CN104271552B - 作为kappa阿片样物质受体(kor)激动剂的取代的杂环乙酰胺 - Google Patents

作为kappa阿片样物质受体(kor)激动剂的取代的杂环乙酰胺 Download PDF

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CN104271552B
CN104271552B CN201380023425.8A CN201380023425A CN104271552B CN 104271552 B CN104271552 B CN 104271552B CN 201380023425 A CN201380023425 A CN 201380023425A CN 104271552 B CN104271552 B CN 104271552B
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ethyl
hydroxypyrrolidin
methyl
oxo
acetamide
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CN104271552A (zh
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P.K.萨斯马
C.瓦姆塞克里斯纳
V.波特鲁里
A.特希姆
Y.盖
H.张
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Dr Reddys Laboratories Ltd
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    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CN201380023425.8A 2012-03-05 2013-03-05 作为kappa阿片样物质受体(kor)激动剂的取代的杂环乙酰胺 Expired - Fee Related CN104271552B (zh)

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US201261606632P 2012-03-05 2012-03-05
US61/606632 2012-03-05
PCT/CN2013/000230 WO2013131408A1 (en) 2012-03-05 2013-03-05 Substituted heterocyclic acetamides as kappa opioid receptor (kor) agonists

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Cited By (1)

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RU2776842C2 (ru) * 2017-12-06 2022-07-27 Цзянсу Хэнжуй Медсин Ко., Лтд. Применение агониста kor в комбинации с агонистом mor для получения лекарственного средства для лечения боли

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CN104271552B (zh) * 2012-03-05 2017-08-08 雷迪博士实验室有限公司 作为kappa阿片样物质受体(kor)激动剂的取代的杂环乙酰胺
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