是中医的中风范畴,中风为中国四大顽症之首,为历代医家所重视。脑梗死好发与中老年人,为各类老年脑血管病发病之首,复发率、致残率和死亡率高,严重威胁着患者的健康和生存。传统中医学认为,中风是由于气血逆乱,长风风、火、痰、淤导致静脉阻塞。发病基础多为积损正衰、烦劳过度导致劳倦内伤,或兼脾失健运、痰浊内生,或兼五志所伤、情志过极,或兼外邪侵袭,痹阻经络。由于患者脏腑功能失调或气血素虚,加之劳倦内伤,忧思恼怒、饮酒饱食、用力过度,而致淤血阻滞,痰热内蕴;或阳化风动,血随气逆导致经脉痹阻引起一系列症状。
中国专利公开号CN103071124B,公告日2014.02.26的发明专利公开了一种治疗脑梗死的中药方剂,其有效成分原料由龙骨、狗骨、山羊角、水牛角、茺蔚子、莴苣子、郁金、柴胡、秦艽、山柰、苏合香、安息香、木香、乌梢蛇、金钱白花蛇、蕲蛇、蜈蚣、全蝎、附子、马钱子、天麻、当归、防风、地龙、水蛭、葛根、三七花、牛黄、琥珀、党参、人参、黄芪、甘草、三七、红花组成。
中医学认为,脑梗死合并颈动脉粥样硬化斑块形成多因肾虚肝亏,脾失健运,肝失疏泄, 膏粱厚味无以化生气血精微, 日久化痰生瘀, 附着血脉,脉络闭阻,属于本虚标实之证,本虚为脾失健运、肝肾亏虚,标实为痰浊血瘀。其中痰浊、血瘀疏泄转化不利,停滞于血脉之上是发病关键。故治以健脾益肾疏肝、 活血化瘀为主。针对其异常的病因病机,主要注重化瘀调脂并重,治疗应以健脾益肾疏肝、 活血化瘀中药为主,以达到化瘀调脂的作用,能够治病而不伤正气,祛瘀而不留邪。
发明内容
本发明所要解决的技术问题是提供一种化瘀调脂汤,它具有调整血脂、降低血液粘度的作用,对治疗脑梗死合并颈动脉粥样硬化斑块有较好的疗效。
为解决上述技术问题,本发明所采用的技术方案是:
一种化瘀调脂汤,其特征在于包含以下质量份的组分:丹参15,当归15,赤芍15,川芎15,制玉竹10,葛根15,生山楂15,制黄精15,荷叶15,熟地黄10,菊花10,赤芍15,怀牛膝15,枸杞子15,制何首乌10。
本发明与现有技术相比,具有以下优点和效果:化瘀调脂汤通过多环节、多途径、多靶点,可以有效纠正脂代谢紊乱,降低血脂,同时具有降低血粘度的功效。临床研究表明本方治疗脑梗死合并颈动脉粥样硬化斑块能明显改善及消除各种症状、调整血脂、改善血液动力学各项指标,疗效较好,可作为脑梗塞合并颈动脉粥样硬化斑块基础治疗的有效辅助药物,与单纯应用西药治疗相比可增强治疗效果、加快病情缓解,提高治疗的总有效率。
附图说明
图1是本发明的化瘀调脂汤的临床试验结果的两组临床疗效比较表。
图2是本发明的化瘀调脂汤的临床试验结果的两组患者治疗前后血脂变化比较表。
图3是本发明的化瘀调脂汤的临床试验结果的两组患者治疗前后血流变的变化比较表。
具体实施方式
下面结合附图并通过实施例对本发明作进一步的详细说明,以下实施例是对本发明的解释而本发明并不局限于以下实施例。
化瘀调脂汤组成成分:丹参15g,当归15g,赤芍15g,川芎15g,制玉竹10g,葛根15g,生山楂15g,制黄精15g,荷叶15g,熟地黄10g,菊花10g,赤芍15g,怀牛膝15g,枸杞子15g,制何首乌10g。制成汤剂。
化瘀调脂汤方剂解析, 方中山楂健脾消积;菊花、葛根、玉竹、荷叶清热疏肝;制黄精、熟地黄、枸杞子、何首乌滋补肝肾、固本培元;丹参、当归、赤芍、川芎、怀牛膝活血化瘀。诸药合用,共奏健脾消积、补肾疏肝、 活血化瘀之功效。
现代药理研究提示:丹参的提取物丹参素,可以抗氧化损伤,对氧化低密度脂蛋白损伤后内皮祖细胞的功能有显著保护作用 ;荷叶可使高脂饮食的兔血脂肪含量降低, 并有阻止脂类在血管内滞留或渗透到血管内壁的功能, 促进胆固醇的运输和清除的作用;山楂可以降低胆固醇、促进脂肪转化等, 其中的有效成分之一的山楂黄酮,对高脂血模型小鼠具有显著的降血清胆固醇、甘油三酯作用, 并发现山楂黄酮通过调控高脂血模型小鼠脂肪、肌肉组织中生脂基因转录表达,从而达到调血脂的作用。药理研究也证实,当归、赤芍、川芎、玉竹、葛根、制黄精、熟地黄等均有降TC、 TG的疗效,与本临床观察结果一致。
临床试验
所有患者均为桐乡市第二人民医院内科住院病人,住院时间为2011年3月至2013年6月,共入选123例,采用随机、单盲对照方法,分为两组,治疗组63例,男35例,女28例;年龄50~75岁,平均(62.8±4.7)岁。对照组60例,男33例,女27例;年龄49~76岁,平均(63.4土3.9)岁;两组患者性别、年龄以及治疗前血脂、血流变等经统计学分析,差异无统计学意义(P>0.05),具有可比性。
试验方法
1)  治疗方法
两组治疗前均予低盐低脂饮食,均给予抗血小板治疗(阿司匹林片100mg/d)、他汀类调脂(阿托伐他汀胶囊20mg/d)、控制血压及血糖在合理水平,对有合并症状者对症处理。治疗组除予正常西医治疗外,加用自拟化瘀调脂汤(组成:丹参15g、当归15g、赤芍15g、川芎15g、玉竹10g、葛根15g、山楂15g、制黄精15g、荷叶15g、熟地黄10g),结合患者病情,四诊合参,随证加减,并由我院制剂室煎药包装一副中药煎制两袋(150ml/袋),每次1袋,每日2次。对照组予以常规西医治疗,不予中药口服。两组均服药4周为1个疗程。
观察指标及方法
观察用药前后血总胆固醇(TC)、甘油三酯(TG)、低密度脂蛋白(LDL-C)、高密度脂蛋白(HDL-C)及血流变指标等。
3) 疗效判定标准
参照卫生部颁布的《中药新药临床研究指导原则》的疗效评定标准。治愈:临床症状基本消失,血脂及血流变均改善明显;显效:临床症状明显好转,血脂及(或)血流变有部分改善;有效:临床症状有好转,血脂及(或)血流变改善不明显;无效:治疗过程中出现急性心脑血管病及临床症状加重,血脂及(或)血流变改善不明显甚至加重。
4) 统计学方法
所有数据采用SPSS12.0软件处理。计量资料采用 ±S表示,两组间均数比较采用t检验、多组间均数比较采用方差分析,计数资料采用X2检验、列联表分析,以P<0.05为有统计学意义。
临床试验结果
两组临床疗效比较
治疗组治愈20例,占31.75%,显效25例,占39.68%,有效14例,占37.50%,无效4例,占6.35%,总有效率93.65%;对照组治愈10例,占16.67%,显效12例,占20.00%,有效27例,占45.00%,无效11例,占18.33%,总有效率81.67%;两组比较差异有统计学意义(P<0.05),见图1。
两组患者治疗前后血脂变化比较
治疗组TC、TG、 LDL-C较治疗前均有下降,其中TC、TG水平与治疗前比较差异均有统计学意义(P<0.05);治疗后两组间比较,治疗组TC、TG的水平较对照组明显下降(P<0.05),见图2。
两组患者治疗前后血流变的变化比较
治疗组全血低切粘度、血浆比黏度与治疗前比较差异均有统计学意义(P<0.05);且血浆比黏度优于对照组(P<0.05),见图3。
不良反应
治疗过程中及治疗后随诊,治疗组未见过敏反应,头颅CT复查均无脑出血;治疗前后肝肾功能、血清肌酸激酶及血、尿、大便常规检查均未见异常。对照组也未见不良反应。
综上所述, 化瘀调脂汤通过多环节、多途径、多靶点,可以有效纠正脂代谢紊乱,降低血脂,同时具有降低血粘度的功效。临床研究表明本方治疗脑梗死合并颈动脉粥样硬化斑块能明显改善及消除各种症状、调整血脂、改善血液动力学各项指标,疗效较好,可作为脑梗塞合并颈动脉粥样硬化斑块基础治疗的有效辅助药物,与单纯应用西药治疗相比可增强治疗效果、加快病情缓解,提高治疗的总有效率。
本说明书中所描述的以上内容仅仅是对本发明所作的举例说明。本发明所属技术领域的技术人员可以对所描述的具体实施例做各种各样的修改或补充或采用类似的方式替代,只要不偏离本发明说明书的内容或者超越本权利要求书所定义的范围,均应属于本发明的保护范围。

Claims (1)

1.一种化瘀调脂汤,其特征在于包含以下质量份的组分:丹参15,当归15,赤芍15,川芎15,制玉竹10,葛根15,生山楂15,制黄精15,荷叶15,熟地黄10,菊花10,赤芍15,怀牛膝15,枸杞子15,制何首乌10。
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